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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"

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  • Pilsicainide

    CAS:
    <p>Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].</p>
    Fórmula:C17H24N2O
    Forma y color:Solid
    Peso molecular:272.39
  • Levolansoprazole

    CAS:
    <p>Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).</p>
    Fórmula:C16H14F3N3O2S
    Pureza:98.629%
    Forma y color:Solid
    Peso molecular:369.36
  • Linerixibat

    CAS:
    <p>Linerixibat (GSK2330672) is a highly effective, nonabsorbable ASBT inhibitor. Linerixibat can lower glucose in an animal model of type 2 diabetes.</p>
    Fórmula:C28H38N2O7S
    Pureza:98.5% - 99.98%
    Forma y color:Solid
    Peso molecular:546.68
  • Verinurad

    CAS:
    <p>Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.</p>
    Fórmula:C20H16N2O2S
    Pureza:97.36% - 99.22%
    Forma y color:Solid
    Peso molecular:348.42
  • Imepitoin

    CAS:
    <p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>
    Fórmula:C13H14ClN3O2
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:279.72
  • MONNA

    CAS:
    <p>MONNA is a potent TMEM16A (Anoctamin-1) blocker (IC50 : 80 nM). It induces vasorelaxation of rodent resistance arteries in presence or absence of chloride ions.</p>
    Fórmula:C18H14N2O5
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:338.31
  • A-803467

    CAS:
    <p>A-803467 is a selective NaV1.8 channel blocker.</p>
    Fórmula:C19H16ClNO4
    Pureza:96.94% - 98%
    Forma y color:Solid
    Peso molecular:357.79
  • Vanilloid receptor antagonist 1

    CAS:
    <p>Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.</p>
    Fórmula:C18H15N3O2
    Pureza:98.14%
    Forma y color:Solid
    Peso molecular:305.33
  • Fenamic acid

    CAS:
    <p>Fenamic acid (N-Phenylanthranilic acid) is a chloride channel blocker that causes renal papillary necrosis in rats.</p>
    Fórmula:C13H11NO2
    Pureza:99.6%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:213.2319
  • AM92016

    CAS:
    <p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>
    Fórmula:C26H30Cl2N2O6S
    Forma y color:Solid
    Peso molecular:569.49
  • SB-366791

    CAS:
    <p>SB-366791 is a new and selective cinnamide TRPV1 antagonist.</p>
    Fórmula:C16H14ClNO2
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:287.74
  • Tiagabine hydrochloride hydrate

    CAS:
    <p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>
    Fórmula:C20H28ClNO3S2
    Forma y color:Solid
    Peso molecular:430.02
  • PPQ-102

    CAS:
    <p>PPQ-102 (CFTR Inhibitor), an effective CFTR inhibitor, can completely inhibit CFTR chloride current (IC50: 90 nM).</p>
    Fórmula:C26H22N4O3
    Pureza:99.7% - ≥95%
    Forma y color:Solid
    Peso molecular:438.48
  • Optovin

    CAS:
    <p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>
    Fórmula:C15H13N3OS2
    Pureza:99.47% - 99.67%
    Forma y color:Solid
    Peso molecular:315.41
  • VU6036720 hydrochloride


    <p>VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.</p>
    Fórmula:C20H23Cl2FN4O2S
    Forma y color:Solid
    Peso molecular:473.39
  • U93631

    CAS:
    <p>GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.</p>
    Fórmula:C17H21N3O2
    Pureza:99.65% - 99.76%
    Forma y color:Solid
    Peso molecular:299.37
  • AMTB hydrochloride

    CAS:
    <p>AMTB HCl: Novel TRPM8 blocker, relieves pain, treats urinary issues, moderates bladder reflexes in rats.</p>
    Fórmula:C23H27ClN2O2S
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:430.99
  • ML365

    CAS:
    <p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>
    Fórmula:C22H20N2O3
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:360.41
  • Azumolene sodium anhydrous

    CAS:
    <p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>
    Fórmula:C13H8BrN4NaO3
    Forma y color:Solid
    Peso molecular:371.13
  • Etripamil

    CAS:
    <p>Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.</p>
    Fórmula:C27H36N2O4
    Pureza:99.47% - 99.83%
    Forma y color:Solid
    Peso molecular:452.59
  • N-Me-aminopyrimidinone9

    CAS:
    <p>N-Me-aminopyrimidinone9 is a sodium channel antagonist</p>
    Fórmula:C16H21N3OS
    Pureza:99.21%
    Forma y color:Solid
    Peso molecular:303.42
  • Vocacapsaicin

    CAS:
    <p>Vocacapsaicin (CA-008), a prodrug of Capsaicin and a first-in-class non-opioid TRPV1 agonist, offers significant and enduring pain relief.</p>
    Fórmula:C26H41N3O4
    Forma y color:Solid
    Peso molecular:459.631
  • Rimeporide hydrochloride

    CAS:
    <p>Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>
    Fórmula:C11H16ClN3O5S2
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:369.84
  • Zoniporide hydrochloride hydrate

