Somatostatina
La somatostatina es una hormona peptídica que inhibe la liberación de varias otras hormonas, incluyendo la hormona de crecimiento, insulina y glucagón. Actúa al unirse a los receptores de somatostatina, que son receptores acoplados a proteínas G expresados en varios tejidos. Los análogos de la somatostatina se utilizan en el tratamiento de la acromegalia, tumores neuroendocrinos y trastornos gastrointestinales. Estos análogos también son herramientas valiosas para estudiar la secreción y señalización hormonal. En CymitQuimica, ofrecemos una gama completa de análogos de somatostatina de alta calidad para apoyar su investigación en endocrinología, regulación hormonal y desarrollo terapéutico.
Se han encontrado 54 productos de "Somatostatina"
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(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.Fórmula:C20H29N3O8Pureza:99.72%Forma y color:SoildPeso molecular:439.46Somatostatin acetate
<p>Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for the study of cancer and neurological disorders.</p>Pureza:99.11%Forma y color:Odour SolidCortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects andFórmula:C80H112N18O19S2Pureza:97.86%Forma y color:SolidPeso molecular:1693.98Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Fórmula:C83H118N20O20S2Pureza:98.24% - 99.63%Forma y color:SoildPeso molecular:1780.08Seglitide acetate
CAS:<p>Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.</p>Fórmula:C46H60N8O9Pureza:98.87%Forma y color:SolidPeso molecular:869.02Seglitide
CAS:<p>Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.</p>Fórmula:C44H56N8O7Pureza:98%Forma y color:SolidPeso molecular:808.98Ilatreotide
CAS:Ilatreotide is a Amadori compound of octreotide.Fórmula:C61H86N10O20S2Pureza:98%Forma y color:SolidPeso molecular:1343.53CYN 154806
CAS:CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).Fórmula:C56H68N12O14S2Pureza:98%Forma y color:SolidPeso molecular:1197.34Cortistatin 14, human, rat
CAS:Cortistatin 14: a neuropeptide similar to somatostatin; induces sleep, depresses neuronal activity; found in cortex, hippocampus.Fórmula:C81H113N19O19S2Pureza:98%Forma y color:SolidPeso molecular:1721.01Veldoreotide
CAS:Veldoreotide (Somatoprim): a somatostatin analogue targeting receptors 2, 4, 5, reduces GH in pituitary adenomas.Fórmula:C60H74N12O10Pureza:98%Forma y color:SolidPeso molecular:1123.3Somatostatin(3-6)
CAS:Somatostatin(3-6) is a somatostatin fragment.Fórmula:C22H34N6O6SForma y color:SolidPeso molecular:510.61MMC(TMZ)-TOC TFA
MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.Fórmula:C74H99F3N20O21S2Forma y color:SolidPeso molecular:1725.82Somatostatin
CAS:Somatostatin: a peptide hormone inhibiting growth hormone, insulin, and glucagon; secreted by hypothalamus and pancreatic D cells.Pureza:98%Forma y color:PowderPeso molecular:1637.88CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Fórmula:C74H96N14O15S2Pureza:98%Forma y color:SolidPeso molecular:1485.8MMC(TMZ)-TOC
MMC(TMZ)-TOC exhibits a high binding affinity and selectivity for somatostatin receptor subtype 2 (SSTR2). It is designed to target and deliver TMZ specifically to SSTR2-positive tumor cells. MMC(TMZ)-TOC is applicable for cancer research.Fórmula:C72H98N20O19S2Peso molecular:1610.67585Somatostatin-28 (1-14)
CAS:Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.Fórmula:C61H105N23O21SPureza:98%Forma y color:SolidPeso molecular:1528.71Cortistatin 29
Cortistatin 29: neuropeptide, relieves neuropathic pain, binds SS receptors (IC50: 2.8-13.7 nM), anti-fibrotic.Fórmula:C161H242N46O41S2Forma y color:SolidPeso molecular:3539.77Satoreotide
CAS:Satoreotide (JR11) is an SSTR2 antagonist, typically conjugated with radiolabeled chelators for use in neuroendocrine tumor imaging [1].Fórmula:C58H72ClN15O14S2Forma y color:SolidPeso molecular:1302.87L-796,778
CAS:<p>L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.</p>Fórmula:C29H40N6O7Pureza:96.20%Forma y color:SolidPeso molecular:584.66BIM-23190 hydrochloride
<p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>Forma y color:LiquidDOTA-JR11
CAS:DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Fórmula:C74H98ClN19O21S2Forma y color:SolidPeso molecular:1689.27Dotanoc
