Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 493 productos de "Canal de calcio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Gallopamil, (-)-
CAS:<p>Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>Fórmula:C28H40N2O5Pureza:98%Forma y color:SolidPeso molecular:484.63AK-2-38
CAS:<p>AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.</p>Fórmula:C26H30N2O4Pureza:98%Forma y color:SolidPeso molecular:434.53Falipamil
CAS:<p>Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.</p>Fórmula:C24H32N2O5Pureza:98%Forma y color:SolidPeso molecular:428.52Tiropramide
CAS:<p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>Fórmula:C28H41N3O3Pureza:98%Forma y color:SolidPeso molecular:467.64Bms 188107
CAS:<p>Bms 188107 is a calcium antagonist, it has cardioprotective effects.</p>Fórmula:C25H26N2O4Pureza:98%Forma y color:SolidPeso molecular:418.48AZD 2066
CAS:<p>AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.</p>Fórmula:C19H16ClN5O2Pureza:98%Forma y color:SolidPeso molecular:381.82BBR 2160
CAS:<p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>Fórmula:C21H25N3O7SForma y color:SolidPeso molecular:463.5DS16570511
CAS:<p>DS16570511 is a novel, cell-permeable inhibitor targeting the mitochondrial calcium uniporter.</p>Fórmula:C30H25Cl2N3O4Pureza:98.34% - 98.45%Forma y color:SolidPeso molecular:562.44Tamolarizine
CAS:<p>Tamolarizine (Tamolarizine free base) free base is a novel calcium antagonist.</p>Fórmula:C27H32N2O3Pureza:98.17%Forma y color:SoildPeso molecular:432.55Tiapamil hydrochloride
CAS:<p>Tiapamil hydrochloride (Ro 11-1781 hydrochloride) is a calcium channel blocker with antihypertensive activity used in the study of angina pectoris.</p>Fórmula:C26H38ClNO8S2Pureza:99.17%Forma y color:SolidPeso molecular:592.16R 56865
CAS:<p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>Fórmula:C23H28FN3OSPureza:99.52%Forma y color:SolidPeso molecular:413.55Enecadin
CAS:<p>Enecadin is a neuroprotective agent.</p>Fórmula:C21H28FN3OPureza:98.53%Forma y color:SolidPeso molecular:357.46Clopimozide
CAS:<p>Clopimozide (R-29764), a long-acting oral antischizophrenic, blocks calcium channels and [3H] nilandipine binding.</p>Fórmula:C28H28ClF2N3OPureza:98.19% - >99.99%Forma y color:SolidPeso molecular:495.99GSK205
CAS:<p>GSK205 is a selective TRPV4 antagonist (IC50: 4.19 μM) for inhibiting TRPV4-mediated Ca2+ influx.</p>Fórmula:C24H25BrN4SPureza:99.46%Forma y color:SolidPeso molecular:481.45SAK3
CAS:<p>SAK3 is a modulator of nAChR activity and is used to study memory deficits and Alzheimer's disease.</p>Fórmula:C20H23N3O4Pureza:98.37% - 99.43%Forma y color:SolidPeso molecular:369.418-Bromo-cGMP sodium
CAS:<p>8-Bromo-cGMP sodium: PKG activator, eases pain, dilates vessels, reduces Ca2+ currents & insulin release.</p>Fórmula:C10H10BrN5NaO7PPureza:99.45%Forma y color:SolidPeso molecular:446.09Gallopamil
CAS:<p>Gallopamil blocks acid secretion (IC50: 10.9 μM), acts as antiarrhythmic, vasodilator, and is a methoxy Verapamil derivative.</p>Fórmula:C28H40N2O5Pureza:99.85%Forma y color:SolidPeso molecular:484.63Cronidipine
CAS:<p>Cronidipine (LF 20254), a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>Fórmula:C30H32ClN3O8Pureza:99.47%Forma y color:SolidPeso molecular:598.04Upacicalcet
CAS:<p>Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.</p>Fórmula:C11H14ClN3O6SPureza:99.83%Forma y color:SolidPeso molecular:351.76Vatanidipine
CAS:<p>Vatanidipine (AE0047) is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.A slow-onset and long-lasting</p>Fórmula:C41H42N4O6Pureza:99.95%Forma y color:SolidPeso molecular:686.8Sulcardine sulfate
CAS:<p>Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, and Ca2+ channels.</p>Fórmula:C24H35N3O8S2Pureza:98.74%Forma y color:SolidPeso molecular:557.68O-1602
CAS:<p>O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatment</p>Fórmula:C17H22O2Pureza:99.85%Forma y color:SolidPeso molecular:258.36VU 0240551
CAS:<p>VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.</p>Fórmula:C16H14N4OS2Pureza:99.9%Forma y color:SolidPeso molecular:342.44SERCA2a activator 1
CAS:<p>SERCA2a activator 1 boosts heart function by reducing phospholamban restraint and enhancing cardiac contraction-relaxation cycles.</p>Fórmula:C32H29N3O4SPureza:99.75%Forma y color:SolidPeso molecular:551.66CERM-11956
CAS:<p>Pelretin (BASF 43915) is a potential protein inhibitor for the study of dermatologic diseases.</p>Fórmula:C29H38N2O7Pureza:99.38%Forma y color:SolidPeso molecular:526.62Ticolubant
CAS:<p>Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.</p>Fórmula:C23H19Cl2NO3SPureza:99.59%Forma y color:SolidPeso molecular:460.37CP-060
