Enzima
Los inhibidores enzimáticos son moléculas que se unen a las enzimas y disminuyen su actividad. Estos inhibidores se utilizan ampliamente en la investigación para estudiar la cinética enzimática, la regulación y el papel de enzimas específicas en las vías metabólicas. Los inhibidores enzimáticos también son cruciales en el desarrollo de fármacos, ya que muchos agentes terapéuticos funcionan inhibiendo enzimas involucradas en procesos patológicos. Al dirigirse a las enzimas, estos inhibidores pueden modular las vías bioquímicas y ofrecer tratamientos potenciales para diversas enfermedades. En CymitQuimica, ofrecemos una amplia selección de inhibidores enzimáticos de alta calidad para apoyar su investigación en bioquímica, farmacología y descubrimiento de fármacos.
Subcategorías de "Enzima"
- Anhídrido carbónico(196 productos)
- Hidroxilasa(36 productos)
- MPO(2 productos)
- Reductasa(53 productos)
- Tirosinasa(76 productos)
Se han encontrado 3590 productos para "Enzima". Se muestran los primeros 500.
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Methazolamide
CAS:Methazolamide (CL 8490) is a carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.Fórmula:C5H8N4O3S2Pureza:99.31% - 99.77%Forma y color:SolidPeso molecular:236.27KW-2450 Formate
KW-2450 Formate is an IGF-1R/IR tyrosine kinase inhibitor with antitumor effects that acts through inhibition of Aurora A and B kinases.KW-2450 Formate inhibits the growth of TNBC xenografts and induces tetraploid accumulation.Fórmula:C29H31N5O5SPureza:99.70%Forma y color:SolidPeso molecular:561.65Topiramate
CAS:Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.Fórmula:C12H21NO8SPureza:99.79% - 99.92%Forma y color:White To Off-White Crystalline PowderPeso molecular:339.36Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24CAIX Inhibitor S4
CAS:CAIX Inhibitor S4 (S4) is an effective inhibitor of carbonic anhydrase IX/XII with a Ki of 7 nM and 2 nM, respectively.Fórmula:C15H17N3O4SPureza:99.07%Forma y color:SolidPeso molecular:335.38Ref: TM-T36758
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg90,00€25mg178,00€50mg334,00€100mg500,00€500mg1.099,00€p-Ethynylphenylalanine hydrochloride
CAS:p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].Fórmula:C11H12ClNO2Pureza:99.03% - 99.83%Forma y color:SolidPeso molecular:225.67Fenclonine
CAS:Fenclonine (CP-10188) is a selective and irreversible inhibitor of tryptophan hydroxylase, a rate-limiting enzyme in the biosynthesis of serotonin.Fórmula:C9H10ClNO2Pureza:98.81% - >99.99%Forma y color:Crystals From Methanol White SolidPeso molecular:199.63Zonisamide
CAS:Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.Fórmula:C8H8N2O3SPureza:99.05% - 99.9%Forma y color:SolidPeso molecular:212.23Tioxolone
CAS:Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.Fórmula:C7H4O3SPureza:97.79%Forma y color:White SolidPeso molecular:168.175-Feruloylquinic acid
CAS:5-Feruloylquinic acid, a potent Sirt1 activator, may aid in developing anti-aging drugs.Fórmula:C17H20O9Pureza:99.03%Forma y color:SolidPeso molecular:368.34Telotristat ethyl
CAS:Telotristat ethyl (LX1606) is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.Fórmula:C27H26ClF3N6O3Pureza:98% - 99.89%Forma y color:White SolidPeso molecular:574.98Benzthiazide
CAS:Benzthiazide treats edema and hypertension by promoting diuresis and inhibiting kidney Na+/Cl- reuptake, but may reduce potassium and raise uric acid.Fórmula:C15H14ClN3O4S3Pureza:98.48% - 99.79%Forma y color:White SolidPeso molecular:431.94Acipimox
CAS:Acipimox (K-9321), a niacin derivative, treats hyperlipidemia in type 2 diabetics.Fórmula:C6H6N2O3Pureza:98.98%Forma y color:Low Yellow Liquid Or CrystallinePeso molecular:154.12Actarit
CAS:Actarit (4-acetylaminophenylacetic acid) is an anti-inflammatory drug.Fórmula:C10H11NO3Pureza:99.64% - 99.74%Forma y color:White Or Off-White Crystal Or Crystalline SolidPeso molecular:193.2Arbutin
CAS:Arbutin, a bearberry extract, blocks melanin by inhibiting tyrosinase.Fórmula:C12H16O7Pureza:99.58% - 99.87%Forma y color:White SolidPeso molecular:272.25Flanvotumab
