
Enzima
Los inhibidores enzimáticos son moléculas que se unen a las enzimas y disminuyen su actividad. Estos inhibidores se utilizan ampliamente en la investigación para estudiar la cinética enzimática, la regulación y el papel de enzimas específicas en las vías metabólicas. Los inhibidores enzimáticos también son cruciales en el desarrollo de fármacos, ya que muchos agentes terapéuticos funcionan inhibiendo enzimas involucradas en procesos patológicos. Al dirigirse a las enzimas, estos inhibidores pueden modular las vías bioquímicas y ofrecer tratamientos potenciales para diversas enfermedades. En CymitQuimica, ofrecemos una amplia selección de inhibidores enzimáticos de alta calidad para apoyar su investigación en bioquímica, farmacología y descubrimiento de fármacos.
Subcategorías de "Enzima"
- Anhídrido carbónico(178 productos)
- Hidroxilasa(30 productos)
- MPO(2 productos)
- Reductasa(52 productos)
- Tirosinasa(67 productos)
Se han encontrado 3587 productos de "Enzima"
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Quinethazone
CAS:<p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>Fórmula:C10H12ClN3O3SForma y color:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)Peso molecular:289.74hCAIX-IN-10
CAS:<p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>Fórmula:C28H21N3O3SForma y color:SolidPeso molecular:479.55hCAI/II-IN-3
CAS:<p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>Fórmula:C16H18N4O4S2Forma y color:SolidPeso molecular:394.47hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Forma y color:SolidPeso molecular:459.65hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Fórmula:C18H12N2O4SForma y color:SolidPeso molecular:352.36hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Fórmula:C21H15ClN4O3Forma y color:SolidPeso molecular:406.82hCAIX/XII-IN-2
CAS:<p>Compound 6a: Selective hCAIX/XII inhibitor; Ki: 30 nM (hCAIX), 3.6 nM (hCAXII); >10,000 nM (hCAI/II).</p>Fórmula:C19H14N2O4Forma y color:SolidPeso molecular:334.33hCAII-IN-1
CAS:<p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>Fórmula:C21H21BrN6O4SForma y color:SolidPeso molecular:533.4HCAIX-IN-2
CAS:HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).Fórmula:C19H16N8O4SForma y color:SolidPeso molecular:452.45LP-533401
CAS:<p>LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.</p>Fórmula:C27H22F4N4O3Pureza:98%Forma y color:SolidPeso molecular:526.48hCAXII-IN-2
CAS:<p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>Fórmula:C21H18ClN3O4Forma y color:SolidPeso molecular:411.84DTP348
CAS:<p>DTP348: Oral carbonic anhydrase IX inhibitor & hypoxic cell radiosensitizer with sulfamide & 5-nitroimidazole components.</p>Fórmula:C6H11N5O4SForma y color:SolidPeso molecular:249.25PPIE Protein, Human, Recombinant (His)
<p>Peptidyl-prolyl cis-trans isomerase E, also known as Cyclophilin E, Cyclophilin-33, Rotamase E, CYP33, PPIE, is an enzyme which belongs to the cyclophilin-type</p>Forma y color:Lyophilized PowderPeso molecular:34 KDa (reducing condition)Phenylthiazolylthiourea
CAS:<p>Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.</p>Fórmula:C10H9N3S2Forma y color:SolidPeso molecular:235.33hCAXII-IN-4
CAS:<p>hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.</p>Fórmula:C22H27N5O6SForma y color:SolidPeso molecular:489.54hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Fórmula:C12H12N4O5S2Forma y color:SolidPeso molecular:356.38Tyrosinase-IN-7
CAS:<p>Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.</p>Fórmula:C15H10O5Pureza:99%Forma y color:SolidPeso molecular:270.24hCA IX-IN-2
<p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>Fórmula:C23H24N2O4STeForma y color:SolidPeso molecular:552.11hCAIX/XII-IN-6
<p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>Fórmula:C26H23N3O6S4Forma y color:SolidPeso molecular:601.74L-693612 HCl
CAS:<p>L-693612 HCl is an inhibitor of carbonic anhydrase.</p>Fórmula:C14H25ClN2O5S3Pureza:98%Forma y color:SolidPeso molecular:433.01
