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Enzima

Enzima

Los inhibidores enzimáticos son moléculas que se unen a las enzimas y disminuyen su actividad. Estos inhibidores se utilizan ampliamente en la investigación para estudiar la cinética enzimática, la regulación y el papel de enzimas específicas en las vías metabólicas. Los inhibidores enzimáticos también son cruciales en el desarrollo de fármacos, ya que muchos agentes terapéuticos funcionan inhibiendo enzimas involucradas en procesos patológicos. Al dirigirse a las enzimas, estos inhibidores pueden modular las vías bioquímicas y ofrecer tratamientos potenciales para diversas enfermedades. En CymitQuimica, ofrecemos una amplia selección de inhibidores enzimáticos de alta calidad para apoyar su investigación en bioquímica, farmacología y descubrimiento de fármacos.

Subcategorías de "Enzima"

Se han encontrado 3587 productos de "Enzima"

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  • Quinethazone

    CAS:
    <p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>
    Fórmula:C10H12ClN3O3S
    Forma y color:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)
    Peso molecular:289.74
  • hCAIX-IN-10

    CAS:
    <p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>
    Fórmula:C28H21N3O3S
    Forma y color:Solid
    Peso molecular:479.55
  • hCAI/II-IN-3

    CAS:
    <p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>
    Fórmula:C16H18N4O4S2
    Forma y color:Solid
    Peso molecular:394.47
  • hCAI/II-IN-1

    CAS:
    <p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>
    Fórmula:C18H29N5O3S3
    Forma y color:Solid
    Peso molecular:459.65
  • hCAIX-IN-6

    CAS:
    <p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>
    Fórmula:C18H12N2O4S
    Forma y color:Solid
    Peso molecular:352.36
  • hCAIX-IN-11

    CAS:
    <p>hCAIX-IN-11 inhibits carbonic anhydrases IX &amp; XII with Ki of 32.7 nM &amp; 623.5 nM, respectively.</p>
    Fórmula:C21H15ClN4O3
    Forma y color:Solid
    Peso molecular:406.82
  • hCAIX/XII-IN-2

    CAS:
    <p>Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); &gt;10,000 nM (hCAI/II).</p>
    Fórmula:C19H14N2O4
    Forma y color:Solid
    Peso molecular:334.33
  • hCAII-IN-1

    CAS:
    <p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>
    Fórmula:C21H21BrN6O4S
    Forma y color:Solid
    Peso molecular:533.4
  • HCAIX-IN-2

    CAS:
    HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).
    Fórmula:C19H16N8O4S
    Forma y color:Solid
    Peso molecular:452.45
  • LP-533401

    CAS:
    <p>LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.</p>
    Fórmula:C27H22F4N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:526.48
  • hCAXII-IN-2

    CAS:
    <p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>
    Fórmula:C21H18ClN3O4
    Forma y color:Solid
    Peso molecular:411.84
  • DTP348

    CAS:
    <p>DTP348: Oral carbonic anhydrase IX inhibitor &amp; hypoxic cell radiosensitizer with sulfamide &amp; 5-nitroimidazole components.</p>
    Fórmula:C6H11N5O4S
    Forma y color:Solid
    Peso molecular:249.25
  • PPIE Protein, Human, Recombinant (His)


    <p>Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-type</p>
    Forma y color:Lyophilized Powder
    Peso molecular:34 KDa (reducing condition)
  • Phenylthiazolylthiourea

    CAS:
    <p>Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.</p>
    Fórmula:C10H9N3S2
    Forma y color:Solid
    Peso molecular:235.33
  • hCAXII-IN-4

    CAS:
    <p>hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.</p>
    Fórmula:C22H27N5O6S
    Forma y color:Solid
    Peso molecular:489.54
  • hCAI/II-IN-2

    CAS:
    <p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>
    Fórmula:C12H12N4O5S2
    Forma y color:Solid
    Peso molecular:356.38
  • Tyrosinase-IN-7

    CAS:
    <p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>
    Fórmula:C15H10O5
    Pureza:99%
    Forma y color:Solid
    Peso molecular:270.24
  • hCA IX-IN-2


    <p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>
    Fórmula:C23H24N2O4STe
    Forma y color:Solid
    Peso molecular:552.11
  • hCAIX/XII-IN-6


    <p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>
    Fórmula:C26H23N3O6S4
    Forma y color:Solid
    Peso molecular:601.74
  • L-693612 HCl

    CAS:
    <p>L-693612 HCl is an inhibitor of carbonic anhydrase.</p>
    Fórmula:C14H25ClN2O5S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:433.01