
Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 563 productos de "Canal de calcio"
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Ro 18-3981
CAS:Ro 18-3981 inhibits myocardial Ca2+ channels; KD is 1.0 nM, close to IC50 for ICa block (2.3 nM).Fórmula:C24H33N3O8SForma y color:SolidPeso molecular:523.6Azelnidipine, (R)-
CAS:Azelnidipine is an L-type CCB that improves HF severity and cardiac nerve activity in HT and HFpEF compared to cilnidipine.Fórmula:C33H34N4O6Forma y color:SolidPeso molecular:582.65SR-33805
CAS:SR-33805: calcium channel blocker for atherosclerosis/heart failure, enhances myocyte function, modulates myofilament phosphorylation.Fórmula:C32H40N2O5SForma y color:SolidPeso molecular:564.74Teludipine hydrochloride
CAS:Teludipine hydrochloride is a blocker of lipophilic calcium channel.Fórmula:C28H39ClN2O6Pureza:98%Forma y color:SolidPeso molecular:535.07AZD-2066 hydrochloride
CAS:AZD-2066 hydrochloride is an mGlu5 antagonist.Fórmula:C19H17Cl2N5O2Forma y color:SolidPeso molecular:418.28Palonidipine HCl
CAS:Palonidipine HCl is a calcium channel antagonist potentially for the treatment of angina pectoris and hypertension.Fórmula:C29H35ClFN3O6Forma y color:SolidPeso molecular:576.06Levosemotiadil
CAS:Levosemotiadil(SA 3212) is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to preventFórmula:C29H32N2O6SPureza:98.53% - 98.88%Forma y color:SolidPeso molecular:536.64CaV1.3 antagonist-1
CAS:CaV1.3 antagonist-1 is a selective CaV1.3L-type calcium channel antagonist useful for researching neurological disorders and cardiovascular diseases.Fórmula:C17H19ClN2O3Forma y color:SolidPeso molecular:334.8Palonidipine
CAS:Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.Fórmula:C29H34FN3O6Pureza:98%Forma y color:SolidPeso molecular:539.6SQ-31765
CAS:SQ-31765 is a blocker of benzazepine calcium channel.Fórmula:C24H27F3N2O4Pureza:98%Forma y color:SolidPeso molecular:464.48McN5691
CAS:McN5691 is a voltage sensitive calcium channel blocker.Fórmula:C30H35NO3Pureza:98.93% - 99.38%Forma y color:SolidPeso molecular:457.6NPS-2143
CAS:NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.Fórmula:C24H25ClN2O2Pureza:99.56%Forma y color:SolidPeso molecular:408.92(R)-Lercanidipine hydrochloride
CAS:(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.Fórmula:C36H42ClN3O6Pureza:98%Forma y color:SolidPeso molecular:648.2PD0176078
CAS:PD0176078 () is a newly blocker of N-type Calcium channel.Fórmula:C23H30F2N2OPureza:99.72%Forma y color:SolidPeso molecular:388.49Ref: TM-T12385
1mg59,00€5mg105,00€10mg172,00€25mg269,00€50mg374,00€100mg515,00€200mg695,00€1mL*10mM (DMSO)131,00€ORM-10962
CAS:ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55Fórmula:C27H29N3O4Pureza:98%Forma y color:SolidPeso molecular:459.54trans-Ned 19
CAS:trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.Fórmula:C30H31FN4O3Pureza:98%Forma y color:SolidPeso molecular:514.59YM 244769 hydrochloride
CAS:inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)Fórmula:C26H23ClFN3O3Pureza:98%Forma y color:SolidPeso molecular:479.93TTA-Q6
CAS:TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.Fórmula:C20H15ClF3N3OPureza:99.97%Forma y color:SolidPeso molecular:405.8TTA-A8
CAS:TTA-A8 is an antagonist of T-type calcium channel.Fórmula:C22H21F3N4O2Pureza:99.22%Forma y color:SolidPeso molecular:430.42JTV-519 fumarate
CAS:Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.Fórmula:C29H36N2O6SForma y color:SolidPeso molecular:540.67
