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Canal de potasio

Canal de potasio

Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.

Se han encontrado 276 productos de "Canal de potasio"

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  • KS176

    CAS:
    <p>KS176: selective BCRP inhibitor, potent against breast cancer drug resistance; ineffective on P-gp, MRP1.</p>
    Fórmula:C22H19N3O5
    Pureza:99.61% - 99.61%
    Forma y color:Solid
    Peso molecular:405.4
  • 5-Hydroxydecanoate sodium

    CAS:
    <p>5-Hydroxydecanoate sodium: KATP channel blocker, IC50 ~30μM; mitochondrial substrate; antioxidant.</p>
    Fórmula:C10H19NaO3
    Pureza:99.24% - 99.89%
    Forma y color:Solid
    Peso molecular:210.25
  • VU0810464

    CAS:
    <p>VU0810464 is a non-ureaG protein-gated inwardly-rectifying potassium channels (GIRK, Kir3) activator.</p>
    Fórmula:C18H21ClFN3O
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:349.83
  • Loureirin B

    CAS:
    <p>Loureirin B suppresses fibrosis by modulating MMPs/TIMPs, hindering fibroblast growth, and targeting TGF-β1/Smad2/3 pathway.</p>
    Fórmula:C18H20O5
    Pureza:99.33% - 99.86%
    Forma y color:Solid
    Peso molecular:316.35
  • Mitiglinide calcium hydrate

    CAS:
    <p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>
    Fórmula:C38H52CaN2O8
    Pureza:98.97% - 99.96%
    Forma y color:White Solid
    Peso molecular:704.91
  • A2793

    CAS:
    <p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>
    Fórmula:C13H12ClNO3
    Pureza:98.54%
    Forma y color:Solid
    Peso molecular:265.69
  • O-Nornuciferine

    CAS:
    <p>O-Nornuciferine reveals distinct in vitro hERG blockages measured in HEK293 cells with the IC50 value of 2.89 uM.</p>
    Fórmula:C18H19NO2
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:281.35
  • ML213

    CAS:
    <p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>
    Fórmula:C17H23NO
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:257.37
  • Levcromakalim

    CAS:
    <p>Levcromakalim (BRL 38227) is an activator of the ATP-sensitive K+ channel.</p>
    Fórmula:C16H18N2O3
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:286.33
  • NS 11021

    CAS:
    <p>NS 11021 (NS11021) , a novel opener of large-conductance Ca(2+)-activated K(+) channels</p>
    Fórmula:C16H9BrF6N6S
    Pureza:97.26%
    Forma y color:Solid
    Peso molecular:511.24
  • Tetraethylammonium bromide

    CAS:
    <p>Tetraethylammonium bromide (TEA bromide) can selectively block potassium channels.</p>
    Fórmula:C8H20BrN
    Pureza:98%
    Forma y color:White Solid
    Peso molecular:210.16
  • ML133 hydrochloride

    CAS:
    <p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>
    Fórmula:C19H19NO·HCl
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:313.82
  • SKF-96365 hydrochloride

    CAS:
    <p>SKF-96365 hydrochloride (SKF96365) , a SOCE inhibitor, exhibits potent anti-neoplastic activity by inducing cell-cycle arrest and apoptosis in colorectal Y</p>
    Fórmula:C22H27ClN2O3
    Pureza:99.47% - 99.92%
    Forma y color:Solid
    Peso molecular:402.91
  • Rimtuzalcap

    CAS:
    <p>Rimtuzalcap (CAD-1883), a selective modulator for SK channels, may treat movement disorders like SCA and ET.</p>
    Fórmula:C18H24F2N6O
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:378.42
  • A2764 dihydrochloride

    CAS:
    <p>A2764 dihydrochloride is a highly selective inhibitor of TRESK.</p>
    Fórmula:C15H21Cl3N2O
    Pureza:99.05%
    Forma y color:Solid
    Peso molecular:351.7
  • (±)-Naringenin

    CAS:
    <p>(±)-Naringenin (Naringenine) is a natural product.</p>
    Fórmula:C15H12O5
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:272.25
  • Dihydroberberine

    CAS:
    <p>Dihydroberberine has anti-atherosclerotic, anti-inflammatory, hypolipidemic and antitumor activities.</p>
    Fórmula:C20H19NO4
    Pureza:93.77%
    Forma y color:Solid
    Peso molecular:337.37
  • Nateglinide

    CAS:
    <p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>
    Fórmula:C19H27NO3
    Pureza:99.93% - 99.94%
    Forma y color:White Crystalline Powder
    Peso molecular:317.42
  • Guanosine 5'-diphosphate

    CAS:
    <p>Guanosine 5'-diphosphate (GDP) as Potential Iron Mobilizer, Preventing the Hepcidin-Ferroportin Interaction and Modulating the Interleukin-6/Stat-3 Pathway.</p>
    Fórmula:C10H15N5O11P2
    Pureza:98.46% - 99.52%
    Forma y color:Solid
    Peso molecular:443.2
  • ML 297

    CAS:
    <p>ML 297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator (IC50 values are 160, 887 and 914 nM for GIRK1/2, GIRK1/4 and GIRK1/3 respectively).</p>
    Fórmula:C17H14F2N4O
    Pureza:97.85%
    Forma y color:Solid
    Peso molecular:328.32