    CAS:
    <p>Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.</p>
    Fórmula:C17H19ClN6O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:374.83
  • SKA-31

    CAS:
    <p>SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).</p>
    Fórmula:C11H8N2S
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:200.26
  • Cariporide

    CAS:
    <p>Cariporide (HOE-642), an NHE1 inhibitor, reduces human platelet degranulation, platelet-leukocyte aggregates, and GPIIb/IIIa activation.</p>
    Fórmula:C12H17N3O3S
    Pureza:95.4% - 99.88%
    Forma y color:Solid
    Peso molecular:283.35
  • Thonzonium Bromide

    CAS:
    <p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>
    Fórmula:C32H55BrN4O
    Pureza:98.48% - 99.94%
    Forma y color:Solid
    Peso molecular:591.71
  • Polyoxyethylene stearate

    CAS:
    <p>Polyoxyethylene stearate (POES) is an agent of non-ionic emulsifying.</p>
    Fórmula:C20H40O3
    Pureza:n~9-10
    Forma y color:Light Amber Semisolid
    Peso molecular:328.29775
  • Nav1.8-IN-1

    CAS:
    <p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>
    Fórmula:C20H15ClF3N3O2
    Pureza:97.59%
    Forma y color:Solid
    Peso molecular:421.8
  • Zosuquidar trihydrochloride

    CAS:
    <p>Zosuquidar trihydrochloride (LY-335979 trihydrochloride) is a potent modulator of P-glycoprotein-mediated multi-drug resistance with Ki of 60 nM. Phase 3.</p>
    Fórmula:C32H31F2N3O2·3HCl
    Pureza:99.49% - >99.99%
    Forma y color:Solid
    Peso molecular:636.99
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Fórmula:C11H11N3O
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:201.22
  • Pirmenol

    CAS:
    <p>Pirmenol is a new antiarrhythmic drug</p>
    Fórmula:C22H30N2O
    Pureza:97.24%
    Forma y color:Solid
    Peso molecular:338.49
  • HBT1

    CAS:
    <p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>
    Fórmula:C16H17F3N4O2S
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:386.39
  • Tulrampator

    CAS:
    <p>Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.</p>
    Fórmula:C20H17FN4O3
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:380.37
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Fórmula:C17H24O4
    Pureza:98.22%
    Forma y color:Solid
    Peso molecular:292.37
  • ML133 hydrochloride

    CAS:
    <p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>
    Fórmula:C19H19NO·HCl
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:313.82
  • AZD3965

    CAS:
    <p>AZD3965 (AZD-3965) is a selective inhibitor of monocarboxylate transporter 1 (MCT1).</p>
    Fórmula:C21H24F3N5O5S
    Pureza:98% - 99.87%
    Forma y color:Solid
    Peso molecular:515.51
  • Chlorothymol

    CAS:
    <p>Chlorothymol (AI3-00120) is a disinfectant used in oral.</p>
    Fórmula:C10H13ClO
    Pureza:99.5%
    Forma y color:White Crystals Or Powder
    Peso molecular:184.66
  • Branaplam

    CAS:
    <p>Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.</p>
    Fórmula:C22H27N5O2
    Pureza:98.28% - 99.72%
    Forma y color:Solid
    Peso molecular:393.48
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Fórmula:C10H12ClNO2
    Pureza:97.20% - 98.94%
    Forma y color:Solid
    Peso molecular:213.66
  • CL 218872

    CAS:
    <p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>
    Fórmula:C13H9F3N4
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:278.23
  • ML-SA1

    CAS:
    <p>ML-SA1 (Mucolipin synthetic agonist 1) is a selective TRPML agonist, inhibits DENV2 and ZIKV by promoting lysosomal acidification and protease activity.</p>
    Fórmula:C22H22N2O3
    Pureza:99.34% - 99.71%
    Forma y color:Solid
    Peso molecular:362.42
  • WS-12

    CAS:
    <p>WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)</p>
    Fórmula:C18H27NO2
    Pureza:99.99%
    Forma y color:Whitish To White Solid Crystalline
    Peso molecular:289.41
  • Revaprazan

    CAS:
    <p>Revaprazan: novel, K⁺-competitive acid blocker; reversibly halts gastric H⁺/K⁺-ATPase; rivals PPIs in acid reduction.</p>
    Fórmula:C22H23FN4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:362.44
  • TGN-020

    CAS:
    <p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>
    Fórmula:C8H6N4OS
    Pureza:99.54% - 99.99%
    Forma y color:Solid
    Peso molecular:206.22
  • Ko 143

    CAS:
    <p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>
    Fórmula:C26H35N3O5
    Pureza:99.01% - 99.89%
    Forma y color:Solid
    Peso molecular:469.57
  • Tenatoprazole

    CAS:
    <p>Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM).</p>
    Fórmula:C16H18N4O3S
    Pureza:99.57%
    Forma y color:White Crystalline Powder
    Peso molecular:346.4
  • (E)-KPT330

