Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 365 productos de "Receptor GABA"
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Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Fórmula:C18H12Cl2N2OForma y color:SolidPeso molecular:343.21Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Fórmula:C15H14N6O3Pureza:98%Forma y color:SolidPeso molecular:326.31ZK-91296
CAS:ZK-91296: GABA agonist, lowers anxiety without sedation, may target specific BZ receptor subtype.Fórmula:C23H22N2O4Pureza:98%Forma y color:SolidPeso molecular:390.432-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98%Forma y color:White SolidPeso molecular:265.71SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Fórmula:C8H15NO3Forma y color:SolidPeso molecular:173.21CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.36Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Fórmula:C14H22ClNOPureza:98%Forma y color:SolidPeso molecular:255.78SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Fórmula:C18H18N4O3Pureza:98%Forma y color:SolidPeso molecular:338.36Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Fórmula:C15H15N3O3Forma y color:SolidPeso molecular:285.3Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Fórmula:C20H22ClN5O3SPureza:98%Forma y color:SolidPeso molecular:447.94Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Fórmula:C15H14ClN3O3Forma y color:SolidPeso molecular:319.74CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Fórmula:C18H17N3O3Pureza:99.06% - 99.74%Forma y color:SolidPeso molecular:323.35Org 20599
CAS:GABAA receptor agonistFórmula:C25H40ClNO3Pureza:98%Forma y color:SolidPeso molecular:438.04U-101017
CAS:U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.Fórmula:C23H27ClN4O3Pureza:98%Forma y color:SolidPeso molecular:442.94TPA-023B
CAS:TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.Fórmula:C21H15F2N5OPureza:98%Forma y color:SolidPeso molecular:391.37CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFórmula:C19H32O2Pureza:98%Forma y color:SolidPeso molecular:292.46BHF-177
CAS:BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.Fórmula:C19H20F3N3Forma y color:SolidPeso molecular:347.38CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Fórmula:C16H11N3OPureza:98.53%Forma y color:SolidPeso molecular:261.28SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Fórmula:C8H16ClNO3Pureza:98%Forma y color:SolidPeso molecular:209.67DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFórmula:C18H12ClN3OSPureza:98%Forma y color:SolidPeso molecular:353.83(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFórmula:C6H12ClNO2Pureza:99.69%Forma y color:SolidPeso molecular:165.62MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Fórmula:C19H17F2N7OPureza:98%Forma y color:SolidPeso molecular:397.3817-PA
CAS:17-PA is a GABAA receptor antagonist.Fórmula:C25H34OPureza:98%Forma y color:SolidPeso molecular:350.54Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Fórmula:C17H20N2O3Pureza:99.62%Forma y color:Solid CrystallinePeso molecular:300.35CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Fórmula:C21H21Cl2N5O2Pureza:98%Forma y color:SolidPeso molecular:446.33E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Fórmula:C9H8F4N2O2SPureza:98.22% - 98.54%Forma y color:SolidPeso molecular:284.23U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Fórmula:C16H24ClN5Pureza:98%Forma y color:SolidPeso molecular:321.85(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:98%Forma y color:SolidPeso molecular:250.12NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Fórmula:C21H22N2O3Pureza:99.70%Forma y color:SolidPeso molecular:350.41AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Fórmula:C19H29NO5Pureza:98.19% - 99.55%Forma y color:SolidPeso molecular:351.44mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Fórmula:C26H31ClN2O2S2Forma y color:SolidPeso molecular:503.12GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Fórmula:C17H24N2OForma y color:SolidPeso molecular:272.39Ro 19-4603
CAS:Benzodiazepine inverse agonistFórmula:C15H17N3O3SPureza:98%Forma y color:SolidPeso molecular:319.38TG41
CAS:TG41 is a GABAA receptors positive modulator.Fórmula:C18H13BrCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:440.12FG8119
