Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 493 productos de "Canal de calcio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Nicardipine-d3 hydrochloride
CAS:<p>Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.</p>Fórmula:C26H30ClN3O6Pureza:98%Forma y color:SolidPeso molecular:519YM-244769 dihydrochloride
CAS:<p>YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.</p>Fórmula:C26H24Cl2FN3O3Pureza:98%Forma y color:SolidPeso molecular:516.39HSK16149
CAS:<p>HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.</p>Fórmula:C12H19NO2Forma y color:SolidPeso molecular:209.28MRS1845
CAS:<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Fórmula:C21H22N2O6Pureza:99.69%Forma y color:SolidPeso molecular:398.41(S)-Nicardipine
CAS:<p>(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).</p>Fórmula:C26H29N3O6Forma y color:SolidPeso molecular:479.53Almorexant hydrochloride
CAS:<p>Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.</p>Fórmula:C29H32ClF3N2O3Pureza:99.85%Forma y color:SolidPeso molecular:549.02Norverapamil-d7
CAS:<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Fórmula:C26H36N2O4Pureza:98%Forma y color:SolidPeso molecular:447.62Hexadecylphosphoserine TFA
<p>Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.</p>Fórmula:C21H41F3NO8PForma y color:SolidPeso molecular:523.52Dronedarone
CAS:<p>Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.</p>Fórmula:C31H44N2O5SPureza:98.85% - 99.58%Forma y color:SolidPeso molecular:556.76Azumolene
CAS:<p>Azumolene (EU4093 free base)</p>Fórmula:C13H9BrN4O3Pureza:98.1% - 98.35%Forma y color:SolidPeso molecular:349.14Ginsenoside Rd
CAS:<p>Ginsenoside Rd (Gypenoside VIII) may have properties that inhibit or prevent the growth of tumors.</p>Fórmula:C48H82O18Pureza:99.13% - 99.92%Forma y color:SolidPeso molecular:947.15JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Fórmula:C9H10N2O2S2Pureza:97.37%Forma y color:SolidPeso molecular:242.32Efonidipine
CAS:<p>Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.</p>Fórmula:C34H38N3O7PPureza:98.35% - 99.47%Forma y color:SolidPeso molecular:631.66Bepridil hydrochloride
CAS:<p>Bepridil hydrochloride (CERM 1978) is a calcium channel blocker and also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels</p>Fórmula:C24H35ClN2OPureza:99.45% - 99.68%Forma y color:SolidPeso molecular:4032,5-Di-tert-butylhydroquinone
CAS:<p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>Fórmula:C14H22O2Pureza:97.11%Forma y color:PelletslargecrystalsPeso molecular:222.32DHBP dibromide
CAS:<p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>Fórmula:C24H38Br2N2Pureza:99.73%Forma y color:Yellow To Yellow-Green Powder Or FlakesPeso molecular:514.38L-Phenylalanine
CAS:<p>L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.</p>Fórmula:C9H11NO2Pureza:99.37% - 99.87%Forma y color:Solid CrystallinePeso molecular:165.19GSK1016790A
CAS:<p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>Fórmula:C28H32Cl2N4O6S2Pureza:97.37% - 99.38%Forma y color:SolidPeso molecular:655.61Propiverine hydrochloride
CAS:<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Fórmula:C23H30ClNO3Pureza:99.93%Forma y color:White Crystalling PowerPeso molecular:403.94Dantrolene sodium hemiheptahydrate
CAS:<p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>Fórmula:C14H9N4NaO5·5H2OPureza:99.72%Forma y color:Orange PowderPeso molecular:399.29Pranidipine
CAS:<p>Pranidipine (OPC-13340) is a novel, long-acting 1,4-dihydropyridine calcium channel blocker.</p>Fórmula:C25H24N2O6Pureza:99.95%Forma y color:Yellow SolidPeso molecular:448.47Aranidipine
CAS:<p>Aranidipine (MPC1304) (MPC1304) is a calcium channel antagonist with potent and long-lasting antihypertensive effects.</p>Fórmula:C19H20N2O7Pureza:99.15%Forma y color:SolidPeso molecular:388.37(±)-Praeruptorin A
CAS:<p>(±)-Praeruptorin A could exhibit its anti-osteoclastogenic activity by inhibiting p38/Akt-c-Fos-NFATc1 signaling and PLCγ-independent Ca(2+) oscillation.</p>Fórmula:C21H22O7Pureza:98.9% - 99.73%Forma y color:SolidPeso molecular:386.4(+)-Kavain
CAS:<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Fórmula:C14H14O3Pureza:97% - ≥95%Forma y color:White Fine PowderPeso molecular:230.26Suvecaltamide
