Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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CP-409092 hydrochloride
CAS:<p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>Fórmula:C17H20ClN3O2Forma y color:SolidPeso molecular:333.81CGP 46381
CAS:<p>CGP 46381 is a GABAB receptor antagonist.</p>Fórmula:C10H22NO2PPureza:98%Forma y color:White SolidPeso molecular:219.26GABAA receptor agent 5
CAS:<p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>Fórmula:C21H25N3O2SForma y color:SolidPeso molecular:383.51BGT1-IN-9
CAS:<p>BGT1-IN-9 is an M1 muscarinic agonist.</p>Fórmula:C5H10ClN3O2Forma y color:SolidPeso molecular:179.605CCD-3693
CAS:<p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C21H31F3O2Pureza:98%Forma y color:SolidPeso molecular:372.46GABA-AT-IN-1
CAS:<p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4GABAA receptor agent 8
CAS:<p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36ZAPA sulfate
CAS:<p>GABAA receptors agonist</p>Fórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25TPMPA
CAS:<p>GABAA-ρ antagonist</p>Fórmula:C6H12NO2PPureza:98%Forma y color:SolidPeso molecular:161.14TG41
CAS:<p>TG41 is a GABAA receptors positive modulator.</p>Fórmula:C18H13BrCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:440.12FG8119
CAS:<p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>Fórmula:C17H15N5O2Pureza:>99.99%Forma y color:SolidPeso molecular:321.33GABAA receptor agent 6
CAS:<p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41TB 21007
CAS:<p>GABAA receptor inverse agonist</p>Fórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5SL-651498
CAS:<p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42Bamaluzole
CAS:<p>Bamaluzole is an agonist of GABA receptor.</p>Fórmula:C14H12ClN3OPureza:98%Forma y color:SolidPeso molecular:273.72NAP-1
CAS:<p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>Fórmula:C20H18ClNO2Forma y color:SolidPeso molecular:339.82GABAA receptor agent 7
CAS:<p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>Fórmula:C18H13ClN4OForma y color:SolidPeso molecular:336.77MRK-623
CAS:<p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>Fórmula:C20H17FN4OForma y color:SolidPeso molecular:348.37Etbicyphat
CAS:<p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>Fórmula:C6H11O4PForma y color:SolidPeso molecular:178.12TCS 1105
CAS:<p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>Fórmula:C17H13FN2O2Pureza:99.75%Forma y color:SolidPeso molecular:296.3Pipazethate
CAS:<p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51NNC052090
CAS:<p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54RU 33965
CAS:<p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>Fórmula:C16H15N3O2Pureza:98%Forma y color:SolidPeso molecular:281.31ZK93423
CAS:<p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43GABAA receptor modulator-2
CAS:<p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>Fórmula:C22H22FN3O5SForma y color:SolidPeso molecular:459.49Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78UMB68 sodium
CAS:<p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.</p>Fórmula:C6H12NaO3Forma y color:SolidPeso molecular:155.149(+)-Nipecotic acid
CAS:<p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>Fórmula:C6H11NO2Pureza:99.38%Forma y color:SolidPeso molecular:129.16(S)-SNAP5114
CAS:<p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>Fórmula:C30H35NO6Pureza:97%Forma y color:SolidPeso molecular:505.6Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Fórmula:C18H14N4O3Pureza:98%Forma y color:SolidPeso molecular:334.333α,21-Dihydroxy-5α-pregnan-20-one
CAS:<p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>Fórmula:C21H34O3Pureza:98.00%Forma y color:SolidPeso molecular:334.49Chlormethiazole edisylate
CAS:<p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>Fórmula:C8H14ClNO6S3Pureza:98%Forma y color:SolidPeso molecular:351.85COR628
CAS:<p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>Fórmula:C16H23NO3SForma y color:SolidPeso molecular:309.42trans-4-Hydroxycrotonic acid
CAS:<p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>Fórmula:C4H6O3Pureza:98%Forma y color:SolidPeso molecular:102.09LY 81067