CAS:FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.Fórmula:C17H15N5O2Pureza:>99.99%Forma y color:SolidPeso molecular:321.33GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41TB 21007
CAS:GABAA receptor inverse agonistFórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Fórmula:C14H12ClN3OPureza:98%Forma y color:SolidPeso molecular:273.72ZAPA sulfate
CAS:GABAA receptors agonistFórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25Lesogaberan
CAS:Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).Fórmula:C3H9FNO2PPureza:98%Forma y color:SolidPeso molecular:141.08NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Fórmula:C20H18ClNO2Forma y color:SolidPeso molecular:339.82GABAA receptor agent 7
CAS:Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.Fórmula:C18H13ClN4OForma y color:SolidPeso molecular:336.77MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Fórmula:C20H17FN4OForma y color:SolidPeso molecular:348.37GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Fórmula:C6H11O4PForma y color:SolidPeso molecular:178.12NCS-382
CAS:γ-Hydroxybutyric acid antagonistFórmula:C13H14O3Pureza:98%Forma y color:SolidPeso molecular:218.25TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Fórmula:C17H13FN2O2Pureza:99.75%Forma y color:SolidPeso molecular:296.3Pipazethate
CAS:Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54RU 33965
CAS:RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.Fórmula:C16H15N3O2Pureza:98%Forma y color:SolidPeso molecular:281.31CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Fórmula:C5H14NO2PPureza:98%Forma y color:SolidPeso molecular:151.14β-CCB
CAS:benzodiazepine receptor ligandFórmula:C16H16N2O2Pureza:98%Forma y color:SolidPeso molecular:268.31GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Fórmula:C15H27NO6Forma y color:SolidPeso molecular:317.38GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Fórmula:C22H22FN3O5SForma y color:SolidPeso molecular:459.49Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Fórmula:C6H12NaO3Forma y color:SolidPeso molecular:155.149Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Fórmula:C16H25ClN4O2Pureza:99.52%Forma y color:SolidPeso molecular:340.85(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Fórmula:C6H11NO2Pureza:99.38%Forma y color:SolidPeso molecular:129.16Phaclofen
CAS:GABAB antagonistFórmula:C9H13ClNO3PPureza:99.32%Forma y color:White SolidPeso molecular:249.63(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Fórmula:C30H35NO6Pureza:98.20%Forma y color:SolidPeso molecular:505.6Ref: TM-T16831
5mg52,00€10mg78,00€25mg160,00€50mg225,00€100mg325,00€200mg445,00€1mL*10mM (DMSO)51,00€Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Fórmula:C18H14N4O3Pureza:98%Forma y color:SolidPeso molecular:334.333α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Fórmula:C21H34O3Pureza:98.00%Forma y color:SolidPeso molecular:334.49HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Fórmula:C21H16N4O2Pureza:98%Forma y color:SolidPeso molecular:356.38BGT1-IN-9
CAS:BGT1-IN-9 is an M1 muscarinic agonist.Fórmula:C5H10ClN3O2Forma y color:SolidPeso molecular:179.605RO 4938581
CAS:RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).Fórmula:C13H8BrF2N5Pureza:98%Forma y color:SolidPeso molecular:352.14Chlormethiazole edisylate
CAS:Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.Fórmula:C8H14ClNO6S3Pureza:98%Forma y color:SolidPeso molecular:351.85COR628
CAS:COR628 is the GABA(B) receptor positive allosteric modulator.Fórmula:C16H23NO3SForma y color:SolidPeso molecular:309.42trans-4-Hydroxycrotonic acid
CAS:ligand of γ-hydroxybutyric acid (GHB) receptorFórmula:C4H6O3Pureza:98%Forma y color:SolidPeso molecular:102.09LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Fórmula:C22H24N4OForma y color:SolidPeso molecular:360.45U 90042
CAS:GABAA receptor ligandFórmula:C17H13ClN6OPureza:98%Forma y color:SolidPeso molecular:352.78COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Fórmula:C20H27NO3SPureza:98%Forma y color:SolidPeso molecular:361.5CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Fórmula:C7H9F2NO2Forma y color:SolidPeso molecular:177.15GABAA receptor agent 5
CAS:Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.Fórmula:C21H25N3O2SPureza:99.39%Forma y color:SolidPeso molecular:383.51JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Fórmula:C22H16FN3O2Pureza:98%Forma y color:SolidPeso molecular:373.38HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Fórmula:C10H12N2O3SPureza:98%Forma y color:SolidPeso molecular:240.28Fengabine
