Serina / treonina quinasa
Los inhibidores de quinasas de serina/treonina son compuestos que se dirigen a las enzimas responsables de la fosforilación de residuos de serina y treonina en proteínas, las cuales desempeñan un papel crucial en la regulación de la apoptosis y otros procesos celulares. Estas quinasas están involucradas en vías de señalización que controlan el crecimiento, la división y la muerte celular programada. Inhibir quinasas específicas de serina/treonina puede alterar el equilibrio entre la supervivencia celular y la apoptosis, lo que convierte a estos inhibidores en herramientas esenciales en la investigación del cáncer y otras áreas de la biología celular. En CymitQuimica, ofrecemos una selección completa de inhibidores de quinasas de serina/treonina de alta calidad para apoyar su investigación en apoptosis, transducción de señales y mecanismos de enfermedades.
Se han encontrado 15 productos de "Serina / treonina quinasa"
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BMT-124110 Formate
<p>BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase</p>Fórmula:C22H20N2O2Pureza:99.52%Forma y color:SoildPeso molecular:344.41CID755673
CAS:<p>CID755673 inhibits PKD (IC50: 182 nM), with selectivity over PLK1, AKT, CAMKIIα, CAK, PKC.</p>Fórmula:C12H11NO3Pureza:97.68% - 99.84%Forma y color:SolidPeso molecular:217.221-Naphthyl PP1
CAS:<p>1-Naphthyl PP1 (1-NA-PP 1) is a selective src inhibitor(v-Src and c-Fyn, c-Abl, CDK2 and CAMK II with IC50s of 1.0, 0.6, 0.6, 18 and 22 μM, respectively)</p>Fórmula:C19H19N5Pureza:99.85%Forma y color:White Cyrstalline SolidPeso molecular:317.39PKD-IN-1
CAS:<p>CRT0066101 is an inhibitor of PKD.</p>Fórmula:C18H19ClN4OPureza:98%Forma y color:SolidPeso molecular:342.82kb NB 142-70
CAS:<p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>Fórmula:C11H9NO2S2Pureza:98.15% - ≥95%Forma y color:SolidPeso molecular:251.321-NM-PP1
CAS:<p>1-NM-PP1 (PP1 Analog II) is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.</p>Fórmula:C20H21N5Pureza:98% - 98.93%Forma y color:White Cyrstalline SolidPeso molecular:331.41N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
CAS:<p>Novel 2,6-naphthyridine inhibits PKC/PKD, identified by HTS.</p>Fórmula:C23H28N6Pureza:98.35%Forma y color:SolidPeso molecular:388.51ML-7 hydrochloride
CAS:<p>ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM);</p>Fórmula:C15H18ClIN2O2SPureza:99% - 99.26%Forma y color:White PowderPeso molecular:452.74CID 2011756
CAS:<p>CID 2011756 is an ATP-competitive and specific PKD1 inhibitor.</p>Fórmula:C22H21ClN2O3Pureza:98.15% - ≥95%Forma y color:SolidPeso molecular:396.87Benzamidine hydrochloride
CAS:<p>Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin.</p>Fórmula:C7H9ClN2Pureza:99.25% - 99.97%Forma y color:White To Off-White PowderPeso molecular:156.61SPHINX31
CAS:<p>SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).</p>Fórmula:C27H24F3N5O2Pureza:98.81% - 99.3%Forma y color:SolidPeso molecular:507.51GAK inhibitor 49
CAS:<p>GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).</p>Fórmula:C20H22N2O5Pureza:98.71%Forma y color:SolidPeso molecular:370.4SGC-GAK-1
CAS:<p>SGC-GAK-1 is a selective cyclin G-associated kinase (GAK) inhibitor (Ki: 3.1 nM).</p>Fórmula:C18H17BrN2O3Pureza:99.85%Forma y color:SolidPeso molecular:389.24SRPKIN-1
CAS:<p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>Fórmula:C27H21FN2O3SPureza:98%Forma y color:SolidPeso molecular:472.53MS-444
CAS:<p>MS-444 (BE-34776) is an MLCK and HuR inhibitor with antitumor activity that can be used to study triple-negative breast cancer and colorectal cancer.</p>Fórmula:C13H10O4Pureza:99.45% - 99.45%Forma y color:SolidPeso molecular:230.22
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