    CAS:
    <p>(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.</p>
    Fórmula:C17H11F6N7O
    Pureza:98.69% - 99.49%
    Forma y color:Solid
    Peso molecular:443.31
  • H3B-120

    CAS:
    <p>H3B-120: selective, competitive CPS1 inhibitor with anti-cancer properties. IC50: 1.5 μM, Ki: 1.4 μM.</p>
    Fórmula:C19H24N4O2S
    Pureza:99.03% - 99.2%
    Forma y color:Solid
    Peso molecular:372.48
  • BZAD01

    CAS:
    <p>BZAD01 is a selective NMDA NR1A/2B receptor antagonist.</p>
    Fórmula:C16H12F6N2O
    Pureza:99.61% - 99.70%
    Forma y color:Solid
    Peso molecular:362.27
  • DHQ

    CAS:
    <p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>
    Fórmula:C8H6N2O2
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:162.15
  • Valbenazine

    CAS:
    <p>Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.</p>
    Fórmula:C24H38N2O4
    Pureza:97.58%
    Forma y color:Solid
    Peso molecular:418.57
  • ICA 110381

    CAS:
    <p>ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsy</p>
    Fórmula:C12H8Cl2N2O
    Pureza:97.72%
    Forma y color:Solid
    Peso molecular:267.11
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Fórmula:C6H6N2O2
    Pureza:99.94%
    Forma y color:Soild
    Peso molecular:138.1238
  • Guanosine 5'-diphosphate

    CAS:
    <p>Guanosine 5'-diphosphate (GDP) as Potential Iron Mobilizer, Preventing the Hepcidin-Ferroportin Interaction and Modulating the Interleukin-6/Stat-3 Pathway.</p>
    Fórmula:C10H15N5O11P2
    Pureza:98.46% - 99.52%
    Forma y color:Solid
    Peso molecular:443.2
  • M8-B Hydrochloride

    CAS:
    <p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>
    Fórmula:C22H25ClN2O3S
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:432.96
  • Rufinamide

    CAS:
    <p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>
    Fórmula:C10H8F2N4O
    Pureza:99.77% - >99.99%
    Forma y color:White Powder
    Peso molecular:238.19
  • Fosphenytoin disodium

    CAS:
    <p>Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blocker</p>
    Fórmula:C16H13N2Na2O6P
    Pureza:99.97%
    Forma y color:White Crystalline Powder
    Peso molecular:406.24
  • Phenyl benzoate

    CAS:
    <p>Phenyl benzoate is a benzoate ester obtained by the formal condensation of phenol with benzoic acid.It is an important organic synthesis intermediate.</p>
    Fórmula:C13H10O2
    Pureza:99.63%
    Forma y color:White Crystalline Powder
    Peso molecular:198.22
  • Chloroprocaine hydrochloride

    CAS:
    <p>Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.</p>
    Fórmula:C13H20Cl2N2O2
    Pureza:99.65%
    Forma y color:White Crystalline Powder
    Peso molecular:307.22
  • Vonoprazan fumarate

    CAS:
    <p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>
    Fórmula:C17H16FN3O2S·C4H4O4
    Pureza:99.16% - 99.98%
    Forma y color:Solid
    Peso molecular:461.46
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:354.38
  • Elobixibat hydrate

    CAS:
    <p>Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.</p>
    Fórmula:C36H47N3O8S2
    Forma y color:Solid
    Peso molecular:713.9
  • Revaprazan hydrochloride

    CAS:
    <p>Revaprazan hydrochloride (YH1885) is the hydrochloride salt form of a lipophilic, weak base with potassium-competitive acid blocking (P-CAB) activity.</p>
    Fórmula:C22H24ClFN4
    Pureza:99.62% - 99.91%
    Forma y color:Solid
    Peso molecular:398.9
  • NS 11021

    CAS:
    <p>NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channels</p>
    Fórmula:C16H9BrF6N6S
    Pureza:97.26%
    Forma y color:Solid
    Peso molecular:511.24
  • L-Phenylalanine-15N

    CAS:
    <p>L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.</p>
    Fórmula:C9H11NO2
    Pureza:98.98%
    Forma y color:Solid
    Peso molecular:166.18
  • Ilaprazole

    CAS:
    <p>Ilaprazole (IY-81149) is a proton pump inhibitor used in the treatment of dyspepsia gastroesophageal reflux disease (GORD/GERD) and duodenal ulcer.</p>
    Fórmula:C19H18N4O2S
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:366.44
  • Elacridar

    CAS:
    <p>Elacridar (GG918) is a potent inhibitor of P-glycoprotein and BCRP.Cost-effective and quality-assured.</p>
    Fórmula:C34H33N3O5
    Pureza:98.12% - >99.99%
    Forma y color:Solid
    Peso molecular:563.64
  • Lansoprazole sodium

    CAS:
    <p>Lansoprazole sodium is a PPI used to treat acid reflux and peptic ulcers.</p>
    Fórmula:C16H13F3N3NaO2S
    Pureza:99.14%
    Forma y color:Solid
    Peso molecular:391.34
  • DS-1971a