CAS:Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Fórmula:C17H17Cl2NOPureza:99.37%Forma y color:SolidPeso molecular:322.23RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Fórmula:C21H19F2N3O3Pureza:99.57% - 99.95%Forma y color:SolidPeso molecular:399.39Ref: TM-T16811
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFórmula:C19H19F2N7OPureza:98.12% - 99.70%Forma y color:SolidPeso molecular:399.4Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Fórmula:C18H19N3O2Pureza:97.07%Forma y color:SolidPeso molecular:309.36Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Fórmula:C21H23Cl2N3OPureza:99.56% - 99.97%Forma y color:White To Off-White SolidPeso molecular:404.33Ref: TM-T26600
1mg62,00€5mg144,00€10mg219,00€25mg393,00€50mg550,00€100mg787,00€500mg1.596,00€1mL*10mM (DMSO)129,00€Panadiplon
CAS:Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment ofFórmula:C18H17N5O2Pureza:98.30% - 98.94%Forma y color:SolidPeso molecular:335.36DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Fórmula:C14H12FNOPureza:99.51% - 99.56%Forma y color:SolidPeso molecular:229.25Ref: TM-T11106
1mg115,00€2mg172,00€5mg255,00€10mg374,00€25mg562,00€50mg787,00€100mg1.074,00€500mg2.147,00€1mL*10mM (DMSO)220,00€DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Fórmula:C17H19ClN2O4Pureza:99.56%Forma y color:SolidPeso molecular:350.8Ref: TM-T11061
1mg37,00€2mg49,00€5mg85,00€10mg111,00€25mg250,00€50mg464,00€100mg655,00€1mL*10mM (DMSO)93,00€NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Fórmula:C21H23ClN2O3Pureza:99.92%Forma y color:SolidPeso molecular:386.87Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Forma y color:SolidPeso molecular:295.34ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Fórmula:C14H16ClN3OPureza:>99.99%Forma y color:SolidPeso molecular:277.75Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Fórmula:C15H14ClN3O3Pureza:99.46%Forma y color:SolidPeso molecular:319.74Suriclone
CAS:Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Forma y color:SolidPeso molecular:477.99BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFórmula:C19H20Cl2N2OPureza:99.43% - 99.95%Forma y color:SolidPeso molecular:363.28Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Fórmula:C18H17N3O2Pureza:99.21%Forma y color:SolidPeso molecular:307.35Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Fórmula:C8H6ClF3N2OSPureza:99.76%Forma y color:SolidPeso molecular:270.66Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Fórmula:C26H25ClN2O3Pureza:98.54%Forma y color:SolidPeso molecular:448.94Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Fórmula:C19H20ClN3OPureza:98.42%Forma y color:SolidPeso molecular:341.83Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Fórmula:C21H31NO2Pureza:99.90% - 99.99%Forma y color:SolidPeso molecular:329.48Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Fórmula:C4H7BrN2O2Pureza:98.13%Forma y color:Off-White PowderPeso molecular:195.01Ref: TM-T20657
1mg119,00€2mg172,00€5mg253,00€10mg406,00€25mg657,00€50mg948,00€100mg1.264,00€500mg2.555,00€1mL*10mM (DMSO)215,00€NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C22H20N4OPureza:99.7% - 99.82%Forma y color:SolidPeso molecular:356.42Progabide
CAS:Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.Fórmula:C17H16ClFN2O2Pureza:99.68%Forma y color:SolidPeso molecular:334.77Cirsimaritin
CAS:<p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>Fórmula:C17H14O6Pureza:99.9%Forma y color:SolidPeso molecular:314.29U 89843A
CAS:U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.Fórmula:C16H23N5Pureza:99.62%Forma y color:SolidPeso molecular:285.39CGP-54626 free base
CAS:CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Fórmula:C18H28Cl2NO3PPureza:98%Forma y color:SolidPeso molecular:408.3CGP 64213
CAS:CGP 64213 is a GABAb receptor agonist.Fórmula:C26H36IN2O7PPureza:98%Forma y color:SolidPeso molecular:646.45Afizagabar
CAS:Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.38mGAT-IN-1
CAS:mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).Fórmula:C28H34ClN3O2S2Forma y color:SolidPeso molecular:544.17Adipiplon
