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Integrin

Integrin

Los inhibidores de integrinas se dirigen a las integrinas, una familia de receptores en la superficie celular que desempeñan un papel crucial en la adhesión celular, la migración y la transducción de señales. Las integrinas están involucradas en la regulación del ciclo celular, particularmente en procesos como la división y la diferenciación celular. Inhibir las integrinas puede interrumpir estos procesos, lo que lleva al arresto del ciclo celular y la apoptosis, lo que hace que estos inhibidores sean valiosos en la investigación del cáncer y el estudio de la metástasis. En CymitQuimica, ofrecemos una amplia gama de inhibidores de integrinas de alta calidad para apoyar su investigación en la regulación del ciclo celular, la biología del cáncer y el desarrollo terapéutico.

Se han encontrado 256 productos de "Integrin"

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  • Lotrafiban hydrochloride

    CAS:
    Lotrafiban hydrochloride is an platelet glycoprotein IIb/IIIa blocker with oral activity.
    Fórmula:C23H33ClN4O4
    Forma y color:Solid
    Peso molecular:464.99
  • BI-1950

    CAS:
    BI-1950: potent inhibitor of LFA-1, key in immune function and drug target.
    Fórmula:C32H26Cl2FN7O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:646.5
  • ATN-161

    CAS:
    ATN-161 is an integrin α5β1 binding peptide and antagonist that inhibits VEGF-induced hCECs migration and angiogenesis.
    Fórmula:C23H35N9O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:597.64
  • αvβ1 integrin-IN-1

    CAS:
    <p>αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.</p>
    Fórmula:C26H34N6O6S
    Pureza:99.74% - >99.99%
    Forma y color:Solid
    Peso molecular:558.65
  • Roxifiban acetate

    CAS:
    Roxifiban acetate(DMP 754 acetate) is a potent GP IIb / IIIa antagonist that exhibits antiplatelet aggregation activity via immune mediation and can be used in
    Fórmula:C23H33N5O8
    Pureza:97.91% - 98.36%
    Forma y color:Solid
    Peso molecular:507.54
  • L 734217

    CAS:
    L 734217 is an antagonist of the fibrinogen receptor.
    Fórmula:C18H31N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:353.46
  • Des-ethyl-carafiban

    CAS:
    Des-ethyl-carafiban (Compound 44) is an antagonist of the fibrinogen receptor, effectively inhibiting platelet aggregation induced by various agonists. It is useful for research in thrombotic diseases.
    Fórmula:C22H23N5O5
    Forma y color:Solid
    Peso molecular:437.448
  • 6-B345TTQ

    CAS:
    6-B345TTQ is an α4 integrin inhibitor that can impede the interaction between α4 and Leupaxin. This compound is applicable for studies focused on inflammation research.
    Fórmula:C22H20BrNO4
    Forma y color:Solid
    Peso molecular:442.303
  • α5β1 integrin agonist-1

    CAS:
    α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.
    Fórmula:C24H26FN5O9
    Forma y color:Solid
    Peso molecular:547.49
  • SF0166

    CAS:
    SF0166: potent αvβ3 antagonist, IC50: 0.6 nM. Blocks cell adhesion, IC50: 7.6 pM-76 nM. Reduces neovascularization in mice.
    Fórmula:C23H27F2N5O4
    Forma y color:Solid
    Peso molecular:475.49
  • Zalunfiban dihydrochloride


    <p>Zalunfiban (RUC-4) is a potent αIIbβ3 platelet antagonist, IC50 45 nM, used in myocardial infarction research.</p>
    Fórmula:C16H20Cl2N8O2S
    Forma y color:Solid
    Peso molecular:459.35
  • OPN expression inhibitor 1

    CAS:
    OPN expression inhibitor 1 is an osteopontin expression inhibitor used in the study of breast cancer metastasis.
    Fórmula:C25H33N3O5
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:455.55
  • Fradafiban

    CAS:
    Fradafiban binds to the human platelet GP IIb/IIIa complex with a Kd value of 148 nM. Fradafiban is a non-polypeptide platelet glycoprotein IIb/IIIa antagonist.
    Fórmula:C20H21N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:367.40
  • GSK3335103

    CAS:
    GSK3335103 is a non-peptide, orally active inhibitor of αvβ6 integrin (pIC50=8), employed in the study of pulmonary fibrosis.
    Fórmula:C27H36FN3O4
    Forma y color:Solid
    Peso molecular:485.59
  • SR121566A

    CAS:
    SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).
    Fórmula:C20H25N5O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:431.51
  • GR 83895

    CAS:
    GR 83895 is an antagonist of prototype fibrinogen receptor.
    Fórmula:C29H39N9O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:673.74