    CAS:
    <p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>
    Fórmula:C20H21ClFN5O3S
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:465.93
  • Tenatoprazole sodium

    CAS:
    <p>Tenatoprazole sodium is a potent proton pump inhibitor with an IC50 of 6.2 μM against hog gastric H+/K+-ATPase.</p>
    Fórmula:C16H17N4NaO3S
    Forma y color:Solid
    Peso molecular:368.39
  • 1-Aminocyclobutanecarboxylic acid

    CAS:
    <p>1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine site, NR1[1].</p>
    Fórmula:C5H9NO2
    Pureza:99.94%
    Forma y color:White To Tan Powder Crystals Crystalline Powder And/Or With Chunks
    Peso molecular:115.13
  • O4I2

    CAS:
    <p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>
    Fórmula:C12H11ClN2O2S
    Pureza:97.97% - 99.84%
    Forma y color:Solid
    Peso molecular:282.75
  • MDK-4025

    CAS:
    <p>MDK-4025 is an inhibitor of the high voltage-activated (HVA) Ca2+ current in pyramidal neurons.</p>
    Fórmula:C19H15ClO
    Pureza:98.65%
    Forma y color:Solid
    Peso molecular:294.77
  • AMG 333

    CAS:
    <p>AMG 333 is TRPM8 antagonist with an IC50 of 13 nM,a Clinical Candidate for the Treatment of Migraine.</p>
    Fórmula:C20H12F5N3O4
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:453.32
  • Efonidipine hydrochloride

    CAS:
    <p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>
    Fórmula:C34H39ClN3O7P
    Forma y color:Solid
    Peso molecular:668.12
  • Lorediplon

    CAS:
    <p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>
    Fórmula:C20H15FN4O2S
    Pureza:99.12% - 99.19%
    Forma y color:Solid
    Peso molecular:394.42
  • Phenibut (hydrochloride)

    CAS:
    <p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>
    Fórmula:C10H14ClNO2
    Pureza:99.93%
    Forma y color:White Crystalline Powder
    Peso molecular:215.68
  • (S)-(-)-5-Fluorowillardiine

    CAS:
    <p>(S)-(-)-5-Fluorowillardiine ((S)-5-Fluorowillardiine) is an AMPA receptor-specific agonist</p>
    Fórmula:C7H8FN3O4
    Pureza:99.69%
    Forma y color:Off-White Solid
    Peso molecular:217.15
  • Tirofiban hydrochloride monohydrate

    CAS:
    <p>Tirofiban(MK383) hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>
    Fórmula:C22H39ClN2O6S
    Pureza:98.81% - >99.99%
    Forma y color:White Solid
    Peso molecular:495.07
  • β-Pompilidotoxin Acetate


    <p>β-Pompilidotoxin Acetate is a wasp venom peptide.</p>
    Fórmula:C73H128N22O19
    Pureza:98.64%
    Forma y color:Solid
    Peso molecular:1617.93
  • L-Allylglycine

    CAS:
    <p>L-Allylglycine is a potent inhibitor of the synthetic enzyme for GABA, glutamic acid decarboxylase.</p>
    Fórmula:C5H9NO2
    Pureza:≥98%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:115.13
  • HC-056456

    CAS:
    <p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>
    Fórmula:C12H6N2O4S2
    Pureza:99.62% - 99.65%
    Forma y color:Solid
    Peso molecular:306.32
  • OAC3

    CAS:
    <p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>
    Fórmula:C15H11FN2O
    Pureza:97.13%
    Forma y color:Solid
    Peso molecular:254.26
  • Azimilide Dihydrochloride

    CAS:
    <p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>
    Fórmula:C23H30Cl3N5O3
    Pureza:97.59% - ≥95%
    Forma y color:Solid
    Peso molecular:530.88
  • QX-222 chloride

    CAS:
    <p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>
    Fórmula:C13H21ClN2O
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:256.77
  • Tiludronate

    CAS:
    <p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>
    Fórmula:C7H9ClO6P2S
    Forma y color:Solid
    Peso molecular:318.61
  • SB-705498

    CAS:
    <p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>
    Fórmula:C17H16BrF3N4O
    Pureza:99.57% - ≥95%
    Forma y color:Solid
    Peso molecular:429.23
  • Felbamate

    CAS:
    <p>Felbamate (W-554) is an Anti-epileptic Agent.</p>
    Fórmula:C11H14N2O4
    Pureza:99% - >99.99%
    Forma y color:White Powder Solid
    Peso molecular:238.24
  • L-DABA

    CAS:
    <p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 &gt; 500 μM).</p>
    Fórmula:C4H10N2O2
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:118.13
  • AMG9810

    CAS:
    <p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>
    Fórmula:C21H23NO3
    Pureza:99.79% - 99.95%
    Forma y color:Solid
    Peso molecular:337.41
  • ML213

    CAS:
    <p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>
    Fórmula:C17H23NO
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:257.37
  • TCN 213

    CAS:
    <p>TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2B</p>
    Fórmula:C18H24N4OS2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:376.54
  • Sepimostat dimethanesulfonate

