
Receptor CGRP
Los receptores de CGRP están involucrados en la transmisión del dolor y la regulación del flujo sanguíneo. El CGRP es un neuropéptido que desempeña un papel crucial en la fisiopatología de la migraña al dilatar los vasos sanguíneos y modular las vías de señalización del dolor. Dirigirse a los receptores de CGRP se ha convertido en un enfoque prometedor en el desarrollo de terapias para la migraña. En CymitQuimica, ofrecemos una gama de moduladores de receptores de CGRP para apoyar su investigación en el manejo del dolor, neurobiología y salud vascular.
Se han encontrado 55 productos de "Receptor CGRP"
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Erenumab
CAS:Erenumab: human antibody blocking CGRP receptors to prevent migraines.Pureza:99.43% (SEC-HPLC) - > 95%Forma y color:LiquidPeso molecular:146.2 kDaPHM-27 (human) acetate
PHM-27 (human) acetate is the endogenous peptide product of prepro-VIP (human), an agonist of the calcitonin receptor (EC 50 = 11 nM). enhanced insulin secretion.
Fórmula:C137H215F3N34O42SPureza:99.20%Forma y color:SoildPeso molecular:3099.44Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Fórmula:C84H130F3N25O23S2Forma y color:SolidPeso molecular:1979.21α-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Fórmula:C163H267N51O49S2Pureza:98%Forma y color:SolidPeso molecular:3789.33α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFórmula:C165H268F3N51O51S2Forma y color:SolidPeso molecular:3903.33CGRP antagonist 6
CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.Forma y color:Odour SolidAdrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Fórmula:C194H304N58O59S4Pureza:98%Forma y color:SolidPeso molecular:4521.17PHM-27 (human)
CAS:Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.Fórmula:C135H214N34O40SPureza:98%Forma y color:SolidPeso molecular:2985.44Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Fórmula:C163H267N51O50S2Pureza:98%Forma y color:SolidPeso molecular:3805.31HCGRP-(8-37)
CAS:Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonistFórmula:C139H230N44O38Pureza:98%Forma y color:SolidPeso molecular:3125.59Calcitonin (human)
CAS:Endogenous calcitonin receptor agonist. Lowers systemic blood calcium levels and inhibits bone resorption.Fórmula:C151H226N40O45S3Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:3417.87Adrenomedullin (16-31), human
CAS:Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Fórmula:C82H129N25O21S2Pureza:98%Forma y color:SolidPeso molecular:1865.19α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFórmula:C162H262N50O52S2Pureza:98%Forma y color:SolidPeso molecular:3806.25β-CGRP, human
CAS:β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascularFórmula:C162H267N51O48S3Pureza:98%Forma y color:SolidPeso molecular:3793.41(3R,5R,6S)-Atogepant
(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.Fórmula:C29H23F6N5O3Forma y color:SolidPeso molecular:603.52Adrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Fórmula:C248H381N77O75S5Pureza:98%Forma y color:SolidPeso molecular:5729.5Adrenomedullin (AM) (22-52), human TFA
Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.Fórmula:C161H253N46F3O50Pureza:98%Forma y color:SolidPeso molecular:3690.06Adrenomedullin (AM) (22-52), human
CAS:Adrenomedullin (ADM) is a 52-aa hypotensive peptide. Adrenomedullin (ADM) has structural similarity with amylin.Fórmula:C159H252N46O48Pureza:98%Forma y color:SolidPeso molecular:3576.04HTL22562
CAS:HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Fórmula:C40H49N11O5Forma y color:SolidPeso molecular:763.904Adrenotensin (human)
CAS:Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.Fórmula:C143H224N42O43Forma y color:SolidPeso molecular:3219.56

