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Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 336 productos de "Receptor GABA"

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  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Forma y color:Light Beige Crystalline Powder
    Peso molecular:109.3
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Fórmula:C11H11N3O
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:201.22
  • Fipronil

    CAS:
    <p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>
    Fórmula:C12H4Cl2F6N4OS
    Pureza:97.21%
    Forma y color:Solid Powder
    Peso molecular:437.15
  • Darigabat

    CAS:
    <p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>
    Fórmula:C22H21FN4O3S
    Pureza:98.42% - 99.29%
    Forma y color:Solid
    Peso molecular:440.49
  • Riluzole

    CAS:
    <p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>
    Fórmula:C8H5F3N2OS
    Pureza:99.71% - 99.88%
    Forma y color:Powder
    Peso molecular:234.2
  • CGP 36216 hydrochloride

    CAS:
    <p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>
    Fórmula:C5H14NO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:151.14
  • β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Fórmula:C16H16N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:268.31
  • NO 711

    CAS:
    <p>NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>
    Fórmula:C21H22N2O3
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:350.41
  • (±)-Homoproline Hydrochloride

    CAS:
    <p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C6H12ClNO2
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:165.62
  • CP-457920

    CAS:
    <p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>
    Fórmula:C18H17N3O3
    Pureza:99.06% - 99.74%
    Forma y color:Solid
    Peso molecular:323.35
  • Ro 41-3290

    CAS:
    <p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>
    Fórmula:C24H21ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.89
  • PF-0713

    CAS:
    <p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>
    Fórmula:C14H22O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:206.32
  • HZ166

    CAS:
    <p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>
    Fórmula:C21H16N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.38
  • Pregabalin arenacarbil

    CAS:
    <p>Pregabalin arenacarbil is a gabamimetic.</p>
    Fórmula:C15H27NO6
    Forma y color:Solid
    Peso molecular:317.38
  • NCS-382

    CAS:
    <p>γ-Hydroxybutyric acid antagonist</p>
    Fórmula:C13H14O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:218.25
  • Ro 19-4603

    CAS:
    <p>Benzodiazepine inverse agonist</p>
    Fórmula:C15H17N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:319.38
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Fórmula:C17H24N2O
    Forma y color:Solid
    Peso molecular:272.39
  • mGAT3/4-IN-1

    CAS:
    <p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>
    Fórmula:C26H31ClN2O2S2
    Forma y color:Solid
    Peso molecular:503.12
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Fórmula:C21H21Cl2N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.33
  • 17-PA

    CAS:
    <p>17-PA is a GABAA receptor antagonist.</p>
    Fórmula:C25H34O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:350.54