CAS:<p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>Fórmula:C22H24N4OForma y color:SolidPeso molecular:360.45U 90042
CAS:<p>GABAA receptor ligand</p>Fórmula:C17H13ClN6OPureza:98%Forma y color:SolidPeso molecular:352.78COR627
CAS:<p>COR627 is the GABA receptor positive allosteric modulator.</p>Fórmula:C20H27NO3SPureza:98%Forma y color:SolidPeso molecular:361.5CPP-115
CAS:<p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>Fórmula:C7H9F2NO2Forma y color:SolidPeso molecular:177.15JY-XHe-053
CAS:<p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>Fórmula:C22H16FN3O2Pureza:98%Forma y color:SolidPeso molecular:373.38HIE-124
CAS:<p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>Fórmula:C10H12N2O3SPureza:98%Forma y color:SolidPeso molecular:240.28Suclofenide
CAS:<p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>Fórmula:C16H13ClN2O4SPureza:98%Forma y color:SolidPeso molecular:364.8(S)-Baclofen
CAS:<p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>Fórmula:C10H12ClNO2Pureza:98%Forma y color:SolidPeso molecular:213.66ABP-700
CAS:<p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>Fórmula:C17H18N2O4Pureza:98%Forma y color:SolidPeso molecular:314.34DAA-1097
CAS:<p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>Fórmula:C24H24ClNO3Pureza:98%Forma y color:SolidPeso molecular:409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:<p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>Fórmula:C9H9NO5Pureza:98%Forma y color:SolidPeso molecular:211.17PNU-107484A
CAS:<p>PNU-107484A is a unique GABA(A) receptor ligand.</p>Fórmula:C18H23ClN6Pureza:98%Forma y color:SolidPeso molecular:358.87GS 39783
CAS:<p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>Fórmula:C15H23N5O2SPureza:99.92%Forma y color:SolidPeso molecular:337.44SCH 50911
CAS:<p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>Fórmula:C8H15NO3Pureza:98%Forma y color:SolidPeso molecular:173.21Anxiolytic/nonsedative agent-1
CAS:<p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>Fórmula:C18H15N3O4Pureza:98.61%Forma y color:SolidPeso molecular:337.33SCH 50911 hydrochloride
CAS:<p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>Fórmula:C8H16ClNO3Pureza:98%Forma y color:SolidPeso molecular:209.67Bifenazate
CAS:<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Fórmula:C17H20N2O3Pureza:99.62%Forma y color:Solid CrystallinePeso molecular:300.35E2730
CAS:<p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>Fórmula:C9H8F4N2O2SPureza:98.22% - 98.54%Forma y color:SolidPeso molecular:284.23U-89843A
CAS:<p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>Fórmula:C16H24ClN5Pureza:98%Forma y color:SolidPeso molecular:321.85(R)-Baclofen hydrochloride
CAS:<p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>Fórmula:C10H13Cl2NO2Pureza:98%Forma y color:SolidPeso molecular:250.12Lesogaberan
CAS:<p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>Fórmula:C3H9FNO2PPureza:98%Forma y color:SolidPeso molecular:141.08Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Fórmula:C16H25ClN4O2Pureza:99.52%Forma y color:SolidPeso molecular:340.85RO 4938581
CAS:<p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>Fórmula:C13H8BrF2N5Pureza:98%Forma y color:SolidPeso molecular:352.14AZD 3043
CAS:<p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>Fórmula:C19H29NO5Pureza:98.19% - 99.55%Forma y color:SolidPeso molecular:351.44Phaclofen
CAS:<p>GABAB antagonist</p>Fórmula:C9H13ClNO3PPureza:99.32%Forma y color:White SolidPeso molecular:249.63Panadiplon
CAS:<p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>Fórmula:C18H17N5O2Pureza:98.30% - 98.94%Forma y color:SolidPeso molecular:335.36Cirsimaritin
CAS:<p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>Fórmula:C17H14O6Pureza:99.9%Forma y color:SolidPeso molecular:314.29Progabide
CAS:<p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>Fórmula:C17H16ClFN2O2Pureza:99.68%Forma y color:SolidPeso molecular:334.77Saripidem
CAS:<p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>Fórmula:C19H20ClN3OPureza:99.45%Forma y color:SolidPeso molecular:341.83NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C22H20N4OPureza:99.7% - 99.82%Forma y color:SolidPeso molecular:356.42ELB-139
