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Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 336 productos de "Receptor GABA"

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  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Fórmula:C16H13ClN2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:364.8
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Fórmula:C10H12ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:213.66
  • ABP-700

    CAS:
    <p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>
    Fórmula:C17H18N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:314.34
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Fórmula:C24H24ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:409.91
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Fórmula:C9H9NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:211.17
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Fórmula:C18H23ClN6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:358.87
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Fórmula:C15H23N5O2S
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:337.44
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Fórmula:C8H15NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:173.21
  • Anxiolytic/nonsedative agent-1

    CAS:
    <p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>
    Fórmula:C18H15N3O4
    Pureza:98.61%
    Forma y color:Solid
    Peso molecular:337.33
  • SCH 50911 hydrochloride

    CAS:
    <p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>
    Fórmula:C8H16ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:209.67
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Fórmula:C17H20N2O3
    Pureza:99.62%
    Forma y color:Solid Crystalline
    Peso molecular:300.35
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Fórmula:C9H8F4N2O2S
    Pureza:98.22% - 98.54%
    Forma y color:Solid
    Peso molecular:284.23
  • U-89843A

    CAS:
    <p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>
    Fórmula:C16H24ClN5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:321.85
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:250.12
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Fórmula:C3H9FNO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:141.08
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Fórmula:C16H25ClN4O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:340.85
  • RO 4938581

    CAS:
    <p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>
    Fórmula:C13H8BrF2N5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.14
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Fórmula:C19H29NO5
    Pureza:98.19% - 99.55%
    Forma y color:Solid
    Peso molecular:351.44
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Fórmula:C9H13ClNO3P
    Pureza:99.32%
    Forma y color:White Solid
    Peso molecular:249.63
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Fórmula:C18H17N5O2
    Pureza:98.30% - 98.94%
    Forma y color:Solid
    Peso molecular:335.36