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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"

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  • NaV1.7 inhibitor-1

    CAS:
    <p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>
    Fórmula:C23H30FNO4S
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:435.55
  • 1-EBIO

    CAS:
    <p>1-EBIO (1-EBIO) is a calium channel agonist.</p>
    Fórmula:C9H10N2O
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:162.19
  • MRZ 2-514

    CAS:
    <p>MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki</p>
    Fórmula:C11H6BrN3O3
    Pureza:98.459%
    Forma y color:Solid
    Peso molecular:308.09
  • Tertiapin-Q

    CAS:
    <p>Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).</p>
    Fórmula:C106H175N35O24S4
    Pureza:98.06% - 98.09%
    Forma y color:Solid
    Peso molecular:2452
  • Z433927330

    CAS:
    <p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>
    Fórmula:C20H20N4O3
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:364.4
  • Glimepiride

    CAS:
    <p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>
    Fórmula:C24H34N4O5S
    Pureza:97.84% - 98.87%
    Forma y color:White Cyrstalline Solid
    Peso molecular:490.62
  • Fluxametamide

    CAS:
    <p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>
    Fórmula:C20H16Cl2F3N3O3
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:474.26
  • ML418

    CAS:
    <p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>
    Fórmula:C19H24ClN3O3
    Pureza:99.3%
    Forma y color:Solid
    Peso molecular:377.87
  • Piracetam

    CAS:
    <p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>
    Fórmula:C6H10N2O2
    Pureza:97.16%
    Forma y color:Crystals From Isopropanol Solid
    Peso molecular:142.16
  • Vocacapsaicin hydrochloride

    CAS:
    <p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>
    Fórmula:C26H42ClN3O4
    Pureza:99.66% - 99.80%
    Forma y color:Solid
    Peso molecular:496.08
  • 5,5-Dimethyloxazolidine-2,4-dione

    CAS:
    <p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>
    Fórmula:C5H7NO3
    Pureza:99.12%
    Forma y color:Drypowder Pelletslargecrystals
    Peso molecular:129.11
  • Etifoxine hydrochloride

    CAS:
    <p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>
    Fórmula:C17H18Cl2N2O
    Pureza:99.36%
    Forma y color:Solid
    Peso molecular:337.24
  • CRAC intermediate 2

    CAS:
    <p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>
    Fórmula:C11H7F6N3
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:295.18
  • VU591 hydrochloride

    CAS:
    <p>VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.</p>
    Fórmula:C16H13ClN6O5
    Pureza:98.93% - 99.22%
    Forma y color:Solid
    Peso molecular:404.76
  • Cromolyn sodium

    CAS:
    <p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>
    Fórmula:C23H14Na2O11
    Pureza:99.4% - 99.95%
    Forma y color:Colorless Crystals From Ethanol + Ether White Crystalline Powder
    Peso molecular:512.33
  • Linoleoyl glycine

    CAS:
    <p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>
    Fórmula:C20H35NO3
    Pureza:98.96%
    Forma y color:Solid
    Peso molecular:337.5
  • Glipizide

    CAS:
    <p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>
    Fórmula:C21H27N5O4S
    Pureza:99.67% - 99.75%
    Forma y color:Solid
    Peso molecular:445.54
  • Moxidectin

    CAS:
    <p>Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.</p>
    Fórmula:C37H53NO8
    Pureza:97.38%
    Forma y color:Appearance White Or Pale Yellow Amorphous Powder
    Peso molecular:639.82
  • Methocarbamol

    CAS:
    <p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>
    Fórmula:C11H15NO5
    Pureza:99.96%
    Forma y color:Crystals From Benzene Solid
    Peso molecular:241.24
  • Azosemide

    CAS:
    <p>Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).</p>
    Fórmula:C12H11ClN6O2S2
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:370.84