CAS:Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.Fórmula:C18H18FN7Forma y color:SolidPeso molecular:351.38(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Fórmula:C21H20INO6Pureza:99.24%Forma y color:SolidPeso molecular:509.29CGP 54626 hydrochloride
CAS:CGP 54626 hydrochloride is a GABAB receptor antagonist.Fórmula:C18H29Cl3NO3PPureza:98%Forma y color:SolidPeso molecular:444.76GMA-839
CAS:GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.Fórmula:C21H31F3O3Pureza:98%Forma y color:SolidPeso molecular:388.46PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Fórmula:C18H15N3O3Pureza:99.79%Forma y color:SolidPeso molecular:321.33Ref: TM-T28479
1mg52,00€5mg111,00€10mg170,00€25mg305,00€50mg472,00€100mg723,00€500mg1.454,00€1mL*10mM (DMSO)202,00€FGIN-1-27
CAS:FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).Fórmula:C28H37FN2OPureza:99.86%Forma y color:SolidPeso molecular:436.6PHP 501 trifluoroacetate
CAS:GABAA antagonistFórmula:C20H21N3OPureza:98%Forma y color:SolidPeso molecular:319.4ADX71441
CAS:ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.Fórmula:C19H15ClF2N4O4Forma y color:SolidPeso molecular:436.8SCS
CAS:SCS is a GABAA receptor antagonist.Fórmula:C14H12N2O3Pureza:99.73%Forma y color:SolidPeso molecular:256.26L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Fórmula:C17H16ClN5O2Pureza:98%Forma y color:SolidPeso molecular:357.79Piperidine-4-sulfonic acid
CAS:Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].Fórmula:C5H11NO3SPureza:98%Forma y color:SolidPeso molecular:165.21(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84CGP36216 hydrochloride
CAS:CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].Fórmula:C5H15ClNO2PForma y color:SolidPeso molecular:187.6Diproqualone
CAS:Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].Fórmula:C12H14N2O3Forma y color:SolidPeso molecular:234.255CGP 55845 hydrochloride
CAS:CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].Fórmula:C18H23Cl3NO3PForma y color:SolidPeso molecular:438.71GABAA receptor agent 2 TFA
CAS:Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.Fórmula:C22H22F3N3O3Forma y color:SolidPeso molecular:433.42NO-711ME
CAS:NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.Fórmula:C22H24N2O3Pureza:99.54%Forma y color:SolidPeso molecular:364.44Ref: TM-T24540
1mg67,00€5mg136,00€10mg198,00€25mg316,00€50mg452,00€100mg607,00€200mg810,00€1mL*10mM (DMSO)145,00€NCS-382 sodium
CAS:NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological diseaseFórmula:C13H13NaO3Pureza:98%Forma y color:SolidPeso molecular:240.23L-822179
CAS:L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.Fórmula:C17H14N8O2Pureza:98.5% - 99.61%Forma y color:SolidPeso molecular:362.35CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Fórmula:C17H19N3O2Pureza:98%Forma y color:SolidPeso molecular:297.35COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Fórmula:C16H16ClNO3SPureza:99.75%Forma y color:SolidPeso molecular:337.82Ref: TM-T36520
1mg40,00€5mg90,00€10mg130,00€25mg227,00€50mg316,00€100mg434,00€200mg590,00€1mL*10mM (DMSO)89,00€Org-21465
CAS:Org-21465, a gamma-aminobutyric acid (GABA) receptor agonist, is used potentially for the use of anesthesia.Fórmula:C27H43NO4Pureza:98%Forma y color:SolidPeso molecular:445.63(R)-4-Amino-3-hydroxybutyric Acid
CAS:(R)-4-Amino-3-hydroxybutyric acid, also known as (R)-GABOB, acts as a modulator of GABA receptors, specifically binding to both GABAA and GABAB receptors and blocking GABA reuptake in rat brain synaptosomes. Additionally, it serves as a GABAC receptor agonist, triggering currents in patch-clamp assays with Xenopus oocytes that express the human receptor. In vivo studies reveal its capability to suppress electrical discharges in the amygdala in cats undergoing N-amidinobenzamide-triggered seizures, indicating its potential therapeutic application in managing seizure disorders.Fórmula:C4H9NO3Forma y color:SolidPeso molecular:119.12mGAT3/4-IN-2
CAS:mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.Fórmula:C26H32ClN3OS2Forma y color:SolidPeso molecular:502.13JM-1232
CAS:JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.Fórmula:C24H27N3O2Forma y color:SolidPeso molecular:389.49RPC425 free base
CAS:RPC425 is a noncompetitive inhibitors of the Betaine-γ-Aminobutyric Acid Transporter 1 (BGT1).Fórmula:C22H27NO2S2Pureza:98%Forma y color:SolidPeso molecular:401.59GABA-IN-2