CAS:Flanvotumab (IMC-20D7S) is a humanized antibody targeting TYRP1 with strong antitumor effects via NK cells and ADCC.Pureza:> 95%Forma y color:LiquidPeso molecular:145.42 kDaACT-678689
CAS:ACT-678689 (Compound Example 1.53.4) (Compound Example 1.53.4) is a tryptophan hydroxylase (TPH) inhibitor with an IC50 of 8 nM[1].Fórmula:C23H22ClFN6O4S2Pureza:99.46%Forma y color:SolidPeso molecular:565.04Ref: TM-T14119
1mg107,00€5mg245,00€1mL*10mM (DMSO)308,00€10mg371,00€25mg620,00€50mg858,00€100mg1.153,00€200mg1.549,00€Hydrochlorothiazide
CAS:Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。Fórmula:C7H8ClN3O4S2Pureza:99.43% - 99.50%Forma y color:White SolidPeso molecular:297.74pNNP
CAS:pNNP is a substrate for PP2C assays and inhibits β-carbonic anhydrase, α-carbonate dehydrogenase, and H. pylori.Fórmula:C6H6NO6PPureza:99.82%Forma y color:White SolidPeso molecular:219.09Brinzolamide
CAS:Brinzolamide (AL-4862) is a Carbonic Anhydrase Inhibitor. The mechanism of action of brinzolamide is as a Carbonic Anhydrase Inhibitor.Fórmula:C12H21N3O5S3Pureza:99.84% - >99.99%Forma y color:SolidPeso molecular:383.512-Methoxy-4-propylphenol
CAS:2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.Fórmula:C10H14O2Forma y color:SolidPeso molecular:166.22Carbonic anhydrase inhibitor 30
Carbonic anhydrase inhibitor30 (compound 17) is an inhibitor of carbonic anhydrase with Ki values of 2.13 μM for hCA I and 0.161 μM for hCA II[1].Fórmula:C23H22FN3O5SForma y color:SolidPeso molecular:471.12642Trypsin, bovine origin
CAS:Pureza:≥ 2000units/mg (USP)Forma y color:White or almost white crystalline powderPeso molecular:-Tyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Forma y color:Odour SolidBarbituric acid
CAS:Barbituric acid is a pyrimidine derivative and the basic skeleton of barbiturate drugs, barbiturate drugs and other heterocyclic compounds.Fórmula:C4H4N2O3Pureza:99.83%Peso molecular:128.09hCAII-IN-8
CAS:Compound CDy9 is a highly selective inhibitor of carbonic anhydrase (CA) with an IC50 value of 0.18 μM for hCA II.Fórmula:C15H16N2O5SPureza:99.73%Forma y color:White SolidPeso molecular:336.36Ref: TM-T67774
5mg42,00€1mL*10mM (DMSO)52,00€10mg64,00€25mg116,00€50mg167,00€100mg241,00€200mg339,00€Calmodulin-dependent Protein Kinase II fragment 290-309
CAS:Fórmula:C103H185N31O24SPeso molecular:2273.83Anhydrotetracycline hydrochloride
CAS:Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.Fórmula:C22H23ClN2O7Pureza:98% - 98.90%Forma y color:SolidPeso molecular:462.885,6-Dihydro-2H-pyran-2-one
CAS:5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.Fórmula:C5H6O2Forma y color:SolidPeso molecular:98.1TPH1-IN-1
TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.Fórmula:C21H18N6O4SForma y color:SolidPeso molecular:450.47Proteinase K
CAS:Pureza:≥ 30units/mg (pH 7.5, 37°C, dried basis)Forma y color:White or almost white lyophilized powderPeso molecular:-Peroxidase, from horseradish, approx. 200 U/mg
CAS:Pureza:≥ 150U/mgForma y color:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecular:-Tyrosinase-IN-32
Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.Fórmula:C15H19NO3Forma y color:SolidPeso molecular:261.32Tyrosinase-IN-43
Tyrosinase-IN-43 (Compound 12j) is a competitive tyrosinase inhibitor with an IC50 value of 10.49 μM for tyrosinase. It exhibits significant antioxidant activity and can be used in the study and treatment of pigmentation-related conditions such as melasma, freckles, age spots, and post-inflammatory hyperpigmentation.Tyrosinase-IN-34
Tyrosinase-IN-34 (compound 5a), a human tyrosinase inhibitor (IC 50: 3.5 μM), shows promise in regulating melanogenesis and pigmentation.Fórmula:C19H14BrClN4OForma y color:SolidPeso molecular:429.7CAIX/CAXII-IN-4
CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.Fórmula:C23H21N5O3SForma y color:SolidPeso molecular:447.51Peroxidase
CAS:Pureza:≥ 85units/mg (dry basis)Forma y color:Beige to light-brown, reddish brown or dark brown lyophilised powderPeso molecular:-
