Enzima
Los inhibidores enzimáticos son moléculas que se unen a las enzimas y disminuyen su actividad. Estos inhibidores se utilizan ampliamente en la investigación para estudiar la cinética enzimática, la regulación y el papel de enzimas específicas en las vías metabólicas. Los inhibidores enzimáticos también son cruciales en el desarrollo de fármacos, ya que muchos agentes terapéuticos funcionan inhibiendo enzimas involucradas en procesos patológicos. Al dirigirse a las enzimas, estos inhibidores pueden modular las vías bioquímicas y ofrecer tratamientos potenciales para diversas enfermedades. En CymitQuimica, ofrecemos una amplia selección de inhibidores enzimáticos de alta calidad para apoyar su investigación en bioquímica, farmacología y descubrimiento de fármacos.
Subcategorías de "Enzima"
- Anhídrido carbónico(196 productos)
- Hidroxilasa(36 productos)
- MPO(2 productos)
- Reductasa(51 productos)
- Tirosinasa(71 productos)
Se han encontrado 3620 productos de "Enzima"
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β-Galactosidase >100KU/g
CAS:beta-Galactosidase (EC 3.2.1.23, shortly beta-Gal, also know as lactase) catalyses the hydrolysis of beta-d-galactoside in the presence of water to galactose and alcohol, or lactose into glucose and galactose. beta-Gal has a molecular weight of 540,000 and is composed of four identical subunits of MW 135,000, each with an independent active site. The enzyme has divalent metals as cofactors, with chelated Mg2+ ions required to maintain active site conformation. The molecule contains numerous sulfhydryl groups and is glycosylated.Forma y color:PowderMyokinase (from Yeast)
CAS:Myokinase (Adenylate kinase, EC 2.7.4.3) catalyzes interconversion between ATP, ADP and AMP by catalyzing the following reaction:ATP + AMP ⇌ 2 ADPOne unit of Myokinase will convert 1.0 µmol ATP and 1.0 µmol AMP to 2.0 µmol ADP per min at 25°C and pH 7.5.D-Alanine Aminotransferase, Bacilus subtilis, Recombinant
D-Alanine aminotransferase (L-glutamic-pyruvic transaminase; EC 2.6.1.21) is an enzyme that catalyzes the following reaction: D-alanine + α-ketoglutarate ⇌ pyruvate + D-glutamate Please enquire for more information about D-Alanine Aminotransferase, Bacilus subtilis, Recombinant including the price, delivery time and more detailed product information at the technical inquiry form on this page
Pureza:>90% By Sds-Page.Tyrosinase-IN-2
CAS:Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Fórmula:C8H8N4O2SPureza:99.78%Forma y color:SolidPeso molecular:224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€Transglutaminase from streptoverticillium mobaraense
CAS:selectively deamidates gluten peptides, which results in strongly enhanced T cell-stimulatory activity. It has also been used in a study to improve quantifiable assays to fully characterize the role of transglutaminase in diseases such as Huntington′s disease and Alzheimer′s disease.Forma y color:PowderhCAIX-IN-16
CAS:hCAIX-IN-16 (Compound 12d), an inhibitor of hCA IX, exhibits inhibition constants (K i) of 190.0 nM for hCA IX and 187.9 nM for hCA XII.Fórmula:C20H20N8O2SPureza:98%Forma y color:SolidPeso molecular:436.49Sezolamide hydrochloride
CAS:Sezolamide hydrochloride is a potent topical carbonic anhydrase inhibitor.Fórmula:C11H19ClN2O4S3Forma y color:SolidPeso molecular:374.93hCAIX/XII-IN-8
CAS:hCAIX/XII-IN-8 (compound 3g) is a potent inhibitor of the human carbonic anhydrases (CAs) IX and XII, with inhibition constants (K i) of 8.5 nM for CA IX and 6.Fórmula:C16H13Cl2N5O3SPureza:98%Forma y color:SolidPeso molecular:426.28Diethyl-pythiDC
CAS:Diethyl-pythiDC is an collagen prolyl 4-hydroxylase inhibitor.Fórmula:C14H14N2O4SPureza:99.98%Forma y color:SolidPeso molecular:306.34Sezolamide
