Serina / treonina quinasa

Piceatannol is an anti-inflammatory, immunomodulatory and antiproliferative agent. It inhibits p56lck and syk protein tyrosine …

Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) …

HA-1004 is a inhibitor of PKG, PKA, PKC and MLC.

Fasudil is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.

BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 …

CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective …

WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all …

SBC-115337 is a PCSK9 inhibitor.

Fasudil Hydrochloride is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of …

CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM …

SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).

WNK-IN-11 is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)

R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells …

CID797718 is a protein kinase D1 (PKD1) inhibitor.

FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.

kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the …

SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor

Benzamidine HCl is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki …

CID-2011756 is an ATP-competitive and specific PKD1 inhibitor.

ML-7 Hcl is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain …

Nafamostat mesylate, a synthetic serine protease inhibitor, has been used for the treatment of allergic …

SRPIN340, a serine/arginine-rich protein kinase (SRPK)-specific inhibitor, is potent for SRPK1 (IC50 = 0.89 uM).

kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, …

Cetraxate HCl is an oral gastrointestinal medication. It has a cytoprotective effect.

Pinostrobin, a potent flavonoid inducer, exerts a neuroprotective effect against Aα2(25-35)-induced neurotoxicity in PC12 cells, …

1 nM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor …

Camostat is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.

SBC-115076 is a potent extracellular proprotein convertase subtilisin kexin type 9 (PCSK9) antagonist.

(+)-Isocorydine is a eukaryote protein kinases Inhibitor.

6-(Dimethylamino)purine is a serine threonine protein kinase and CDK inhibitor

Wortmannin is the first described PI3K inhibitor with IC50 of 3 nM, with little selectivity …

N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein …

CRT0066101 dihydrochloride is an inhibitor of PKD.

MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase …

SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).

IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 …

CRT0066101 is an inhibitor of PKD.