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Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 336 productos de "Receptor GABA"

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  • MK-0343

    CAS:
    <p>MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.</p>
    Fórmula:C19H17F2N7O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:397.38
  • DS2

    CAS:
    <p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>
    Fórmula:C18H12ClN3OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:353.83
  • CGS8216

    CAS:
    <p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>
    Fórmula:C16H11N3O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:261.28
  • BHF-177

    CAS:
    <p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>
    Fórmula:C19H20F3N3
    Forma y color:Solid
    Peso molecular:347.38
  • SKF 97541

    CAS:
    <p>GABAB agonist</p>
    Fórmula:C4H12NO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:137.12
  • CGP 7930

    CAS:
    <p>Positive allosteric modulator of GABAB receptors</p>
    Fórmula:C19H32O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:292.46
  • TPA-023B

    CAS:
    <p>TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.</p>
    Fórmula:C21H15F2N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:391.37
  • U-101017

    CAS:
    <p>U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.</p>
    Fórmula:C23H27ClN4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:442.94
  • Org 20599

    CAS:
    <p>GABAA receptor agonist</p>
    Fórmula:C25H40ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.04
  • SX-3228

    CAS:
    <p>SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).</p>
    Fórmula:C18H18N4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.36
  • CGS 20625

    CAS:
    <p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>
    Fórmula:C18H19N3O2
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:309.36
  • 2-Hydroxysaclofen

    CAS:
    <p>2-Hydroxysaclofen is a GABAB receptor antagonist.</p>
    Fórmula:C9H12ClNO4S
    Pureza:98%
    Forma y color:White Solid
    Peso molecular:265.71
  • Ro15-4513

    CAS:
    <p>Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.</p>
    Fórmula:C15H14N6O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:326.31
  • 3-Methyl-GABA

    CAS:
    <p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>
    Fórmula:C20H30N2O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:522.59
  • DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Fórmula:C18H10Br2ClN3OS
    Forma y color:Solid
    Peso molecular:511.62
  • Cyprodenate

    CAS:
    <p>Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.</p>
    Fórmula:C13H25NO2
    Forma y color:Solid
    Peso molecular:227.34
  • Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Fórmula:C18H13ClN2O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.83
  • U-7524

    CAS:
    <p>U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.</p>
    Fórmula:C2H5NO3
    Forma y color:Solid
    Peso molecular:91.07
  • Ethyl dirazepate

    CAS:
    <p>Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.</p>
    Fórmula:C18H14Cl2N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:377.22
  • Arbaclofen placarbil

    CAS:
    <p>Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.</p>
    Fórmula:C19H26ClNO6
    Forma y color:Solid
    Peso molecular:399.87