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Receptor de glucocorticoides

Receptor de glucocorticoides

El receptor de glucocorticoides (GR) es un receptor hormonal nuclear que media los efectos de los glucocorticoides, una clase de hormonas esteroides involucradas en la regulación del metabolismo, la respuesta inmunitaria y el estrés. Los agonistas y antagonistas del receptor de glucocorticoides se utilizan ampliamente en el tratamiento de enfermedades inflamatorias y autoinmunes, así como en la terapia contra el cáncer. Los moduladores de GR también son herramientas importantes para estudiar los roles fisiológicos y patológicos de los glucocorticoides. En CymitQuimica, ofrecemos una amplia gama de moduladores del receptor de glucocorticoides de alta calidad para apoyar su investigación en endocrinología, inmunología y regulación hormonal.

Se han encontrado 153 productos de "Receptor de glucocorticoides"

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  • Halcinonide

    CAS:
    <p>Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.</p>
    Fórmula:C24H32ClFO5
    Pureza:99.32% - 99.93%
    Forma y color:Solid
    Peso molecular:454.96
  • Prednisolone disodium phosphate

    CAS:
    <p>Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.</p>
    Fórmula:C21H27Na2O8P
    Pureza:97.1% - 99.16%
    Forma y color:Solid
    Peso molecular:484.39
  • Dexamethasone Phosphate disodium

    CAS:
    <p>Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.</p>
    Fórmula:C22H28FNa2O8P
    Pureza:99.76% - 99.848%
    Forma y color:White To Off White Powder
    Peso molecular:516.4
  • Loteprednol etabonate

    CAS:
    <p>Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.</p>
    Fórmula:C24H31ClO7
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:466.95
  • Nimodipine

    CAS:
    <p>Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle cells.</p>
    Fórmula:C21H26N2O7
    Pureza:99.64% - 99.79%
    Forma y color:Solid
    Peso molecular:418.44
  • Prednisolone

    CAS:
    <p>Prednisolone (Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.</p>
    Fórmula:C21H28O5
    Pureza:99.59% - 99.85%
    Forma y color:Crystals Solid
    Peso molecular:360.44
  • Hydrocortisone acetate

    CAS:
    <p>Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive</p>
    Fórmula:C23H32O6
    Pureza:98.89% - 99.22%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:404.5
  • Hydrocortisone Valerate

    CAS:
    <p>Hydrocortisone Valerate (Westcort) has anti-inflammatory, antipruritic and vasoconstrictive properties.</p>
    Fórmula:C26H38O6
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:446.58
  • Dexamethasone

    CAS:
    <p>Dexamethasone: a glucocorticoid agonist; modulates IL receptors; reduces inflammatory miRNA-155 exosomes in macrophage responses.</p>
    Fórmula:C22H29FO5
    Pureza:98% - 99.91%
    Forma y color:Crystals From Ether (Ntp 1992)
    Peso molecular:392.46
  • Miricorilant

    CAS:
    <p>Miricorilant (CORT 118335) is a glucocorticoid receptor modulator for the study of digestive and metabolic disorders.</p>
    Fórmula:C24H23F3N2O2
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:428.45
  • Amcinonide

    CAS:
    <p>Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.</p>
    Fórmula:C28H35FO7
    Pureza:98.33% - 99.62%
    Forma y color:Solid
    Peso molecular:502.57
  • Hydrocortisone

    CAS:
    <p>Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.</p>
    Fórmula:C21H30O5
    Pureza:98.4% - 99.95%
    Forma y color:Plates From Alc Or Iso-Propyl Alc Solid
    Peso molecular:362.46
  • Fluocinolone (Acetonide)

    CAS:
    <p>Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin disorders.</p>
    Fórmula:C24H30F2O6
    Pureza:99.29% - 99.82%
    Forma y color:Crystals From Acetone & Hexane Solid
    Peso molecular:452.49
  • Fluticasone (propionate)

    CAS:
    <p>Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR agonist.</p>
    Fórmula:C25H31F3O5S
    Pureza:98.98% - >99.99%
    Forma y color:Crystalline Solid
    Peso molecular:500.57
  • GW-870086

    CAS:
    <p>GW-870086 is an effective anti-inflammatory agent.</p>
    Fórmula:C31H39F2NO6
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:559.64
  • Dexamethasone acetate

    CAS:
    <p>Dexamethasone acetate (NSC 39471) is a potent anti-inflammatory steroid, blocks NF-kB, and lacks salt-retention.</p>
    Fórmula:C24H31FO6
    Pureza:99.22% - 99.65%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:434.50
  • Medroxyprogesterone Acetate

    CAS:
    <p>Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a long-acting contraceptive.</p>
    Fórmula:C24H34O4
    Pureza:99.05% - 99.44%
    Forma y color:White Powder
    Peso molecular:386.52
  • Esaxerenone

    CAS:
    <p>Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.</p>
    Fórmula:C22H21F3N2O4S
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:466.47
  • Mirodenafil

    CAS:
    <p>Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.</p>
    Fórmula:C26H37N5O5S
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:531.67
  • Betamethasone valerate

    CAS:
    <p>Betamethasone valerate (Luxiq) is a synthetic glucocorticoid with metabolic, immunosuppressive and anti-inflammatory actions.</p>
    Fórmula:C27H37FO6
    Pureza:99.32% - >99.99%
    Forma y color:Mixed With A Solvent
    Peso molecular:476.58