
Canal de potasio
Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.
Se han encontrado 327 productos para "Canal de potasio".
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Ropivacaine hydrochloride
CAS:Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activityFórmula:C17H26N2O·HClPureza:99.85% - 99.95%Forma y color:SolidPeso molecular:310.86Doxapram hydrochloride hydrate
CAS:Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.Fórmula:C24H33ClN2O3C24H30N2O2·ClH·H2OPureza:99.64% - >99.99%Forma y color:SolidPeso molecular:432.99Glibenclamide
CAS:Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.Fórmula:C23H28ClN3O5SPureza:99.05% - 99.75%Forma y color:White SolidPeso molecular:494DCPIB
CAS:DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μMFórmula:C22H28Cl2O4Pureza:99.77% - 99.79%Forma y color:SolidPeso molecular:427.36Ref: TM-T10979
2mg39,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg87,00€25mg177,00€50mg301,00€100mg485,00€200mg690,00€N-Acetylprocainamide
CAS:N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmicFórmula:C15H23N3O2Pureza:99.65% - 99.95%Forma y color:SolidPeso molecular:277.36VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuitFórmula:C20H22ClFN4O2SPureza:98.1%Forma y color:SolidPeso molecular:436.93Clofilium tosylate
CAS:Clofilium tosylate is a potassium channel blocker, induces apoptosis on human promyelocytic leukemia (HL-60) cells.Fórmula:C28H44ClNO3SPureza:99.61% - >99.99%Forma y color:White SolidPeso molecular:510.17Astemizole
CAS:Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.Fórmula:C28H31FN4OPureza:98.24% - 99.67%Forma y color:White Crystals SolidPeso molecular:458.57Glipizide
CAS:Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.Fórmula:C21H27N5O4SPureza:99.67% - 99.75%Forma y color:SolidPeso molecular:445.54Brompheniramine maleate
CAS:Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Forma y color:SolidPeso molecular:435.31NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Fórmula:C17H16ClN7Pureza:99.55%Forma y color:White SolidPeso molecular:353.81Mefloquine hydrochloride
CAS:Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.Fórmula:C17H17ClF6N2OPureza:99% - 99.99%Forma y color:SolidPeso molecular:414.77Dronedarone hydrochloride
CAS:Dronedarone hydrochloride (SR33589) is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.Fórmula:C31H44N2O5S·HClPureza:99.61%Forma y color:White SolidPeso molecular:593.22Ref: TM-T1073
5mg35,00€1mL*10mM (DMSO)49,00€10mg50,00€25mg82,00€50mg111,00€100mg166,00€200mg236,00€500mg403,00€IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFórmula:C31H32N4O2Pureza:98.9%Forma y color:SolidPeso molecular:492.61Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Fórmula:C16H16ClN3O3SPureza:98.97% - 99.83%Forma y color:SolidPeso molecular:365.83VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Fórmula:C20H32BrClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:447.84Ketanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Forma y color:SolidPeso molecular:395.4268Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Fórmula:C21H17ClF3N3O3Pureza:99.86%Forma y color:SolidPeso molecular:451.83Ref: TM-T15207
1mg58,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg166,00€25mg268,00€50mg403,00€100mg532,00€200mg705,00€Ropivacaine
CAS:Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.Fórmula:C17H26N2OPureza:97.75% - >99.99%Forma y color:SolidPeso molecular:274.40Tertiapin-Q
CAS:Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).Fórmula:C106H175N35O24S4Pureza:98.06% - 98.09%Forma y color:SolidPeso molecular:2452