CAS:Sezolamide is a carbonic anhydrase inhibitor.Fórmula:C11H18N2O4S3Forma y color:SolidPeso molecular:338.47N-Desethyl Brinzolamide oxalate
CAS:N-Desethyl Brinzolamide oxalate functions as a dual inhibitor targeting Carbonic anhydrase II and Carbonic anhydrase IV, exhibiting inhibitory concentrations (IC50) of 1.28 nM and 128 nM, respectively [1].Fórmula:C12H19N3O9S3Forma y color:SolidPeso molecular:445.49CAXII-IN-1
CAS:CAXII-IN-1, antitumor, selectively inhibits CA XII with Ki of 3.8 nM for hCA XII and 56 nM for hCA IX.Fórmula:C13H7Cl2NO3SForma y color:SolidPeso molecular:328.17LX-1031
CAS:LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally.Fórmula:C28H25F3N4O4Pureza:97.123% - 98.97%Forma y color:SolidPeso molecular:538.52Ref: TM-T15796
1mg55,00€5mg120,00€10mg187,00€25mg376,00€50mg597,00€100mg938,00€200mg1.264,00€1mL*10mM (DMSO)143,00€COX-2-IN-30
CAS:COX-2-IN-30, a benzenesulfonamide derivative, is an orally active, dual inhibitor of cyclooxygenase-2 (COX-2; IC50 = 49 nM) and cyclooxygenase-1 (COX-1; IC50 =Fórmula:C17H16N6O3SPureza:98%Forma y color:SolidPeso molecular:384.41ALP/Carbonic anhydrase-IN-1
CAS:Compound 1e, also known as ALP/Carbonic anhydrase-IN-1, is a dual inhibitor targeting both carbonic anhydrase (CA) isozymes II, IX, and XII, as well as alkalineFórmula:C15H16N2Pureza:98%Forma y color:SolidPeso molecular:224.3Carbonic anhydrase inhibitor 12
CAS:CA Inhibitor 12 strongly blocks CA II (K_i 1.72 nM), also inhibits CA I (271 nM), shows anticancer effects.Fórmula:C27H22BrN5O5S2Pureza:98%Forma y color:SolidPeso molecular:640.53hCAIX-IN-15
CAS:hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancerFórmula:C18H14FN7O2SPureza:98%Forma y color:SolidPeso molecular:411.41Sulfatase, from helix pomatia ≥10,000 units/g solid
CAS:Sulfatase from Helix pomatia is a highly potent enzyme that is capable of hydrolyzing sulfated compounds and sulfate esters. It has been widely used in various applications such as glucosinolate analysis, genistein extraction preparation, and regiospecificity studies. With a concentration of ≥10,000 units per gram of solid, this sulfatase offers exceptional enzymatic activity for sulfatase assays. It effectively catalyzes the hydrolysis of sulfated substrates, including p-nitrocatechol sulfate, naphthyl sulfate and phenyl sulfates.The enzyme can be incubated with the desired sample to facilitate the release of sulfate groups from sulfated compounds. Sulfatase from Helix pomatia is a valuable tool for researchers and scientists working in diverse fields requiring efficient and reliable enzymatic hydrolysis capabilities. Additionally the enzyme has been found to have industrial applications, such as in the bioconversion of industrial chemicals, where it can be used as a catalyst.
Forma y color:Powderp-Ethynylphenylalanine
CAS:p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a tryptophan hydroxylase (TPH) inhibitor, is competitive, effective, selective, and reversible, with a Ki ofFórmula:C11H11NO2Pureza:99.44%Forma y color:SolidPeso molecular:189.21Glycerol 3-phosphate oxidase, from pediococcus sp., 40-84U/mg
CAS:Glycerol-3-phosphate oxidase (EC 1.1.3.21) is an enzyme that catalyzes the following reaction: glycerol-3-phosphate + O2 ⇌ dihydroxyacetone phosphate + H2O2 One unit of Glycerol-3-phosphate oxidase will generate 1.0 μmole H2O2 per min at 37°C, under the presence of O2 and the optimal pH. If required, you can remove the build-up of hydrogen peroxide using catalase.Pureza:Min. 95%Triose phosphate isomerase
CAS:Triose-phosphate isomerase (TPI, TIM; EC 5.3.1.1) is an enzyme that catalyzes the reversible isomerisation of dihydroxyacetone phosphate and D-glyceraldehyde 3-phosphate: DHAP ⇌ GADP The reaction mechanism involves the formation of an enediol intermediate. One unit of Triose-phosphate isomerase will convert 1.0 μmole glyceraldehyde 3-phosphate to dihydroxyacetone phosphate per min at pH 7.6 and 25 °C.Pureza:Min. 95%Glycerokinase, cellulomonas species
