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CAS 932973-77-8

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  • VU0514009

    CAS:
    VU0514009 is a competitive antagonist of chemokine-like receptor 1 (CMKLR1) with an EC50 of 2 nM. It effectively inhibits chemerin-9-induced arrestin recruitment and receptor internalization, significantly reducing Ca2+ flux responses in HEK293 cells. This compound shows potential for research in inflammatory diseases and metabolic syndrome.
    Fórmula:C21H20ClN3O5S2
    Forma y color:Solid
    Peso molecular:493.98