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Canal de sodio

Canal de sodio

Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.

Se han encontrado 202 productos de "Canal de sodio"

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  • BI-9627

    CAS:
    <p>BI-9627 is an inhibitor of sodium-hydrogen exchanger isoform 1 (NHE1) (EC50: 31 nM).</p>
    Fórmula:C16H19F3N4O2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:356.34
  • Poneratoxin acetate


    <p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>
    Fórmula:C129H215N33O31S·xC2H4O2
    Forma y color:Solid
    Peso molecular:2756.35 (free base)
  • Ethacizine hydrochloride

    CAS:
    <p>Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.</p>
    Fórmula:C22H28ClN3O3S
    Pureza:98.08% - 98.08%
    Forma y color:Solid
    Peso molecular:449.99
  • Dibucaine hydrochloride

    CAS:
    <p>Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.</p>
    Fórmula:C20H30ClN3O2
    Pureza:99.66%
    Forma y color:White Powder
    Peso molecular:379.92
  • Bulleyaconitine A

    CAS:
    <p>Bulleyaconitine A, an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.</p>
    Fórmula:C35H49NO9
    Pureza:99.56% - 99.76%
    Forma y color:Solid
    Peso molecular:627.76
  • AM-2099

    CAS:
    <p>AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.</p>
    Fórmula:C19H13F3N4O3S2
    Forma y color:Solid
    Peso molecular:466.46
  • PF-04856264

    CAS:
    <p>PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.</p>
    Fórmula:C20H15N5O3S2
    Pureza:97.43%
    Forma y color:Solid
    Peso molecular:437.5
  • Mepivacaine

    CAS:
    <p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>
    Fórmula:C15H22N2O
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:246.35
  • Raxatrigine

    CAS:
    <p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>
    Fórmula:C18H19FN2O2
    Pureza:98% - 99.43%
    Forma y color:Solid
    Peso molecular:314.35
  • DS-1971a

    CAS:
    <p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>
    Fórmula:C20H21ClFN5O3S
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:465.93
  • A-803467

    CAS:
    <p>A-803467 is a selective NaV1.8 channel blocker.</p>
    Fórmula:C19H16ClNO4
    Pureza:96.94% - 98%
    Forma y color:Solid
    Peso molecular:357.79
  • Flecainide hydrochloride

    CAS:
    <p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>
    Fórmula:C17H21ClF6N2O3
    Pureza:97.79%
    Forma y color:Solid
    Peso molecular:450.81
  • Ropivacaine hydrochloride monohydrate

    CAS:
    <p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>
    Fórmula:C17H29ClN2O2
    Pureza:99.94% - 99.95%
    Forma y color:White Solid
    Peso molecular:328.88
  • Fosphenytoin disodium

    CAS:
    <p>Fosphenytoin disodium (ACC-9653) is a prodrug of phenytoin that is rapidly converted to phenytoin, a voltage-gated sodium channel blocker</p>
    Fórmula:C16H13N2Na2O6P
    Pureza:99.97%
    Forma y color:White Crystalline Powder
    Peso molecular:406.24
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:403.52
  • Rimeporide

    CAS:
    <p>Rimeporide (EMD-87580) (EMD-87580) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>
    Fórmula:C11H15N3O5S2
    Pureza:97.66%
    Forma y color:Solid
    Peso molecular:333.38
  • λ-Cyhalothrin

    CAS:
    <p>λ-Cyhalothrin (Icon) is a type II synthetic pyrethroid insecticide featuring a high-efficiency, broad-spectrum formula with an α-cyano group.</p>
    Fórmula:C23H19ClF3NO3
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:449.85
  • Flecainide acetate

    CAS:
    <p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>
    Fórmula:C19H24F6N2O5
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:474.39
  • Nicainoprol

    CAS:
    <p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>
    Fórmula:C21H27N3O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:369.46
  • Pilsicainide HCl

    CAS:
    <p>Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker</p>
    Fórmula:C17H25ClN2O
    Pureza:99.01% - 99.80%
    Forma y color:Solid
    Peso molecular:308.85