CAS:GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1Fórmula:C12H4Cl2F6N4SeForma y color:SolidPeso molecular:468.04TPA 023
CAS:<p>TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).</p>Fórmula:C20H22FN7OPureza:99.75%Forma y color:SolidPeso molecular:395.43CGP 55845
CAS:CGP 55845: potent, selective GABAB blocker, IC50=5 nM, hinders agonist binding, reduces GABA/glutamate release.Fórmula:C18H22Cl2NO3PForma y color:SolidPeso molecular:402.256,2'-Dihydroxyflavone
CAS:6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.Fórmula:C15H10O4Pureza:99.44% - 99.67%Forma y color:SolidPeso molecular:254.24GABA-IN-4
CAS:GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.Fórmula:C17H13ClN2O2Forma y color:SolidPeso molecular:312.75S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Fórmula:C12H13N4O6PPureza:98%Forma y color:SolidPeso molecular:340.23EF1502 free base
CAS:EF1502 is a potent and selective GABA transporter inhibitor.Fórmula:C22H26N2O2S2Pureza:98%Forma y color:SolidPeso molecular:414.58Tuclazepam
CAS:Tuclazepam (KC 1956) is a derivative of the benzodiazepine class of drugs, exhibiting anti-anxiety and sedative properties.Fórmula:C17H16Cl2N2OForma y color:SolidPeso molecular:335.23Refisolone
CAS:Refisolone is an antagonist of the GABAA receptor.Fórmula:C18H24O3Peso molecular:288.381Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Fórmula:C7H10ClNO2Forma y color:SolidPeso molecular:175.61SGE-516
CAS:SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.Fórmula:C23H35N3O2Pureza:98%Forma y color:SolidPeso molecular:385.54CGS-9895
CAS:CGS-9895 is a GABA antagonist that operates by interacting with the benzodiazepine binding site on GABA receptors containing the γ subunit (ag).Fórmula:C17H13N3O2Peso molecular:291.304GABAA receptor agonist 2
Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.Fórmula:C22H36O5Forma y color:SolidPeso molecular:380.52β-CCM
CAS:β-CCM is a benzodiazepine receptor inverse agonist with anxiogenic and convulsant effects. It enhances emotional reactivity and reduces interference sensitivity in spatial working memory tasks. β-CCM is applicable in research related to anxiety disorders.Fórmula:C13H10N2O2Peso molecular:226.231Moxetomidate
CAS:<p>Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.</p>Fórmula:C15H18N2O3Forma y color:SolidPeso molecular:274.315GABAA receptor agonist 1
Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45ZK 93426 hydrochloride
CAS:benzodiazepine receptor antagonist,competitiveFórmula:C18H21ClN2O3Pureza:98%Forma y color:SolidPeso molecular:348.82TP003
CAS:<p>TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.</p>Fórmula:C23H16F3N3OPureza:99.17%Forma y color:SolidPeso molecular:407.39BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.14Cyproflanilide
CAS:Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.Fórmula:C28H17BrF12N2O2Forma y color:SolidPeso molecular:721.33Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Fórmula:C4H6N2OSPureza:98%Forma y color:SolidPeso molecular:130.17Fletazepam
CAS:Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.Fórmula:C17H13ClF4N2Forma y color:SolidPeso molecular:356.74(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Fórmula:C21H20BrNO6Forma y color:WhitePeso molecular:462.29Alfadolone acetate
CAS:Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.Fórmula:C23H34O5Forma y color:SolidPeso molecular:390.512-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Fórmula:C3H10NO3PPureza:98%Forma y color:SolidPeso molecular:139.0913-Methylglutaconic acid
CAS:3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].Fórmula:C6H8O4Pureza:98%Forma y color:SolidPeso molecular:144.13CGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Fórmula:C4H12NO3PPureza:98%Forma y color:SolidPeso molecular:153.12Pipequaline
CAS:Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.Fórmula:C22H24N2Pureza:98%Forma y color:SolidPeso molecular:316.44Ref: TM-T4655
Producto descatalogadoPazinaclone
CAS:Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.Fórmula:C25H23ClN4O4Pureza:97.79% - 98.65%Forma y color:SolidPeso molecular:478.93Xilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Fórmula:C26H37N3O2Pureza:98%Forma y color:SolidPeso molecular:423.59Ref: TM-T78670
Producto descatalogadoCGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Fórmula:C19H30NO5PPureza:98%Forma y color:SolidPeso molecular:383.42