    CAS:
    <p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>
    Fórmula:C23H27N5O8S2
    Forma y color:Solid
    Peso molecular:565.62
  • Levcromakalim

    CAS:
    <p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>
    Fórmula:C16H18N2O3
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:286.33
  • Flecainide acetate

    CAS:
    <p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>
    Fórmula:C19H24F6N2O5
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:474.39
  • NS6180

    CAS:
    <p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>
    Fórmula:C16H12F3NOS
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:323.33
  • Selamectin

    CAS:
    <p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>
    Fórmula:C43H63NO11
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:769.96
  • O4I1

    CAS:
    <p>O4I1 is an effective Oct3/4 inducer.</p>
    Fórmula:C16H15NO2
    Pureza:96.25% - 99.47%
    Forma y color:Solid
    Peso molecular:253.3
  • 9-Phenanthrol

    CAS:
    <p>9-Phenanthrol is inhibitor of the transient receptor potential melastatin 4 (TRPM) channel, a Ca2+ -activated non-selective cation channel.</p>
    Fórmula:C14H10O
    Pureza:98.48%
    Forma y color:Solid
    Peso molecular:194.23
  • Methyl homoveratrate

    CAS:
    <p>Methyl homoveratrate, a McN5691 (RWJ-26240) metabolite detected in vivo in plasma, urine, and fecal extracts, functions as a voltage-sensitive calcium channel</p>
    Fórmula:C11H14O4
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:210.23
  • MK6-83

    CAS:
    <p>MK6-83 is the transient receptor potential channel ML3 agonist.</p>
    Fórmula:C16H20N2O2S2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:336.47
  • VK-II-36

    CAS:
    <p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>
    Fórmula:C26H26N2O5
    Pureza:99.12%
    Forma y color:Solid
    Peso molecular:446.49
  • ICA-069673

    CAS:
    <p>ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).</p>
    Fórmula:C11H6ClF2N3O
    Pureza:99.04% - 99.68%
    Forma y color:Solid
    Peso molecular:269.63
  • Tricaine methanesulfonate

    CAS:
    <p>Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.</p>
    Fórmula:C10H15NO5S
    Pureza:99.259% - 99.86%
    Forma y color:White Powder
    Peso molecular:261.30
  • TKIM

    CAS:
    <p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>
    Fórmula:C18H14ClN3O2S
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:371.84
  • Budipine

    CAS:
    <p>Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.</p>
    Fórmula:C21H27N
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:293.45
  • SSD114 HCl

    CAS:
    <p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>
    Fórmula:C18H21ClF3N3O
    Pureza:99.03% - 99.95%
    Forma y color:Solid
    Peso molecular:387.83
  • 2'-O-Methylisoliquiritigenin

    CAS:
    <p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>
    Fórmula:C16H14O4
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:270.28
  • Saclofen

    CAS:
    <p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>
    Fórmula:C9H12ClNO3S
    Pureza:99.17%
    Forma y color:White Crystalline Solid
    Peso molecular:249.71
  • TRPM4-IN-1

    CAS:
    <p>TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.</p>
    Fórmula:C15H11Cl2NO4
    Pureza:97.22%
    Forma y color:Solid
    Peso molecular:340.16
  • BzATP triethylammonium salt

    CAS:
    <p>BzATP triethylammonium salt is a P2X7 receptor agonist.</p>
    Fórmula:C30H39N6O15P3
    Pureza:95% - 99.57%
    Forma y color:Solid
    Peso molecular:816.59
  • Bifemelane

    CAS:
    <p>Bifemelane, a nootropic, releases Ca2+ from stores and enables its entry via channels for astrocyte research.</p>
    Fórmula:C18H23NO
    Forma y color:Solid
    Peso molecular:269.38
  • YHO-13351

    CAS:
    <p>YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.</p>
    Fórmula:C27H37N3O7S2
    Pureza:97.88%
    Forma y color:Solid
    Peso molecular:579.73
  • AER-271

    CAS:
    <p>AER-271 is an inhibitor of aquaporin-4.</p>
    Fórmula:C15H9ClF6NO5P
    Pureza:97.45%
    Forma y color:Solid
    Peso molecular:463.65
  • Pico145

    CAS:
    <p>Pico145 (HC-608) is a remarkable inhibitor of TRPC1/4/5 channels.</p>
    Fórmula:C23H20ClF3N4O5
    Pureza:99.06%
    Forma y color:Solid
    Peso molecular:524.88
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Fórmula:C6H11NO3
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:145.16
  • Esomeprazole potassium salt

    CAS:
    <p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>
    Fórmula:C17H18KN3O3S
    Forma y color:Solid
    Peso molecular:383.51
  • 7-Chlorokynurenic acid sodium salt

    CAS:
    <p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>
    Fórmula:C10H6ClNNaO3
    Forma y color:Solid
    Peso molecular:246.6
  • Ilaprazole sodium

