
Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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MK-0343
CAS:<p>MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.</p>Fórmula:C19H17F2N7OPureza:98%Forma y color:SolidPeso molecular:397.38DS2
CAS:<p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>Fórmula:C18H12ClN3OSPureza:98%Forma y color:SolidPeso molecular:353.83CGS8216
CAS:<p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>Fórmula:C16H11N3OPureza:98.53%Forma y color:SolidPeso molecular:261.28BHF-177
CAS:<p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>Fórmula:C19H20F3N3Forma y color:SolidPeso molecular:347.38SKF 97541
CAS:<p>GABAB agonist</p>Fórmula:C4H12NO2PPureza:98%Forma y color:SolidPeso molecular:137.12CGP 7930
CAS:<p>Positive allosteric modulator of GABAB receptors</p>Fórmula:C19H32O2Pureza:98%Forma y color:SolidPeso molecular:292.46TPA-023B
CAS:<p>TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.</p>Fórmula:C21H15F2N5OPureza:98%Forma y color:SolidPeso molecular:391.37U-101017
CAS:<p>U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.</p>Fórmula:C23H27ClN4O3Pureza:98%Forma y color:SolidPeso molecular:442.94Org 20599
CAS:<p>GABAA receptor agonist</p>Fórmula:C25H40ClNO3Pureza:98%Forma y color:SolidPeso molecular:438.04SX-3228
CAS:<p>SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).</p>Fórmula:C18H18N4O3Pureza:98%Forma y color:SolidPeso molecular:338.36CGS 20625
CAS:<p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>Fórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.362-Hydroxysaclofen
CAS:<p>2-Hydroxysaclofen is a GABAB receptor antagonist.</p>Fórmula:C9H12ClNO4SPureza:98%Forma y color:White SolidPeso molecular:265.71Ro15-4513
CAS:<p>Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.</p>Fórmula:C15H14N6O3Pureza:98%Forma y color:SolidPeso molecular:326.313-Methyl-GABA
CAS:<p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>Fórmula:C20H30N2O10S2Pureza:98%Forma y color:SolidPeso molecular:522.59DS1
CAS:<p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>Fórmula:C18H10Br2ClN3OSForma y color:SolidPeso molecular:511.62Cyprodenate
CAS:<p>Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.</p>Fórmula:C13H25NO2Forma y color:SolidPeso molecular:227.34Y 23684
CAS:<p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>Fórmula:C18H13ClN2O2SPureza:98%Forma y color:SolidPeso molecular:356.83U-7524
CAS:<p>U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.</p>Fórmula:C2H5NO3Forma y color:SolidPeso molecular:91.07Ethyl dirazepate
CAS:<p>Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.</p>Fórmula:C18H14Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:377.22Arbaclofen placarbil
CAS:<p>Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.</p>Fórmula:C19H26ClNO6Forma y color:SolidPeso molecular:399.87
