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Canal de potasio

Canal de potasio

Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.

Se han encontrado 276 productos de "Canal de potasio"

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  • B-TPMF

    CAS:
    <p>B-TPMF is a highly efficient and selective KCa2.1 channel inhibitor with an IC50 of 31 nM, interacting with serine residue at position 293 to inhibit KCa2.1.</p>
    Fórmula:C19H24N6O2
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:368.43
  • SCH-23390 maleate

    CAS:
    <p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>
    Fórmula:C21H22ClNO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:403.86
  • Vernakalant

    CAS:
    <p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>
    Fórmula:C20H31NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:349.46
  • CM-TPMF

    CAS:
    <p>CM-TPMF is a highly efficient and potent activator of the K(Ca)2.1 channel, Ser293 in the transmembrane segment 5, neurological disorders.</p>
    Fórmula:C16H17ClN6O2
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:360.8
  • HN37

    CAS:
    <p>HN37, KCNQ2 activator (EC50=37 nM). Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C20H21FN2O2
    Pureza:99.27%
    Forma y color:Solid
    Peso molecular:340.39
  • Pinacidil

    CAS:
    <p>Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and</p>
    Fórmula:C13H19N5
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:245.32
  • VU0405601

    CAS:
    <p>VU0405601 is a hERG channel activator that protects against drug-induced cardiac arrhythmias.</p>
    Fórmula:C17H13BrN2O2
    Pureza:99.16%
    Forma y color:Solid
    Peso molecular:357.2
  • Nifekalant hydrochloride

    CAS:
    <p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>
    Fórmula:C19H28ClN5O5
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:441.91
  • Almokalant

    CAS:
    <p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>
    Fórmula:C18H28N2O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.49
  • Aprikalim

    CAS:
    <p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>
    Fórmula:C12H16N2OS2
    Pureza:99.42% - 99.90%
    Forma y color:Solid
    Peso molecular:268.4
  • TWIK-1/TREK-1-IN-1

    CAS:
    <p>Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and</p>
    Fórmula:C21H24F3NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:395.42
  • AVE1231

    CAS:
    <p>AVE1231 is a TASK-1 channel blocker that inhibits TASK-1 and can be used in the study of atrial fibrillation.</p>
    Fórmula:C20H27N3O4S
    Pureza:98.03%
    Forma y color:Solid
    Peso molecular:405.51
  • GAL-021 sulfate

    CAS:
    <p>GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.</p>
    Fórmula:C11H24N6O5S
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:352.41
  • TRAM 39

    CAS:
    <p>TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.</p>
    Fórmula:C20H14ClN
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:303.78
  • RY796

    CAS:
    <p>RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.</p>
    Fórmula:C21H27N3O2
    Pureza:98.59%
    Forma y color:Solid
    Peso molecular:353.46
  • Psora 4

    CAS:
    <p>Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.</p>
    Fórmula:C21H18O4
    Forma y color:Solid
    Peso molecular:334.37
  • Vernakalant Hydrochloride

    CAS:
    <p>Vernakalant Hydrochloride (RSD1235 hydrochloride) is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel blocker.</p>
    Fórmula:C20H32ClNO4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:385.93
  • Amsacrine

    CAS:
    <p>Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.</p>
    Fórmula:C21H19N3O3S
    Pureza:99.2%
    Forma y color:Yellow Crystalline Powder Solid
    Peso molecular:393.46
  • DMP-543

    CAS:
    <p>DMP-543 (XR-543) is a potassium channel (KV7 channel) blocker that enhances the release of neurotransmitters.</p>
    Fórmula:C26H18F2N2O
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:412.43
  • TASK-1-IN-1

    CAS:
    <p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>
    Fórmula:C22H20N2O2
    Pureza:99.57%
    Forma y color:Soild
    Peso molecular:344.41