    CAS:
    <p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>
    Fórmula:C19H17N4NaO2S
    Pureza:99.06%
    Forma y color:Solid
    Peso molecular:388.42
  • Dotinurad

    CAS:
    <p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>
    Fórmula:C14H9Cl2NO4S
    Pureza:97.43% - 98.04%
    Forma y color:Solid
    Peso molecular:358.2
  • AC1903

    CAS:
    <p>AC1903 is a specific inhibitor of TRPC5 channel, and has been shown to suppress severe proteinuria and prevent podocyte loss.</p>
    Fórmula:C19H17N3O
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:303.36
  • Basmisanil

    CAS:
    <p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>
    Fórmula:C21H20FN3O5S
    Pureza:99.21% - 99.42%
    Forma y color:Solid
    Peso molecular:445.46
  • Ralfinamide

    CAS:
    <p>Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.</p>
    Fórmula:C17H19FN2O2
    Pureza:99.41%
    Forma y color:Solid
    Peso molecular:302.34
  • Homo-VK-II-36

    CAS:
    <p>Homo-VK-II-36 (Homo-V-II-36) is a carvedilol analogue that acts by inhibiting store- overload-induced calcium release through the RyR2 channel.</p>
    Fórmula:C27H28N2O5
    Pureza:99.26%
    Forma y color:Solid
    Peso molecular:460.52
  • Acamprosate calcium

    CAS:
    <p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>
    Fórmula:C10H20CaN2O8S2
    Pureza:98% - 99.93%
    Forma y color:White Odorless Or Nearly Odorless Powder
    Peso molecular:400.48
  • Quadrol

    CAS:
    <p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>
    Fórmula:C14H32N2O4
    Pureza:99.91% - 99.92%
    Forma y color:Viscous Liquid Liquid Viscous
    Peso molecular:292.41
  • S107

    CAS:
    <p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>
    Fórmula:C11H15NOS
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:209.31
  • Ocinaplon

    CAS:
    <p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>
    Fórmula:C17H11N5O
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:301.3
  • Quinine hydrobromide

    CAS:
    <p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>
    Fórmula:C20H25BrN2O2
    Forma y color:Solid
    Peso molecular:405.336
  • (-)-Blebbistatin

    CAS:
    <p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>
    Fórmula:C18H16N2O2
    Pureza:99.38% - 99.61%
    Forma y color:Solid
    Peso molecular:292.33
  • Vanillyl butyl ether

    CAS:
    <p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>
    Fórmula:C12H18O3
    Pureza:99.57%
    Forma y color:Yellowish Liquid Liquid
    Peso molecular:210.27
  • Metaflumizone

    CAS:
    <p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>
    Fórmula:C24H16F6N4O2
    Pureza:98.73%
    Forma y color:Solid
    Peso molecular:506.40
  • Esomeprazole hemistrontium

    CAS:
    <p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>
    Fórmula:C34H36N6O6S2Sr
    Forma y color:Solid
    Peso molecular:776.44
  • LY 303511 hydrochloride

    CAS:
    <p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>
    Fórmula:C19H19ClN2O2
    Pureza:98.47%
    Forma y color:Solid
    Peso molecular:342.82
  • NBI-98782

    CAS:
    <p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>
    Fórmula:C19H29NO3
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:319.44
  • ICA-121431

    CAS:
    <p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>
    Fórmula:C23H19N3O3S2
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:449.55
  • Ropivacaine hydrochloride monohydrate

    CAS:
    <p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>
    Fórmula:C17H29ClN2O2
    Pureza:99.94% - 99.95%
    Forma y color:White Solid
    Peso molecular:328.88
  • Arecaidine hydrochloride

    CAS:
    <p>Arecaidine hydrochloride may have carcinogenesis.</p>
    Fórmula:C7H12ClNO2
    Pureza:99.69% - ≥95%
    Forma y color:Solid
    Peso molecular:177.63
  • Cis-ACBD

    CAS:
    <p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>
    Fórmula:C6H9NO4
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:159.14
  • Neboglamine

    CAS:
    <p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>
    Fórmula:C13H24N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:256.34
  • Guan-fu base A hydrochloride(1394-48-5 free base)

    CAS:
    <p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>
    Fórmula:C24H32NO6Cl
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:465.97
  • Parimifasor

    CAS:
    <p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>
    Fórmula:C18H11Cl2F4N5O
    Pureza:96.77% - 98.97%
    Forma y color:Solid
    Peso molecular:460.21
  • Lansoprazole sulfone

    CAS:
    <p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>
    Fórmula:C16H14F3N3O3S
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:385.36
  • Ralfinamide mesylate

    CAS:
    <p>Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.</p>
    Fórmula:C18H23FN2O5S
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:398.45
  • A2793

    CAS:
    <p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>
    Fórmula:C13H12ClNO3
    Pureza:98.54%
    Forma y color:Solid
    Peso molecular:265.69
  • PF-06869206

    CAS:
    <p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>
    Fórmula:C15H14ClF3N4O2
    Pureza:99.79% - 99.88%
    Forma y color:Solid
    Peso molecular:374.75
  • Vonoprazan Fumarate

