CymitQuimica logo
Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 336 productos de "Receptor GABA"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • Flufiprole

    CAS:
    <p>Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.</p>
    Fórmula:C16H10Cl2F6N4OS
    Forma y color:Solid
    Peso molecular:491.24
  • AHN-683

    CAS:
    <p>AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.</p>
    Fórmula:C42H32FN3O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:709.72
  • LU-32-176B

    CAS:
    <p>LU32-176B is a bioactive chemical.</p>
    Fórmula:C23H24F2N2O2
    Forma y color:Solid
    Peso molecular:398.45
  • Imagabalin

    CAS:
    <p>Imagabalin is an active compound used in the study of neurological diseases.</p>
    Fórmula:C9H19NO2
    Forma y color:Solid
    Peso molecular:173.25
  • Inaperisone

    CAS:
    <p>Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.</p>
    Fórmula:C16H23NO
    Pureza:99.48%
    Forma y color:Solid
    Peso molecular:245.36
  • Fipronil sulfone

    CAS:
    <p>Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.</p>
    Fórmula:C12H4Cl2F6N4O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:453.14
  • Nitrazolam

    CAS:
    <p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>
    Fórmula:C17H13N5O2
    Forma y color:Solid
    Peso molecular:319.32
  • Azocarnil


    <p>Azocarnil is a GABAergic agonist-enhancer used in neurological system research.</p>
    Forma y color:Odour Solid
  • Furosemide sodium

    CAS:
    <p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>
    Fórmula:C12H10ClN2NaO5S
    Pureza:99.52% - >99.99%
    Forma y color:Solid
    Peso molecular:352.73
  • 12,14-Dichlorodehydroabietic acid

    CAS:
    <p>12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.</p>
    Fórmula:C20H26Cl2O2
    Forma y color:Solid
    Peso molecular:369.33
  • DAA-1106

    CAS:
    <p>DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.</p>
    Fórmula:C23H22FNO4
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:395.42
  • RuBi-GABA

    CAS:
    <p>Ruthenium-bipyridine-triphenylphosphine caged GABA</p>
    Fórmula:C42H39F6N5O2P2Ru
    Pureza:98%
    Forma y color:Solid
    Peso molecular:922.8
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Forma y color:Odour Solid
  • Anticonvulsant agent 8


    <p>Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.</p>
    Fórmula:C15H11N5O
    Forma y color:Solid
    Peso molecular:277.28
  • CGP 35348

    CAS:
    <p>CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。</p>
    Fórmula:C8H20NO4P
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:225.22
  • (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Fórmula:C6H11NO2
    Forma y color:Solid
    Peso molecular:129.16
  • Atagabalin

    CAS:
    <p>Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.</p>
    Fórmula:C10H19NO2
    Forma y color:Solid
    Peso molecular:185.26
  • Ion Channel Targeted Library


    <p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>
    Forma y color:Odour Solid
  • Nipecotic acid

    CAS:
    <p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Fórmula:C6H11NO2
    Forma y color:Off-White To Pale Yellow-Beige Powder
    Peso molecular:129.16
  • GABAA receptor modulator-3


    <p>GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.</p>
    Fórmula:C18H22O2
    Forma y color:Solid
    Peso molecular:270.37