CAS:Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Fórmula:C69H94N14O17S2Forma y color:SolidPeso molecular:1455.71Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Fórmula:C53H71N11O14S2Forma y color:SolidPeso molecular:1150.33Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Fórmula:C46H58F3N7O8Forma y color:SolidPeso molecular:893.99L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Fórmula:C31H44N6O9Pureza:98%Forma y color:SoildPeso molecular:644.72Tau conotoxin CnVA
CAS:Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Fórmula:C72H116N24O17S4Forma y color:SolidPeso molecular:1718.1SSTR4 agonist-1
CAS:<p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>Fórmula:C16H23N3O2Forma y color:SolidPeso molecular:289.37L-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Fórmula:C38H50ClN5O2Pureza:98.65% - >99.99%Forma y color:SoildPeso molecular:644.30Neuronostatin-13 (human)
CAS:Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.Fórmula:C64H110N20O16Pureza:98%Forma y color:SolidPeso molecular:1415.68[D-Trp8,Tyr11] Somatostatin
CAS:[D-Trp8,Tyr11] Somatostatin, an analogue of the hormone somatostatin that modulates numerous bodily functions, is characterized by the substitution of DTrp8,Fórmula:C76H104N18O20S2Peso molecular:1653.88[Tyr11]-Somatostatin
CAS:[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Fórmula:C76H104N18O20S2Peso molecular:1653.89DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Fórmula:C105H133N21O30S5Peso molecular:2329.63Cortistatin-14
CAS:Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Fórmula:C81H114N20O18S2Pureza:98.06% - 98.23%Forma y color:SolidPeso molecular:1720.03Cyclosomatostatin Acetate
<p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>Fórmula:C46H61N7O8Pureza:98.83%Forma y color:SolidPeso molecular:840.02L803
CAS:L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.Fórmula:C50H80N13O19PForma y color:SolidPeso molecular:1198.22Somatostatin 1-28 acetate
Somatostatin 1-28 acetate circulates in human plasma.Pureza:99.22%Forma y color:Soild(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide
CAS:Somatostatin analog (Compound 4) with Kd: SSTR5-0.61nM, SSTR3-11.05nM, SSTR2-23.5nM, SSTR1-1.2µM, SSTR4->1µM.Fórmula:C50H67N11O10S2Peso molecular:1046.26[Tyr1]-Somatostatin-14
CAS:[Tyr1]-Somatostatin-14 could binds to SSTR2.Fórmula:C82H108N18O20S2Peso molecular:1729.99Anti-Somatostatin Antibody (9L93)
Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.Forma y color:Odour LiquidLanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Fórmula:C54H69N11O10S2Forma y color:SolidPeso molecular:1096.32BIM-23190 aceate
<p>BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.</p>Fórmula:C59H83N13O14S2Pureza:99.7%Forma y color:SolidPeso molecular:1262.5Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Fórmula:C27H22F2N4OPureza:99.91%Forma y color:SolidPeso molecular:456.49Pasireotide Acetate
CAS:The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Fórmula:C60H70N10O11Pureza:98.64% - 99.92%Forma y color:SolidPeso molecular:1107.26Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Fórmula:C51H70N10O12S2Pureza:99.03% - 99.87%Forma y color:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidPeso molecular:1079.3FK962
CAS:FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Fórmula:C14H17FN2O2Pureza:99.89%Forma y color:SolidPeso molecular:264.3Somatostatin Impurity 2 (13-Dha) Trifluoroacetate
Fórmula:C76H102N18O18S2·C2HF3O2Peso molecular:1619.88 114.02CYN 154806 TFA
CAS:CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.Fórmula:C58H69F3N12O16S2Pureza:99.7%Forma y color:SolidPeso molecular:1311.36Edotreotide
CAS:Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.Fórmula:C65H92N14O18S2Pureza:96.95%Forma y color:SolidPeso molecular:1421.64L-803087
CAS:L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Fórmula:C25H29F2N5O3Pureza:99.37%Forma y color:SolidPeso molecular:485.53L-796778 acetate
CAS:L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.Fórmula:C31H44N6O9Forma y color:SolidPeso molecular:644.716SST1 receptor antagonist-1
CAS:SST1 receptor antagonist-1 (Compound 23) is a selective antagonist of the somatostatin receptor 1 (SST1), showing a pKd of 9.11 for rSST1 and 8.79 for hSST1. This compound is applicable in research related to retinal and endocrine dysfunction, cancer, and neuropsychiatric disorders.Fórmula:C29H31F2N3O2Forma y color:SolidPeso molecular:491.57SSTR5 antagonist 6
CAS:SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].Fórmula:C22H28ClN3O4Forma y color:SolidPeso molecular:433.93
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