    CAS:
    <p>Vonoprazan Fumarate (TAK438) , a novel potassium-competitive acid blocker, inhibits gastric acid secretion.</p>
    Fórmula:C21H20FN3O6S
    Pureza:98.94%
    Forma y color:Solid
    Peso molecular:461.46
  • MDR-652

    CAS:
    <p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>
    Fórmula:C22H23ClFN3O2S
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:447.95
  • Kv2-IN-A1

    CAS:
    <p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>
    Fórmula:C20H17ClN4OS
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:396.89
  • Adjudin

    CAS:
    <p>Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.</p>
    Fórmula:C15H12Cl2N4O
    Pureza:96.51% - ≥95%
    Forma y color:Solid
    Peso molecular:335.19
  • Almitrine mesylate

    CAS:
    <p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>
    Fórmula:C28H37F2N7O6S2
    Pureza:99.96%
    Forma y color:Coa
    Peso molecular:669.76
  • KB-R7943 mesylate

    CAS:
    <p>KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.</p>
    Fórmula:C17H21N3O6S2
    Pureza:99.88% - ≥95%
    Forma y color:Solid
    Peso molecular:427.5
  • Eperisone hydrochloride

    CAS:
    <p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>
    Fórmula:C17H26ClNO
    Pureza:99.80%
    Forma y color:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter Taste
    Peso molecular:295.85
  • Miltirone

    CAS:
    <p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>
    Fórmula:C19H22O2
    Pureza:99.22% - 99.66%
    Forma y color:Solid
    Peso molecular:282.38
  • α-Asarone

    CAS:
    <p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>
    Fórmula:C12H16O3
    Pureza:99.64% - 99.64%
    Forma y color:Monoclinic Needles From Water Monoclinic Needles From Water
    Peso molecular:208.25
  • Levamlodipine hydrochloride

    CAS:
    <p>Levamlodipine hydrochloride is a medication used to lower blood pressure and prevent chest pain.</p>
    Fórmula:C20H26Cl2N2O5
    Forma y color:Solid
    Peso molecular:445.34
  • Baclofen hydrochloride

    CAS:
    <p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:250.122
  • Raxatrigine hydrochloride

    CAS:
    <p>Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.</p>
    Fórmula:C18H20ClFN2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:350.82
  • Ataluren

    CAS:
    <p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>
    Fórmula:C15H9FN2O3
    Pureza:99.16% - 99.84%
    Forma y color:Solid
    Peso molecular:284.24
  • Cyclothiazide

    CAS:
    <p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>
    Fórmula:C14H16ClN3O4S2
    Pureza:98.23% - 99.49%
    Forma y color:Crystals From Dilute Alcohol Solid
    Peso molecular:389.88
  • PF-05186462

    CAS:
    <p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>
    Fórmula:C19H10ClF4N5O3S2
    Pureza:99.10% - 99.37%
    Forma y color:Solid
    Peso molecular:531.89
  • Mitiglinide calcium hydrate

    CAS:
    <p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>
    Fórmula:C38H52CaN2O8
    Pureza:98.97% - 99.96%
    Forma y color:White Solid
    Peso molecular:704.91
  • Guanosine 5'-diphosphate disodium salt

    CAS:
    <p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>
    Fórmula:C10H13N5Na2O11P2
    Pureza:99.40%
    Forma y color:White Powder
    Peso molecular:487.16
  • CLP290

    CAS:
    <p>CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatric</p>
    Fórmula:C19H21FN4O3S
    Pureza:99.93% - >99.99%
    Forma y color:Solid
    Peso molecular:404.46
  • DAAO inhibitor-1

    CAS:
    <p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>
    Fórmula:C7H5FN2O
    Pureza:97.84%
    Forma y color:Solid
    Peso molecular:152.13
  • TRPM8 antagonist 2

    CAS:
    <p>TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.</p>
    Fórmula:C26H26N2O2
    Pureza:98.1%
    Forma y color:Solid
    Peso molecular:398.5
  • Amifampridine phosphate

    CAS:
    <p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>
    Fórmula:C5H10N3O4P
    Forma y color:Solid
    Peso molecular:207.12
  • Argireline

    CAS:
    <p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>
    Fórmula:C34H60N14O12S
    Pureza:96.79% - 99.65%
    Forma y color:White Powder
    Peso molecular:888.99
  • CFTR corrector 2

    CAS:
    <p>CFTR corrector 2 (FDL169) is a novel and potent CFTR corrector for treating cystic fibrosis (CF) patients who carry the F508del mutation.</p>
    Fórmula:C27H23FN4O4
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:486.49
  • N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride

    CAS:
    <p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>
    Fórmula:C16H17ClN4
    Pureza:99.25%
    Forma y color:Solid
    Peso molecular:300.79
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Fórmula:C10H12N2O3
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:208.21
  • KM11060