CAS:Glycerokinase (glycerol kinase, GP, ATP-glycerol 3-phosphotransferase; EC 2.7.1.30) is an enzyme that catalyzes the following reaction: ATP + glycerol ⇌ ADP + glycerol 3-phosphate One unit of Glycerokinase will convert 1.0 μmole of glycerol and ATP to glycerol 3-phosphate and ADP per min at pH 9.8 and 25 °C.Forma y color:PowderOxalate Oxidase, freeze-dried, from Wheat
CAS:Oxalate Oxidase, freeze-dried, is an enzymatic preparation that serves as a catalyst in biochemical reactions. This enzyme is derived from wheat, a common plant source, ensuring a naturally occurring origin. Its primary mode of action is the oxidation of oxalate into carbon dioxide and hydrogen peroxide. This biochemical activity is significant in various scientific applications, specifically in the breakdown of oxalate, which plays a crucial role in metabolic and environmental processes.Forma y color:PowderThioredoxin reductase from escherichia coli
CAS:Thioredoxin reductase (TR, TrxR) (EC 1.8.1.9) is an enzyme that reduce thioredoxin using NADPH as a co-factor, and also contains FAD. One unit of thioredoxin reductase will raise increase light absorbance by 1.0 per minute at 412nm in the presence of thioredoxin and Ellman's reagent at pH 7.0 and 25 °C.Pureza:Min. 95%Sarcosine oxidase from bacillus sp., >15 units/mg solid, lyophilized powder
CAS:Sarcosine oxidase (Monomeric sarcosine oxidase, MSOX, EC 1.5.3.1) is an enzyme that catalyzes the oxidative demethylation of sarcosine to yield glycine, H2O2 and formaldehyde in the following reaction: CH3-NH2+-CH2-COO- + H2O + O2 → NH3+-CH2-COO- + H2O2 + CH2O or sarcosine + water + oxygen → glycine + hydrogen peroxyde + formaldehydeOne unit of Sarcosine oxidase will form 1.0 micromole of formaldehyde from sarcosine per minute at pH 8.3 and 37 °C. You can remove the build-up of hydrogen peroxide using catalase.Fórmula:C10H12N8O3Pureza:Min. 95%Forma y color:PowderPeso molecular:292.25 g/molβ-Glucuronidase from Helix pomatia - Type H-2, aqueous solution, ≥85,000 units/mL
CAS:β-Glucuronidase (EC 3.2.1.31) is an enzyme that hydrolyzes glucuronides. It can also be used to cleave benzodiazepine and steroid conjugates. One unit of β-Glucuronidase will hydrolyze a chromogenic substrate mimic 4-nitrophenyl-β-D-glucuronide to produce 1.0 μmole of 4-nitrophenol per minute at pH 5.0 and 37 °C.Pureza:Min. 95%Forma y color:Clear LiquidCA IX-IN-1
CA IX-IN-1 (compound 12g) is a potent and highly selective hCA IX inhibitor (IC50: 7 nM) that exhibits antitumour effects.Fórmula:C16H22N4O8SForma y color:SolidPeso molecular:430.43CAII-IN-3
CAII-IN-3, a thiosemicarbazone, potently inhibits CA-II with an IC50 of 13.4 μM.Fórmula:C18H18F2N4SForma y color:SolidPeso molecular:360.42hCAII-IN-4
CAS:hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Fórmula:C31H23NO9Forma y color:SolidPeso molecular:553.52Sulclamide
CAS:Sulclamide, a sulfamoylbenzoic acid derivative, exhibits diuretic activity and functions as an inhibitor of carbonic anhydrase [1].Fórmula:C7H7ClN2O3SForma y color:SolidPeso molecular:234.66Tyrosinase-IN-20
CAS:Tyrosinase-IN-20 (compound 6a) acts as a potent Tyrosinase inhibitor, demonstrating an IC 50 value of 28.50 μM [1].Fórmula:C17H18N2O2SForma y color:SolidPeso molecular:314.44-Acetylphenylboronic acid
CAS:4-Acetylphenylboronic acid acts as an effective inhibitor targeting carbonic anhydrase II (CAII), displaying inhibitory concentrations (IC50) of 246 μM for bovine CAII (bCA II) and 281.40 μM for human CAII (hCA II).Fórmula:C8H9BO3Forma y color:SolidPeso molecular:163.97hCAII-IN-3
hCAII-IN-3 inhibits key hCA isoforms with Ki: hCA I (403.8 nM), hCA II (5.1 nM), hCA IX (10.2 nM), hCA XII (5.2 nM); shows anticancer potential.
