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Canal de sodio

Canal de sodio

Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.

Se han encontrado 202 productos de "Canal de sodio"

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  • Metaflumizone

    CAS:
    <p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>
    Fórmula:C24H16F6N4O2
    Pureza:98.73%
    Forma y color:Solid
    Peso molecular:506.40
  • Cyfluthrin

    CAS:
    <p>Cyfluthrin binds to voltage-sensitive sodium channel such as Nav 1.8 sodium channel and modify their gating kinetics, thereby disrupting nerve function of pests</p>
    Fórmula:C22H18Cl2FNO3
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:434.29
  • A-803467

    CAS:
    <p>A-803467 is a selective NaV1.8 channel blocker.</p>
    Fórmula:C19H16ClNO4
    Pureza:96.94% - 98%
    Forma y color:Solid
    Peso molecular:357.79
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:403.52
  • Tenapanor

    CAS:
    <p>Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.</p>
    Fórmula:C50H66Cl4N8O10S2
    Pureza:99.49% - 99.85%
    Forma y color:Solid
    Peso molecular:1145.05
  • Dimethyl lithospermate B

    CAS:
    <p>Dimethyl lithospermate B (dmLSB) is a selective Na+ channel agonist.</p>
    Fórmula:C38H34O16
    Pureza:98.34% - 99.62%
    Forma y color:Solid
    Peso molecular:746.67
  • Eslicarbazepine Acetate

    CAS:
    <p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>
    Fórmula:C17H16N2O3
    Pureza:99.58% - >99.99%
    Forma y color:White To Off-White Solid
    Peso molecular:296.32
  • Nicainoprol

    CAS:
    <p>Nicainoprol (RU-42924) is a fast-sodium-channel blocking drug. Nicainoprol is a potent antiarrhythmic agent.</p>
    Fórmula:C21H27N3O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:369.46
  • Sodium ionophore III

    CAS:
    <p>Sodium ionophore III (ETH2120) is a Na+ ionophore suitable for the test of sodium activity in plasma, serum, and blood.</p>
    Fórmula:C34H52N2O4
    Pureza:99.51% - 99.78%
    Forma y color:Solid
    Peso molecular:552.79
  • BI 01383298

    CAS:
    <p>BI 01383298 is a selective inhibitor of the sodium-citrate co-transporter (SLC13A5).</p>
    Fórmula:C19H19Cl2FN2O3S
    Pureza:99.71%
    Forma y color:Solid
    Peso molecular:445.34
  • GS967

    CAS:
    <p>GS967 is a potent, and selective inhibitor of cardiac late sodium current (late INa ).</p>
    Fórmula:C14H7F6N3O
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:347.22
  • Ranolazine

    CAS:
    <p>Ranolazine (RS 43285-003) inhibits calcium uptake, treats chronic angina by targeting sodium/calcium channels to modulate intracellular sodium.</p>
    Fórmula:C24H33N3O4
    Pureza:98.13%
    Forma y color:White Solid
    Peso molecular:427.54
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Fórmula:C34H31F2N3O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:567.62
  • RY785

    CAS:
    <p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>
    Fórmula:C21H20N4O2S
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:392.47
  • 6-Benzoylheteratisine

    CAS:
    <p>6-Benzoylheteratisine (Heteratisan-14-one, 6-(benzoyloxy)-20-ethyl-8-hydroxy-1-methoxy-4-meth) is a Aconitum alkaloid.</p>
    Fórmula:C29H37NO6
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:495.61
  • Benzonatate

    CAS:
    <p>Benzonatate is an antagonist of sodium channel protein.</p>
    Fórmula:C30H53NO11
    Pureza:99.92%
    Forma y color:Colorless To Faintly Yellow Oil Liquid
    Peso molecular:603.74
  • PF-06869206

    CAS:
    <p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>
    Fórmula:C15H14ClF3N4O2
    Pureza:99.79% - 99.88%
    Forma y color:Solid
    Peso molecular:374.75
  • Levobupivacaine hydrochloride

    CAS:
    <p>Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) is a reversible neuronal sodium channel inhibitor, used as a long-acting local anesthetic.</p>
    Fórmula:C18H28N2O·HCl
    Pureza:99.74%
    Forma y color:White Crystalline Powder
    Peso molecular:324.89
  • 3-Deoxyaconitine

    CAS:
    <p>3- Deoxyaconitine is a derivative of Aconitine (A189875), which activates tetrodotoxin-sensitive Na+ channels, inducing presynaptic depolarization, thus</p>
    Fórmula:C34H47NO10
    Pureza:98.31%
    Forma y color:Solid
    Peso molecular:629.74
  • Ralfinamide

    CAS:
    <p>Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.</p>
    Fórmula:C17H19FN2O2
    Pureza:99.41%
    Forma y color:Solid
    Peso molecular:302.34