CAS:<p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>Fórmula:C20H23F3N2O2Pureza:99.29% - 99.70%Forma y color:SolidPeso molecular:380.4NS-638
CAS:<p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>Fórmula:C15H11ClF3N3Pureza:98.44%Forma y color:SolidPeso molecular:325.72NFAT Inhibitor-2
CAS:<p>NFAT Inhibitor-2 is a compound used as a molecular building block.</p>Fórmula:C22H20F2N2O4SPureza:97.37%Forma y color:SolidPeso molecular:446.47Efonidipine hydrochloride monoethanolate
CAS:<p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>Fórmula:C36H45ClN3O8PPureza:>99.99%Forma y color:SolidPeso molecular:714.18Praeruptorin E
CAS:<p>Praeruptorin C/E relaxes arteries, reduces heart contractility, acting like calcium blockers. D/E protect mice from acid lung injury by halting PMNs and IL-6.</p>Fórmula:C24H28O7Pureza:98.04% - 99.95%Forma y color:SolidPeso molecular:428.47SR33805
CAS:<p>SR33805 is a potent antagonist of Ca2+ channel(EC50s of 4.1 nM and 33 nM in depolarized and polarized conditions, respectively)</p>Fórmula:C32H40N2O5SPureza:99.15%Forma y color:SolidPeso molecular:564.74Ibutilide Fumarate
CAS:<p>Ibutilide Fumarate is a class III antiarrhythmic, prolonging action potentials by enhancing sodium influx, and can extend QT interval.</p>Fórmula:(C20H36N2O3S)2·C4H4O4Pureza:99.68% - 99.74%Forma y color:SolidPeso molecular:885.23Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Fórmula:C13H8BrN4NaO3Forma y color:SolidPeso molecular:371.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Fórmula:C34H60N14O12SPureza:96.79% - 99.65%Forma y color:White PowderPeso molecular:888.99TGR5 Receptor Agonist
CAS:<p>TGR5 is a potent TGR5(GPCR19) agonist.</p>Fórmula:C18H14Cl2N2O2Pureza:99.77% - ≥95%Forma y color:SolidPeso molecular:361.22Ethacrynic acid
CAS:<p>Ethacrynic acid (Edecrin) 是谷胱甘肽 S-转移酶抑制剂，也是NF-κB 信号传导途径的有效抑制剂，并且还调节白三烯的形成。它还可抑制 L 型电压依赖性和储存操作的钙通道，从而导致气道平滑肌细胞松弛。它是利尿剂，具有抗炎特性，可减轻类维生素 A 诱导的小鼠耳部水肿。</p>Fórmula:C13H12Cl2O4Pureza:98.61% - 99.85%Forma y color:Crystals Physical Description White Solid (Ntp 1992)Peso molecular:303.14Glaucine
CAS:<p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>Fórmula:C21H25NO4Pureza:99.42% - 99.56%Forma y color:SolidPeso molecular:355.43HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Fórmula:C12H6N2O4S2Pureza:99.62% - 99.65%Forma y color:SolidPeso molecular:306.32Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Fórmula:C14H32N2O4Pureza:99.91% - 99.92%Forma y color:Viscous Liquid Liquid ViscousPeso molecular:292.41Mirogabalin
CAS:<p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>Fórmula:C12H19NO2Pureza:98.57%Forma y color:SolidPeso molecular:209.28Efonidipine hydrochloride
CAS:<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Fórmula:C34H39ClN3O7PForma y color:SolidPeso molecular:668.12NP118809
CAS:<p>NP118809 (39-1B4) is a potent N-type calcium channel blocker(IC50 : 0.11 μM).</p>Fórmula:C32H32N2OPureza:97.74% - 98.68%Forma y color:SolidPeso molecular:460.61Praeruptorin C
CAS:<p>Praeruptorin C: an antioxidant, calcium antagonist, protects neurons, reduces vascular hypertrophy, affects cellular signals.</p>Fórmula:C24H28O7Pureza:99.6% - 99.92%Forma y color:SolidPeso molecular:428.47CDN1163
CAS:<p>CDN1163 is a small molecule activator of sarco/endoplasmic reticulum Ca2+-ATPase (SERCA).</p>Fórmula:C20H20N2O2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:320.39ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Fórmula:C20H21Cl2F2N3O3SForma y color:SolidPeso molecular:492.36Pyr6
CAS:<p>Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influx</p>Fórmula:C17H9F7N4OPureza:98.89%Forma y color:SolidPeso molecular:418.27Gabapentin hydrochloride
CAS:<p>Gabapentin hydrochloride (Neurontin HCl) is a GABA analogue, used to treat seizures and neuropathic pain.</p>Fórmula:C9H17NO2·HClPureza:99.71%Forma y color:Off-White SolidPeso molecular:207.7Pinaverium bromide
CAS:<p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>Fórmula:C26H41Br2NO4Pureza:99.52%Forma y color:White Crystalline PowderPeso molecular:591.42Taurolithocholic acid sodium salt
CAS:<p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>Fórmula:C26H44NNaO5SPureza:99.79% - 99.93%Forma y color:SolidPeso molecular:505.69FPL64176
CAS:<p>FPL64176 is a L-type calcium channels activator.</p>Fórmula:C22H21NO3Pureza:98.68%Forma y color:SolidPeso molecular:347.41
