
Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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Flufiprole
CAS:<p>Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.</p>Fórmula:C16H10Cl2F6N4OSForma y color:SolidPeso molecular:491.24AHN-683
CAS:<p>AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.</p>Fórmula:C42H32FN3O7Pureza:98%Forma y color:SolidPeso molecular:709.72LU-32-176B
CAS:<p>LU32-176B is a bioactive chemical.</p>Fórmula:C23H24F2N2O2Forma y color:SolidPeso molecular:398.45Imagabalin
CAS:<p>Imagabalin is an active compound used in the study of neurological diseases.</p>Fórmula:C9H19NO2Forma y color:SolidPeso molecular:173.25Inaperisone
CAS:<p>Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.</p>Fórmula:C16H23NOPureza:99.48%Forma y color:SolidPeso molecular:245.36Fipronil sulfone
CAS:<p>Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.</p>Fórmula:C12H4Cl2F6N4O2SPureza:98%Forma y color:SolidPeso molecular:453.14Nitrazolam
CAS:<p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>Fórmula:C17H13N5O2Forma y color:SolidPeso molecular:319.32Azocarnil
<p>Azocarnil is a GABAergic agonist-enhancer used in neurological system research.</p>Forma y color:Odour SolidFurosemide sodium
CAS:<p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>Fórmula:C12H10ClN2NaO5SPureza:99.52% - >99.99%Forma y color:SolidPeso molecular:352.7312,14-Dichlorodehydroabietic acid
CAS:<p>12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.</p>Fórmula:C20H26Cl2O2Forma y color:SolidPeso molecular:369.33DAA-1106
CAS:<p>DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.</p>Fórmula:C23H22FNO4Pureza:99.54%Forma y color:SolidPeso molecular:395.42RuBi-GABA
CAS:<p>Ruthenium-bipyridine-triphenylphosphine caged GABA</p>Fórmula:C42H39F6N5O2P2RuPureza:98%Forma y color:SolidPeso molecular:922.8Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>Forma y color:Odour SolidAnticonvulsant agent 8
<p>Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.</p>Fórmula:C15H11N5OForma y color:SolidPeso molecular:277.28CGP 35348
CAS:<p>CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。</p>Fórmula:C8H20NO4PPureza:≥98%Forma y color:SolidPeso molecular:225.22(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Fórmula:C6H11NO2Forma y color:SolidPeso molecular:129.16Atagabalin
CAS:<p>Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.</p>Fórmula:C10H19NO2Forma y color:SolidPeso molecular:185.26Ion Channel Targeted Library
<p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>Forma y color:Odour SolidNipecotic acid
CAS:<p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C6H11NO2Forma y color:Off-White To Pale Yellow-Beige PowderPeso molecular:129.16GABAA receptor modulator-3
<p>GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.</p>Fórmula:C18H22O2Forma y color:SolidPeso molecular:270.37

