Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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Pipazethate
CAS:<p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51NNC052090
CAS:<p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54RU 33965
CAS:<p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>Fórmula:C16H15N3O2Pureza:98%Forma y color:SolidPeso molecular:281.31ZK93423
CAS:<p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43GABAA receptor modulator-2
CAS:<p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>Fórmula:C22H22FN3O5SForma y color:SolidPeso molecular:459.49Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78UMB68 sodium
CAS:<p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.</p>Fórmula:C6H12NaO3Forma y color:SolidPeso molecular:155.149(+)-Nipecotic acid
CAS:<p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>Fórmula:C6H11NO2Pureza:99.38%Forma y color:SolidPeso molecular:129.16(S)-SNAP5114
CAS:<p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>Fórmula:C30H35NO6Pureza:97%Forma y color:SolidPeso molecular:505.6Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Fórmula:C18H14N4O3Pureza:98%Forma y color:SolidPeso molecular:334.333α,21-Dihydroxy-5α-pregnan-20-one
CAS:<p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>Fórmula:C21H34O3Pureza:98.00%Forma y color:SolidPeso molecular:334.49Chlormethiazole edisylate
CAS:<p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>Fórmula:C8H14ClNO6S3Pureza:98%Forma y color:SolidPeso molecular:351.85COR628
CAS:<p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>Fórmula:C16H23NO3SForma y color:SolidPeso molecular:309.42trans-4-Hydroxycrotonic acid
CAS:<p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>Fórmula:C4H6O3Pureza:98%Forma y color:SolidPeso molecular:102.09LY 81067
CAS:<p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>Fórmula:C22H24N4OForma y color:SolidPeso molecular:360.45U 90042
CAS:<p>GABAA receptor ligand</p>Fórmula:C17H13ClN6OPureza:98%Forma y color:SolidPeso molecular:352.78COR627
CAS:<p>COR627 is the GABA receptor positive allosteric modulator.</p>Fórmula:C20H27NO3SPureza:98%Forma y color:SolidPeso molecular:361.5CPP-115
CAS:<p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>Fórmula:C7H9F2NO2Forma y color:SolidPeso molecular:177.15JY-XHe-053
CAS:<p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>Fórmula:C22H16FN3O2Pureza:98%Forma y color:SolidPeso molecular:373.38HIE-124
CAS:<p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>Fórmula:C10H12N2O3SPureza:98%Forma y color:SolidPeso molecular:240.28
