Enzimas inhibidoras
Los inhibidores enzimáticos son compuestos que disminuyen o detienen la actividad de las enzimas al unirse a ellas de manera específica. Estos inhibidores desempeñan un papel crucial en la regulación de procesos biológicos y se utilizan ampliamente en la investigación médica y el desarrollo de fármacos. Al bloquear la acción de las enzimas, permiten estudiar la función enzimática y desarrollar tratamientos contra diversas enfermedades. En CymitQuimica, ofrecemos una amplia gama de inhibidores enzimáticos de alta calidad para apoyar su investigación en biología y farmacología.
Se han encontrado 123 productos de "Enzimas inhibidoras"
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(R)-Pinocembrin
CAS:Producto controlado<p>Applications (2R)-Pinocembrin is the (R)-enantiomer of Pinocembrin, a flavanoid with antioxidant activity found in damiana, honey, and propolis. (2R)-Pinocembrin is a potential inhibitor of PIM1 kinase, an oncogene that has been implicated in the development of leukemias, lymphomas, and prostate cancer.<br>References Zhao, J. et al.: J. Ethnopharmacol., 120, 387 (2008); Holder, S. et al.: Mol. Cancer Ther., 6, 163 (2007); Holder, S. et al.: Bioorg. Med. Chem., 15, 6463 (2007);<br></p>Fórmula:C15H12O4Forma y color:WhitePeso molecular:256.25O,O-Dimethyl Dithiophosphate
CAS:Producto controladoFórmula:C2H7O2PS2Forma y color:ColourlessPeso molecular:158.18Morusin
CAS:Producto controlado<p>Stability Light Sensitive<br>Applications Morusin is an inhibitor of human cervical cancer stem cell growth, attenuating NF-kB activity, and initiating apoptosis.<br>References Wang, L. et al.: Mol. Cell. Biochem., 379, 7 (2013);<br></p>Fórmula:C25H24O6Forma y color:NeatPeso molecular:420.45GDC 0152
CAS:Producto controlado<p>Applications GDC 0152 is a peptidomimetic small molecule antagonist of inhibitor of apoptosis (IAP) proteins with antitumor activity.<br>References Yue, Q., et. al.: Drug Metab. Dispos., 41, 508 (2013)<br></p>Fórmula:C25H34N6O3SForma y color:NeatPeso molecular:498.643a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-diol
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications 3a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-diol, can be used in the synthesis of Hexosaminidase inhibitors, which are the new drug candidates for the therapy of osteoarthritis.<br>References Liu, J. et al.: Chem. Bio., 8, 701 (2001);<br></p>Fórmula:C8H13NO4SForma y color:White To Light BeigePeso molecular:219.26Bisindolylmaleimide VIII Acetic Acid Salt
CAS:Producto controlado<p>Applications It is a potent inhibitor of protein kinase C (PKC) activity. Bisindolylmaleimide VIII (Bis VIII) has been previously shown to enhance Fas-mediated apoptosis through a protein kinase C-independent mechanism.<br>References Emery, J., et al.: J. Biol. Chem., 273, 14363 (1998), Wiley, S., et al.: Immunity, 3, 673 (1995), MacFarlane, M., et al.: Biochem. J., 348, 93 (2000),<br></p>Fórmula:C26H26N4O4Forma y color:NeatPeso molecular:458.511-(5-Isoquinolinesulfonyl)-2-methylpiperazine Dihydrochloride
CAS:Producto controlado<p>Applications A selective inhibitor of protein kinase C or cyclic-nucleotide-dependent protein kinases.<br>References Hidaka, H. and Kawamoto, S.: Biochem. and Biophys. Res. Comm., 125, 1, 258 (1984)<br></p>Fórmula:C14H17N3O2S·2ClHForma y color:NeatPeso molecular:364.29O,S-Diethyl Methylphosphonothioate
CAS:Producto controlado<p>Stability Moisture Sensitive<br>Applications An inhibitor of cholinesterase.<br>References Berman, H., et al.: J. Biol. Chem., 264, 3951 (1989), Millard, C., et al.: Biochemistry, 37, 237 (1998), Koellner, G., et al.: J. Mol. Biol., 296, 713 (2000),<br></p>Fórmula:C5H13O2PSForma y color:NeatPeso molecular:168.193-Acetyl-11-keto-β-boswellic Acid