CAS:<p>CP-060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.</p>Fórmula:C30H42N2O5SPureza:99.54%Forma y color:SolidPeso molecular:542.73PD173212
CAS:<p>PD 173212 is a blocker that blocks N-type voltage sensitive calcium channel (Cav2.2).</p>Fórmula:C38H53N3O3Pureza:99.84%Forma y color:SolidPeso molecular:599.85Terflavoxate
CAS:<p>Terflavoxate is a novel, orally active, semisynthetic statin microtubule inhibitor commonly used in combination with capecitabine.</p>Fórmula:C26H29NO4Pureza:98%Forma y color:SolidPeso molecular:419.51Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Fórmula:C26H35F2NO7Pureza:99.71%Forma y color:SolidPeso molecular:511.56Fenoverine
CAS:<p>Fenoverine (Spasmopriv) has antispasmodic activity and can be used to study gastrointestinal spasms.</p>Fórmula:C26H25N3O3SPureza:98.34%Forma y color:SolidPeso molecular:459.56NecroX-5
CAS:<p>NecroX-5, a derivative of NecroX, exhibits anti-inflammatory and anti-cancer activities. NecroX-5 reduces intracellular calcium concentration.</p>Fórmula:C27H39N3O9S3Pureza:99.944%Forma y color:SolidPeso molecular:645.81Diproteverine HCl
CAS:<p>Diproteverine HCl is a novel calcium antagonist with antianginal properties, antispasmodic and vasoactive.</p>Fórmula:C26H36ClNO4Pureza:98.55% - 99.84%Forma y color:SolidPeso molecular:462.02Opc 8490
CAS:<p>Opc 8490 is a cardiotonic agent and a positive inotropic vasodilator, which prolongs the atrial action potential in a concentration-dependent manner.</p>Fórmula:C30H35N3O10Pureza:98.88%Forma y color:SolidPeso molecular:597.61Lifarizine
CAS:<p>Lifarizine (RS-87476), a calcium-sodium channel antagonist, shows neuroprotective activity in a simplified rat survival model of double vessel occlusion.</p>Fórmula:C29H32N4Pureza:99.88%Forma y color:SolidPeso molecular:436.59AZD-1305
CAS:<p>AZD-1305: novel anti-arrhythmic blocking IKr, Ca, Na currents; useful in arrhythmia research.</p>Fórmula:C22H31FN4O4Pureza:99.31% - 99.86%Forma y color:SolidPeso molecular:434.5N106
CAS:<p>N106 is an activator of the SUMO-activating enzyme, E1 ligase, and triggers intrinsic sumoylation of SERCA2a. N106 can be used in studies about heart failure.</p>Fórmula:C17H14N4O3SPureza:99.69%Forma y color:SolidPeso molecular:354.38Crobenetine
CAS:<p>Crobenetine (BIII 890 CL) Free Base is a selective NaV channel blocker that eliminates VTD-induced [Ca2+] elevation.</p>Fórmula:C25H33NO2Pureza:98.99%Forma y color:SolidPeso molecular:379.54Mioflazine
CAS:<p>Mioflazine suppresses nucleoside uptake. Mioflazine is an orally active nucleoside transport inhibitor. It has the potential for sleep disorders treatment.</p>Fórmula:C29H30Cl2F2N4O2Pureza:98%Forma y color:SolidPeso molecular:575.48Iganidipine
CAS:<p>Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.</p>Fórmula:C28H38N4O6Pureza:96.3%Forma y color:SolidPeso molecular:526.62RS 5773
CAS:<p>RS 5773 is a benzothiazepine derivative with antianginal effects.</p>Fórmula:C29H33ClN2O4SPureza:98%Forma y color:SolidPeso molecular:541.1Budiodarone
CAS:<p>Budiodarone (ATI-2042) resembles amiodarone, potentially preventing atrial fibrillation.</p>Fórmula:C27H31I2NO5Forma y color:SolidPeso molecular:703.35Coelenterazine h
CAS:<p>Coelenterazine H, a Ca2+ sensitive synthetic derivative, is a luminescent biomolecule used to measure Ca2+ changes.</p>Fórmula:C26H21N3O2Pureza:99.49%Forma y color:Yellow To Brownish PowderPeso molecular:407.46TROX-1
CAS:<p>TROX-1 is the activation state-dependent Cav2 channel antagonist.</p>Fórmula:C22H16ClFN6OPureza:98%Forma y color:SolidPeso molecular:434.85Piprofurol
CAS:<p>Piprofurol is used as a Calcium channel blocker.</p>Fórmula:C26H33NO6Pureza:98%Forma y color:SolidPeso molecular:455.54A 425619
CAS:<p>A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) is a potent TRPV1 antagonist</p>Fórmula:C18H14F3N3OPureza:99.75%Forma y color:SolidPeso molecular:345.32Cavα2δ1&NET-IN-3
CAS:<p>Cavα2δ1&NET-IN-3 (example 216) is an inhibitor targeting both the α2δ subunit of voltage-gated calcium channels (VGCC) and the noradrenaline transporter (NET).</p>Fórmula:C24H30N6O2SForma y color:SolidPeso molecular:466.6N-type calcium channel blocker-1
CAS:<p>N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.</p>Fórmula:C31H47N3Pureza:98%Forma y color:SolidPeso molecular:461.73(S)-(-)-Bay-K-8644
CAS:<p>(S)-(-)-Bay-K-8644 ((S)-(-)-Bay K 8644) is an agonist of L-type Ca2+ channel and activates Ba2+ currents with an EC50 of 32 nM.</p>Fórmula:C16H15F3N2O4Pureza:98.28% - 99.37%Forma y color:SolidPeso molecular:356.3KCa1.1 channel activator-1
<p>A selective vascular KCa1.1 channel stimulator with CaV1.2 blocking ability and mild myorelaxant effects.</p>Fórmula:C25H16O10Forma y color:SolidPeso molecular:476.39
