
Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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CP-409092 hydrochloride
CAS:<p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>Fórmula:C17H20ClN3O2Forma y color:SolidPeso molecular:333.81CGP 46381
CAS:<p>CGP 46381 is a GABAB receptor antagonist.</p>Fórmula:C10H22NO2PPureza:98%Forma y color:White SolidPeso molecular:219.26GABAA receptor agent 5
CAS:<p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>Fórmula:C21H25N3O2SForma y color:SolidPeso molecular:383.51BGT1-IN-9
CAS:<p>BGT1-IN-9 is an M1 muscarinic agonist.</p>Fórmula:C5H10ClN3O2Forma y color:SolidPeso molecular:179.605CCD-3693
CAS:<p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C21H31F3O2Pureza:98%Forma y color:SolidPeso molecular:372.46GABA-AT-IN-1
CAS:<p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4GABAA receptor agent 8
CAS:<p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36ZAPA sulfate
CAS:<p>GABAA receptors agonist</p>Fórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25TPMPA
CAS:<p>GABAA-ρ antagonist</p>Fórmula:C6H12NO2PPureza:98%Forma y color:SolidPeso molecular:161.14TG41
CAS:<p>TG41 is a GABAA receptors positive modulator.</p>Fórmula:C18H13BrCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:440.12FG8119
CAS:<p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>Fórmula:C17H15N5O2Pureza:>99.99%Forma y color:SolidPeso molecular:321.33GABAA receptor agent 6
CAS:<p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41TB 21007
CAS:<p>GABAA receptor inverse agonist</p>Fórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5SL-651498
CAS:<p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42Bamaluzole
CAS:<p>Bamaluzole is an agonist of GABA receptor.</p>Fórmula:C14H12ClN3OPureza:98%Forma y color:SolidPeso molecular:273.72NAP-1
CAS:<p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>Fórmula:C20H18ClNO2Forma y color:SolidPeso molecular:339.82GABAA receptor agent 7
CAS:<p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>Fórmula:C18H13ClN4OForma y color:SolidPeso molecular:336.77MRK-623
CAS:<p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>Fórmula:C20H17FN4OForma y color:SolidPeso molecular:348.37Etbicyphat
CAS:<p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>Fórmula:C6H11O4PForma y color:SolidPeso molecular:178.12TCS 1105
CAS:<p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>Fórmula:C17H13FN2O2Pureza:99.75%Forma y color:SolidPeso molecular:296.3
