
Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 493 productos de "Canal de calcio"
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Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Fórmula:(C20H36N2O3S)2·C4H4O4Pureza:99.68% - 99.74%Forma y color:SolidPeso molecular:885.23Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Fórmula:C13H8BrN4NaO3Forma y color:SolidPeso molecular:371.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Fórmula:C34H60N14O12SPureza:96.79% - 99.65%Forma y color:White PowderPeso molecular:888.99TGR5 Receptor Agonist
CAS:<p>TGR5 is a potent TGR5(GPCR19) agonist.</p>Fórmula:C18H14Cl2N2O2Pureza:99.77% - ≥95%Forma y color:SolidPeso molecular:361.22Ethacrynic acid
CAS:<p>Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂,也是NF-κB 信号传导途径的有效抑制剂,并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道,从而导致气道平滑肌细胞松弛。它是利尿剂,具有抗炎特性,可减轻类维生素 A 诱导的小鼠耳部水肿。</p>Fórmula:C13H12Cl2O4Pureza:98.61% - 99.85%Forma y color:Crystals Physical Description White Solid (Ntp 1992)Peso molecular:303.14Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Fórmula:C21H25NO4Pureza:99.42% - 99.56%Forma y color:SolidPeso molecular:355.43HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Fórmula:C12H6N2O4S2Pureza:99.62% - 99.65%Forma y color:SolidPeso molecular:306.32Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Fórmula:C14H32N2O4Pureza:99.91% - 99.92%Forma y color:Viscous Liquid Liquid ViscousPeso molecular:292.41Mirogabalin
CAS:<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Fórmula:C12H19NO2Pureza:98.57%Forma y color:SolidPeso molecular:209.28Efonidipine hydrochloride
CAS:<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Fórmula:C34H39ClN3O7PForma y color:SolidPeso molecular:668.12NP118809
CAS:<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Fórmula:C32H32N2OPureza:97.74% - 98.68%Forma y color:SolidPeso molecular:460.61Praeruptorin C
CAS:<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Fórmula:C24H28O7Pureza:99.6% - 99.92%Forma y color:SolidPeso molecular:428.47CDN1163
CAS:<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Fórmula:C20H20N2O2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:320.39ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Fórmula:C20H21Cl2F2N3O3SForma y color:SolidPeso molecular:492.36Pyr6
CAS:<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Fórmula:C17H9F7N4OPureza:98.89%Forma y color:SolidPeso molecular:418.27Gabapentin hydrochloride
CAS:<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Fórmula:C9H17NO2·HClPureza:99.71%Forma y color:Off-White SolidPeso molecular:207.7Pinaverium bromide
CAS:<p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>Fórmula:C26H41Br2NO4Pureza:99.52%Forma y color:White Crystalline PowderPeso molecular:591.42Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Fórmula:C26H44NNaO5SPureza:99.79% - 99.93%Forma y color:SolidPeso molecular:505.69FPL64176
CAS:<p>FPL64176 is a L-type calcium channels activator.</p>Fórmula:C22H21NO3Pureza:98.68%Forma y color:SolidPeso molecular:347.41
