
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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NaV1.7 inhibitor-1
CAS:<p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>Fórmula:C23H30FNO4SPureza:99.89%Forma y color:SolidPeso molecular:435.551-EBIO
CAS:<p>1-EBIO (1-EBIO) is a calium channel agonist.</p>Fórmula:C9H10N2OPureza:98.75%Forma y color:SolidPeso molecular:162.19MRZ 2-514
CAS:<p>MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki</p>Fórmula:C11H6BrN3O3Pureza:98.459%Forma y color:SolidPeso molecular:308.09Tertiapin-Q
CAS:<p>Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).</p>Fórmula:C106H175N35O24S4Pureza:98.06% - 98.09%Forma y color:SolidPeso molecular:2452Z433927330
CAS:<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Fórmula:C20H20N4O3Pureza:99.78%Forma y color:SolidPeso molecular:364.4Glimepiride
CAS:<p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C24H34N4O5SPureza:97.84% - 98.87%Forma y color:White Cyrstalline SolidPeso molecular:490.62Fluxametamide
CAS:<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26ML418
CAS:<p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>Fórmula:C19H24ClN3O3Pureza:99.3%Forma y color:SolidPeso molecular:377.87Piracetam
CAS:<p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>Fórmula:C6H10N2O2Pureza:97.16%Forma y color:Crystals From Isopropanol SolidPeso molecular:142.16Vocacapsaicin hydrochloride
CAS:<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Fórmula:C26H42ClN3O4Pureza:99.66% - 99.80%Forma y color:SolidPeso molecular:496.085,5-Dimethyloxazolidine-2,4-dione
CAS:<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Fórmula:C5H7NO3Pureza:99.12%Forma y color:Drypowder PelletslargecrystalsPeso molecular:129.11Etifoxine hydrochloride
CAS:<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Fórmula:C17H18Cl2N2OPureza:99.36%Forma y color:SolidPeso molecular:337.24CRAC intermediate 2
CAS:<p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>Fórmula:C11H7F6N3Pureza:99.69%Forma y color:SolidPeso molecular:295.18VU591 hydrochloride
CAS:<p>VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.</p>Fórmula:C16H13ClN6O5Pureza:98.93% - 99.22%Forma y color:SolidPeso molecular:404.76Cromolyn sodium
CAS:<p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>Fórmula:C23H14Na2O11Pureza:99.4% - 99.95%Forma y color:Colorless Crystals From Ethanol + Ether White Crystalline PowderPeso molecular:512.33Linoleoyl glycine
CAS:<p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>Fórmula:C20H35NO3Pureza:98.96%Forma y color:SolidPeso molecular:337.5Glipizide
CAS:<p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C21H27N5O4SPureza:99.67% - 99.75%Forma y color:SolidPeso molecular:445.54Moxidectin
CAS:<p>Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.</p>Fórmula:C37H53NO8Pureza:97.38%Forma y color:Appearance White Or Pale Yellow Amorphous PowderPeso molecular:639.82Methocarbamol
CAS:<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24Azosemide
CAS:<p>Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).</p>Fórmula:C12H11ClN6O2S2Pureza:99.84%Forma y color:SolidPeso molecular:370.84