    CAS:
    <p>KM11060 is a novel corrector of the F508del-CFTR trafficking defect, Correcting F508del-CFTR trafficking, increasing the amount of functional CFTR at the plasma</p>
    Fórmula:C19H17Cl2N3O2S
    Pureza:98.86%
    Forma y color:Solid
    Peso molecular:422.33
  • Rimeporide

    CAS:
    <p>Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>
    Fórmula:C11H15N3O5S2
    Pureza:97.66%
    Forma y color:Solid
    Peso molecular:333.38
  • (R)-Lansoprazole

    CAS:
    <p>(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitor</p>
    Fórmula:C16H14F3N3O2S
    Pureza:98.09% - 98.99%
    Forma y color:Brown Solid
    Peso molecular:369.36
  • Cabotegravir

    CAS:
    <p>Cabotegravir (S/GSK1265744) (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (</p>
    Fórmula:C19H17F2N3O5
    Pureza:98.55% - 99.92%
    Forma y color:Solid
    Peso molecular:405.35
  • γ-Acetylenic GABA

    CAS:
    <p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>
    Fórmula:C6H9NO2
    Forma y color:Solid
    Peso molecular:127.143
  • PF-4840154

    CAS:
    <p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) &amp; 23 nM (human); triggers nociception in mice.</p>
    Fórmula:C26H38N6O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:466.62
  • DL-Willardiine

    CAS:
    <p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>
    Fórmula:C7H9N3O4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:199.16
  • Co 101244 hydrochloride

    CAS:
    <p>Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.</p>
    Fórmula:C21H28ClNO3
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:377.9
  • Procyclidine hydrochloride

    CAS:
    <p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>
    Fórmula:C19H30ClNO
    Pureza:99.24% - 99.88%
    Forma y color:Crystals From Petroleum Ether White Powder
    Peso molecular:323.9
  • CTP disodium dihydrate

    CAS:
    <p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>
    Fórmula:C9H18N3Na2O16P3
    Pureza:98.51%
    Forma y color:White Crystalline Powder
    Peso molecular:563.15
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Fórmula:C34H31F2N3O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:567.62
  • KPT185

    CAS:
    <p>KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.</p>
    Fórmula:C16H16F3N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:355.31
  • JNJ 303

    CAS:
    <p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>
    Fórmula:C21H29ClN2O4S
    Pureza:99.28%
    Forma y color:Solid
    Peso molecular:440.98
  • Anthracene-9-carboxylic acid

    CAS:
    <p>Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI.</p>
    Fórmula:C15H10O2
    Pureza:99.05%
    Forma y color:Yellow Cystalline Powder
    Peso molecular:222.24
  • FGH10019

    CAS:
    <p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>
    Fórmula:C18H19N3O2S2
    Pureza:98.93%
    Forma y color:Solid
    Peso molecular:373.49
  • Evenamide

    CAS:
    <p>Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.</p>
    Fórmula:C16H26N2O2
    Pureza:96.74% - 99.15%
    Forma y color:Solid
    Peso molecular:278.39
  • Trofinetide

    CAS:
    <p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>
    Fórmula:C13H21N3O6
    Pureza:98.70% - 99.50%
    Forma y color:Solid
    Peso molecular:315.32
  • Prilocaine

    CAS:
    <p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>
    Fórmula:C13H20N2O
    Pureza:98.49%
    Forma y color:Needles Solid
    Peso molecular:220.31
  • Transdermal Peptide Disulfide Acetate


    <p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>
    Fórmula:C42H68N14O18S2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:1121.2
  • 4-Chlorophenylguanidine hydrochloride

    CAS:
    <p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity.  </p>
    Fórmula:C7H9Cl2N3
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:206.07
  • HC067047 Hydrochloride(883031-03-6 free base)

    CAS:
    <p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>
    Fórmula:C26H29ClF3N3O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:507.98
  • Esomeprazole

    CAS:
    <p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>
    Fórmula:C17H19N3O3S
    Pureza:97.3%
    Forma y color:Solid
    Peso molecular:345.42
  • Epaminurad

    CAS:
    <p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>
    Fórmula:C14H10Br2N2O3
    Forma y color:Solid
    Peso molecular:414.05
  • ML335

    CAS:
    <p>ML335 is a selective activator of TREK-1 and TREK-2.</p>
    Fórmula:C15H14Cl2N2O3S
    Pureza:99.73% - 99.79%
    Forma y color:Solid
    Peso molecular:373.25
  • Glibenclamide potassium

    CAS:
    <p>Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.</p>
    Fórmula:C23H27ClKN3O5S
    Forma y color:Solid
    Peso molecular:532.09
  • JNJ-26990990

    CAS:
    <p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>
    Fórmula:C9H10N2O2S2
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:242.32
  • Isoflurane

    CAS:
    <p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>
    Fórmula:C3H2ClF5O
    Pureza:98%
    Forma y color:Clear Colorless Liquid Liquid
    Peso molecular:184.49
  • Bisaramil

    CAS:
    <p>Bisaramil is a new class I antiarrhythmic agent.</p>
    Fórmula:C17H23ClN2O2
    Forma y color:Solid
    Peso molecular:322.83