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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"

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  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Fórmula:C6H11NO2
    Forma y color:Solid
    Peso molecular:129.16
  • CP-628006

    CAS:
    <p>CP-628006 is a small molecule CFTR potentiator that effectively restores ATP-dependent channel gating to G551D-CFTR, the mutant form found in cystic fibrosis.</p>
    Fórmula:C32H35F3N2O2
    Forma y color:Solid
    Peso molecular:536.639
  • P2X4 antagonist-3


    <p>P2X4 antagonist-3 (Compound 14c) is a P2X4 inhibitor with an IC50 value of 1.2 μM. It holds potential for research into neuroinflammation, chronic pain, and cancer progression.</p>
    Fórmula:C19H20FN3O4
    Forma y color:Solid
    Peso molecular:373.38
  • (±)8(9)-EpETE

    CAS:
    <p>(±)8(9)-EpETE ((±)8,9-EEQ) is an epoxide of arachidonic acid biosynthesized by CYP450 epoxygenase.1.2 In rat and rabbit liver microsomes.</p>
    Fórmula:C20H30O3
    Forma y color:Solid
    Peso molecular:318.45
  • GsMTx4

    CAS:
    <p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>
    Fórmula:C185H273N49O45S6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:4095.84
  • Jingzhaotoxin-XII TFA


    <p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>
    Forma y color:Odour Solid
  • Tiludronate disodium hemihydrate

    CAS:
    <p>Tiludronate: an oral bisphosphonate for bone disorder research; inhibits osteoclasts and reduces inflammation.</p>
    Fórmula:C14H16Cl2Na4O13P4S2
    Forma y color:Solid
    Peso molecular:743.16
  • Nitrazolam

    CAS:
    <p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>
    Fórmula:C17H13N5O2
    Forma y color:Solid
    Peso molecular:319.32
  • ω-Agatoxin IVA

    CAS:
    <p>Selective blocker of P-type calcium channels (IC50 &lt; 1 - 3 nM). Also inhibits N-type channels at micromolar concentrations.</p>
    Fórmula:C217H360N68O60S10
    Pureza:98%
    Forma y color:Solid
    Peso molecular:5202.25
  • PDDHV

    CAS:
    <p>PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.</p>
    Fórmula:C49H72O11
    Forma y color:Solid
    Peso molecular:837.09
  • Leptomycin A

    CAS:
    <p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>
    Fórmula:C32H46O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:526.7
  • LY393615


    <p>LY393615 (NCC1048) is a novel blocker of both neuronal Ca²⁺ (calcium) and Na⁺ (sodium) channels, exhibiting half-maximal inhibitory concentrations (IC₅₀) of 1.9</p>
    Pureza:98%
    Forma y color:Odour Solid
  • N-Oleoyl Glutamine

    CAS:
    <p>N-Oleoyl Glutamine (Oleoyl-L-glutamine) antagonizes TRPV1 of the transient receptor potential (TRP) calcium channel.</p>
    Fórmula:C23H42N2O4
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:410.59
  • ABCB1-IN-1


    <p>ABCB1-IN-1 (compound 3) is a potent inhibitor of ABCB1 that promotes cell apoptosis.</p>
    Fórmula:C36H33F3FeN2O4PS
    Forma y color:Solid
    Peso molecular:733.54
  • LTGO-33

    CAS:
    <p>LTGO-33 is a voltage-gated sodium channel NaV1.8 inhibitor that inhibits NaV1.8, NaV1.1-NaV1.7, and NaV1.9.</p>
    Fórmula:C21H17F4N3O3S
    Pureza:97.6%
    Forma y color:Soild
    Peso molecular:467.44
  • 5-Hydroxy-2′,3,4′,7-tetramethoxyflavone

    CAS:
    <p>5-Hydroxy-2′,3,4′,7-tetramethoxyflavone shows weak ABCG2 inhibitory potency with IC50s of 3.27 and 3.89 µM in the Hoechst 33342 and pheophorbide A assays.</p>
    Fórmula:C19H18O7
    Pureza:98%
    Forma y color:Soild
    Peso molecular:358.34
  • AChE/Aβ-IN-1


    <p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>
    Fórmula:C20H25BrN4
    Forma y color:Solid
    Peso molecular:401.34
  • SG-094

    CAS:
    <p>SG-094 inhibits TPC2, halts RIL175 cell growth, IC50: 3.7 μM for cancer research.</p>
    Fórmula:C30H29NO3
    Pureza:97.06%
    Forma y color:Soild
    Peso molecular:451.56
  • Cyclocreatine

    CAS:
    <p>Cyclocreatine, a creatine analogue and substrate for creatine kinase, inhibits creatine metabolism and prostate cancer cell proliferation.</p>
    Fórmula:C5H9N3O2
    Pureza:99.864%
    Forma y color:Solid
    Peso molecular:143.14
  • TRPA1-IN-2

    CAS:
    <p>TRPA1-IN-2 is a potent and orally active TRPA1 inhibitor with an IC50 value of 0.04 µM.TRPA1-IN-2 has anti-inflammatory activity.</p>
    Fórmula:C24H25F3N4O
    Pureza:98.05%
    Forma y color:Soild
    Peso molecular:442.48