Fórmula:C17H21N3O3SForma y color:SolidPeso molecular:347.43hCAIX/XII-IN-15
CAS:hCAIX/XII-IN-15 (Compound 17β) is an inhibitor of hCA IX and hCA XII, exhibiting Ki values of 0.42 and 4.37 μM, respectively. It demonstrates a pro-apoptotic effect in multiple myeloma cells.Fórmula:C17H18O4SForma y color:SolidPeso molecular:318.387Tyrosinase-IN-37
CAS:Tyrosinase-IN-37 (Compound 3c) is a potent inhibitor of tyrosinase, with an IC50 value of 1.02 μM, which is 14 times more effective than kojic acid (IC50 of 14.74 μM). This compound effectively prevents the browning of Rosa roxburghii and can also inhibit browning not caused by tyrosinase.Fórmula:C12H12N6SForma y color:SolidPeso molecular:272.33hCA XII/II/IX-IN-1
hCA XII/II/IX-IN-1 inhibits hCA I/II/IX/XII (IC50: 2.6, 0.004, 0.005, 0.001 μM) with anticancer properties.Fórmula:C25H34N4O7SForma y color:SolidPeso molecular:534.63Carbonic anhydrase inhibitor 8
R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).Fórmula:C20H25N3O4SForma y color:SolidPeso molecular:403.5CAII-IN-2
CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.Fórmula:C18H19BrN4SForma y color:SolidPeso molecular:403.34Valerate sodium
CAS:Valerate sodium is a potential Carbonic anhydrase 1/2 inhibitor for biochemical experiments.Fórmula:C5H9NaO2Pureza:99.84% - 99.91%Forma y color:SolidPeso molecular:124.11β-Glucuronidase/hCAII-IN-1
CAS:β-Glucuronidase/hCAII-IN-2 (Compound 12e) is a compound that effectively inhibits both β-glucuronidase and human Carbonic Anhydrase II (hCA II), exhibiting IC50Fórmula:C30H21NO9Forma y color:SolidPeso molecular:539.49NSC 828467
NSC 828467 is one of the top five CA-IX inhibitors with significant in vitro anticancer activity (IC50: 27.2 nM).Fórmula:C21H19N9O2SForma y color:SolidPeso molecular:461.5Carbonic anhydrase inhibitor 9
Carbonic anhydrase inhibitor 9 targets hCA II and IX with Ki of 56.4 and 56.9 nM respectively; shows antiproliferative activity.Fórmula:C22H20BrN5O4SForma y color:SolidPeso molecular:530.39Carbonic anhydrase inhibitor 19
CAS:Carbonic anhydrase inhibitor19 (compound 26a) targets glaucoma-associated isozymes hCA II and hCA XII, with inhibition constants (Kis) of 9.4 nM and 6.7 nM, respectively. This compound is effective in reducing intraocular pressure.Fórmula:C23H25N3O6S2Peso molecular:503.59Carbonic anhydrase inhibitor 17
CAS:Carbonic anhydrase inhibitor 17 (compound 7c) is a pyrazine-based sulfonamide that acts as a carbonic anhydrase II inhibitor, with an IC50 value of 0.63 nM.Fórmula:C18H15ClN4O3S2Peso molecular:434.92Carbonic anhydrase inhibitor 16
CAS:Carbonic anhydrase inhibitor 16 (compound 1) is a CA I/CA II inhibitor with potential antiviral activity, used in virus infection studies.Fórmula:C14H10N2O4SPureza:99.65%Forma y color:SolidPeso molecular:302.31Carbonic anhydrase inhibitor 5
Potent hCA inhibitor: targets hCA II, IX & XII with IC50s of 42.9, 47.6, & 6.7 nM respectively.Fórmula:C24H20ClN3O3SForma y color:SolidPeso molecular:465.95hCAIX-IN-20
CAS:hCAIX-IN-20 (compound APBS-5m) is a potent inhibitor of carbonic anhydrase IX (hCA IX), with a Ki of 2.7 nM, playing a significant role in cancer research.Fórmula:C19H13Cl2N5O4S2Peso molecular:510.37Tyrosinase-IN-33
CAS:Tyrosinase-IN-33 (compound 5), a pyridine-based compound, acts as an effective inhibitor of diphenolase activity in mushroom tyrosinase. It significantly reduces enzyme activity with an IC50 of 9.0 μM.Fórmula:C19H17NS2Forma y color:SolidPeso molecular:323.48Tyrosinase-IN-35
CAS:Tyrosinase-IN-35 (compound 6g), exhibiting a IC 50 value of 2.09 μM, serves as a more effective inhibitor of human tyrosinase compared to Kojic Acid (IC 50: 16.38 μM). At concentrations of 4 μM and 8 μM, this compound effectively lowers melanin levels in melanoma B16F10 cells in vitro.Fórmula:C17H15N5OSForma y color:SolidPeso molecular:337.40hCA VB-IN-1
hCA VB-IN-1 (compound 15) is a potent and selective inhibitor of hCA VB (carbonic anhydrase) with a KI of 515.7 nM [1].Fórmula:C9H13N3O4SForma y color:SolidPeso molecular:259.28