CAS:Producto controladoFórmula:C32H48O5Forma y color:WhitePeso molecular:512.721-Propan-1,1,2,2,3,3,3-d7-amine
CAS:Producto controladoFórmula:C3H2D7NForma y color:NeatPeso molecular:66.15O-(2,4-Dinitrophenyl)hydroxylamine
CAS:<p>Applications O-(2,4-Dinitrophenyl)hydroxylamine is a rapid active-site-directed inhibitor of D-amino acid oxidase; modification results in specific incorporation of an amine group into an accessible nucleophilic residue with concomitant release of 2,4-dinitrophenol.<br>References D'Silva, C., et al.: Biochemi., 25, 5602 (1986),<br></p>Fórmula:C6H5N3O5Forma y color:Brown SolidPeso molecular:199.12N-Acetyl-Lys-Octreotide Trifluoroacetic Acid Salt
CAS:<p>Stability Hygroscopic<br>Applications N-Acetyl-Phe-Octreotide is used as reactant/reagent in inhibition of octreotide acylation inside PLGA microspheres by derivatization of amines of peptide with self-immolative protecting group.<br>References Shirangi, M., et al.: Bioconjugate Chem., 27, 576-585 (2016)<br></p>Fórmula:C51H68N10O11S2·xC2HF3O2Forma y color:NeatPeso molecular:1061.284Resolvin E1 Sodium Salt
CAS:Producto controladoFórmula:C20H29NaO5Forma y color:NeatPeso molecular:372.431(5E)-6-(4-Hydroxy-3-methoxyphenyl)-5-hexene-2,4-dione
CAS:Producto controlado<p>Applications Curcumin (C838500) and gingerdione derivative. A possible human glyoxalase I inhibitor. Flavor modifier.<br>References Yuan, M. et al.; Bioorg. Med. Chem. 19, 1189 (2011); Ley, J. et al.; J. Agr. Food Chem. 56, 6656 (2008)<br></p>Fórmula:C13H14O4Forma y color:NeatPeso molecular:234.25(±)-Procinolol Hydrochloride
CAS:Producto controlado<p>Applications (±)-Procinolol is a beta adrenergic receptor antagonist.<br>References Singh, K.: Indian J. Phsiol. Pharmacol., 27, 311 (1983)<br></p>Fórmula:C15H24ClNO2Forma y color:NeatPeso molecular:285.81Baohuoside I
CAS:Producto controlado<p>Applications Baohuoside I is an inhibitor of cell growth and also is a down-regulator of durvivin and cyclin D1 expression. Used in the treatment of esophageal cancer. Anti-cancer agent.<br>References Lifang, W. et al.: Oncology Rep., 26, 1149 (2011); Jin, X. et al.: Drug Dev. Ind. Pharm., 39, 1421 (2013);<br></p>Fórmula:C27H30O10Forma y color:NeatPeso molecular:514.52Raloxifene 4’-β-D-Glucuronide Lithium Salt
CAS:Producto controlado<p>Stability Hygroscopic<br>Applications Raloxifene 4’-Glucuronide Lithium Salt is a metabolite of Raloxifene (R099995), a nonsteroidal estrogen receptor mixed agonist/antagonist.<br>References Dodge, J., et al.: Bioorg. Med. Chem. Lett., 7, 993 (1997); Jeong, E., et al.: Drug Metab. Dispos., 33, 785 (2005); Trontelj, J., et al.: Pharmacol. Res., 52, 334 (2005); Oswald, S., et al.: Clin. Pharmacol. Ther., 79 206 (2006)<br></p>Fórmula:C34H34LiNO10SForma y color:NeatPeso molecular:655.644-Amino-5-(bromomethyl)-2-methylpyrimidine Dihydrobromide
CAS:Producto controlado<p>Applications A pyrimidine derivative as G protein-coupled receptor kinase (GRK) inhibitor.<br>References Bigham, E., et al.: J. Med. Chem., 35, 1399 (1992), Jansen, M., et al.: Biochem. Pharmacol., 47, 1067 (1994), Hasbi, A., et al.: J. Neurochem., 70, 2129 (1998),<br></p>Fórmula:C17H17N3O2SForma y color:NeatPeso molecular:327.40N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamide Dihydrochloride
CAS:Producto controlado<p>Applications Found to have a potent inhibitory action against casein kinase 1 completely with respect to ATP and a much weaker effect on casein kinase 2 and other protein kinases.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hidaka, H., et al.: J. of Biol. Chem., 264, 9, 4924 (1989)<br></p>Fórmula:C11H12ClN3O2S·2ClHForma y color:NeatPeso molecular:358.67
![3a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-di…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FT293625.webp&w=3840&q=75)
