
Canal de sodio
Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.
Se han encontrado 202 productos de "Canal de sodio"
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Metaflumizone
CAS:<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Fórmula:C24H16F6N4O2Pureza:98.73%Forma y color:SolidPeso molecular:506.40Cyfluthrin
CAS:<p>Cyfluthrin binds to voltage-sensitive sodium channel such as Nav 1.8 sodium channel and modify their gating kinetics, thereby disrupting nerve function of pests</p>Fórmula:C22H18Cl2FNO3Pureza:99.76%Forma y color:SolidPeso molecular:434.29A-803467
CAS:<p>A-803467 is a selective NaV1.8 channel blocker.</p>Fórmula:C19H16ClNO4Pureza:96.94% - 98%Forma y color:SolidPeso molecular:357.79Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Forma y color:SolidPeso molecular:403.52Tenapanor
CAS:<p>Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.</p>Fórmula:C50H66Cl4N8O10S2Pureza:99.49% - 99.85%Forma y color:SolidPeso molecular:1145.05Dimethyl lithospermate B
CAS:<p>Dimethyl lithospermate B (dmLSB) is a selective Na+ channel agonist.</p>Fórmula:C38H34O16Pureza:98.34% - 99.62%Forma y color:SolidPeso molecular:746.67Eslicarbazepine Acetate
CAS:<p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>Fórmula:C17H16N2O3Pureza:99.58% - >99.99%Forma y color:White To Off-White SolidPeso molecular:296.32Nicainoprol
CAS:<p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>Fórmula:C21H27N3O3Pureza:99.54%Forma y color:SolidPeso molecular:369.46Sodium ionophore III
CAS:<p>Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.</p>Fórmula:C34H52N2O4Pureza:99.51% - 99.78%Forma y color:SolidPeso molecular:552.79BI 01383298
CAS:<p>BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).</p>Fórmula:C19H19Cl2FN2O3SPureza:99.71%Forma y color:SolidPeso molecular:445.34GS967
CAS:<p>GS967 is a potent, and selective inhibitor of cardiac late sodium current (late INa ).</p>Fórmula:C14H7F6N3OPureza:98% - >99.99%Forma y color:SolidPeso molecular:347.22Ranolazine
CAS:<p>Ranolazine (RS 43285-003) inhibits calcium uptake, treats chronic angina by targeting sodium/calcium channels to modulate intracellular sodium.</p>Fórmula:C24H33N3O4Pureza:98.13%Forma y color:White SolidPeso molecular:427.54AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Fórmula:C34H31F2N3O3Pureza:99.61%Forma y color:SolidPeso molecular:567.62RY785
CAS:<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Fórmula:C21H20N4O2SPureza:99.78%Forma y color:SolidPeso molecular:392.476-Benzoylheteratisine
CAS:<p>6-Benzoylheteratisine (Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth) is a Aconitum alkaloid.</p>Fórmula:C29H37NO6Pureza:99.87%Forma y color:SolidPeso molecular:495.61Benzonatate
CAS:<p>Benzonatate is an antagonist of sodium channel protein.</p>Fórmula:C30H53NO11Pureza:99.92%Forma y color:Colorless To Faintly Yellow Oil LiquidPeso molecular:603.74PF-06869206
CAS:<p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>Fórmula:C15H14ClF3N4O2Pureza:99.79% - 99.88%Forma y color:SolidPeso molecular:374.75Levobupivacaine hydrochloride
CAS:<p>Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.</p>Fórmula:C18H28N2O·HClPureza:99.74%Forma y color:White Crystalline PowderPeso molecular:324.893-Deoxyaconitine
CAS:<p>3- Deoxyaconitine is a derivative of Aconitine (A189875), which activates tetrodotoxin-sensitive Na+ channels, inducing presynaptic depolarization, thus</p>Fórmula:C34H47NO10Pureza:98.31%Forma y color:SolidPeso molecular:629.74Ralfinamide
CAS:<p>Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.</p>Fórmula:C17H19FN2O2Pureza:99.41%Forma y color:SolidPeso molecular:302.34