CAS:<p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>Fórmula:C14H16ClN3OPureza:>99.99%Forma y color:SolidPeso molecular:277.75Ru-32514
CAS:<p>Ru-32514 is a benzodiazepine receptor agonist.</p>Fórmula:C18H17N3O2Pureza:99.21%Forma y color:SolidPeso molecular:307.35Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Fórmula:C17H17Cl2NOPureza:99%Forma y color:SolidPeso molecular:322.23Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Fórmula:C18H19N3O2Pureza:97.07%Forma y color:SolidPeso molecular:309.36DMCM hydrochloride
CAS:<p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>Fórmula:C17H19ClN2O4Pureza:99.56%Forma y color:SolidPeso molecular:350.8Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Forma y color:SolidPeso molecular:477.99NNC 05-711
CAS:<p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>Fórmula:C21H23ClN2O3Pureza:99.92%Forma y color:SolidPeso molecular:386.87Riluzole hydrochloride
CAS:<p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>Fórmula:C8H6ClF3N2OSPureza:99.76%Forma y color:SolidPeso molecular:270.66BPDBA
CAS:<p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>Fórmula:C19H20Cl2N2OPureza:99.37% - 99.95%Forma y color:SolidPeso molecular:363.28RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Fórmula:C21H19F2N3O3Pureza:99.57% - 99.95%Forma y color:SolidPeso molecular:399.39Lirequinil
CAS:<p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>Fórmula:C26H25ClN2O3Pureza:98.54%Forma y color:SolidPeso molecular:448.94L-838417
CAS:<p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>Fórmula:C19H19F2N7OPureza:98.12% - 99.70%Forma y color:SolidPeso molecular:399.4Divaplon
CAS:<p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Forma y color:SolidPeso molecular:295.34Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Fórmula:C21H23Cl2N3OPureza:99.56% - 99.97%Forma y color:White To Off-White SolidPeso molecular:404.33Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Fórmula:C15H14ClN3O3Pureza:99.46%Forma y color:SolidPeso molecular:319.74Golexanolone
CAS:<p>Golexanolone can be used to study neurological diseases.</p>Fórmula:C21H31NO2Pureza:99.90% - 99.99%Forma y color:SolidPeso molecular:329.48Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Fórmula:C4H7BrN2O2Pureza:98.13%Forma y color:Off-White PowderPeso molecular:195.01DSP-0565
CAS:<p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>Fórmula:C14H12FNOPureza:99.51% - 99.56%Forma y color:SolidPeso molecular:229.25CGP 55845 hydrochloride
CAS:<p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>Fórmula:C18H23Cl3NO3PForma y color:SolidPeso molecular:438.71FGIN-1-27
CAS:<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Fórmula:C28H37FN2OPureza:99.86%Forma y color:SolidPeso molecular:436.6GMA-839
CAS:<p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>Fórmula:C21H31F3O3Pureza:98%Forma y color:SolidPeso molecular:388.46NO-711ME
CAS:<p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>Fórmula:C22H24N2O3Pureza:99.54%Forma y color:SolidPeso molecular:364.44U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Fórmula:C16H23N5Pureza:99.62%Forma y color:SolidPeso molecular:285.39(+)-Bicuculline methiodide
CAS:<p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>Fórmula:C21H20INO6Pureza:99.24%Forma y color:SolidPeso molecular:509.29CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Fórmula:C17H19N3O2Pureza:98%Forma y color:SolidPeso molecular:297.35mGAT3/4-IN-2
CAS:<p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>Fórmula:C26H32ClN3OS2Forma y color:SolidPeso molecular:502.13COR659
CAS:<p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>Fórmula:C16H16ClNO3SPureza:99.75%Forma y color:SolidPeso molecular:337.82Diproqualone
CAS:<p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>Fórmula:C12H14N2O3Forma y color:SolidPeso molecular:234.255ADX71441
CAS:<p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.</p>Fórmula:C19H15ClF2N4O4Forma y color:SolidPeso molecular:436.8Adipiplon
CAS:<p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>Fórmula:C18H18FN7Forma y color:SolidPeso molecular:351.38PZ-II-029
CAS:<p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>Fórmula:C18H15N3O3Pureza:99.79%Forma y color:SolidPeso molecular:321.33CGP 64213
CAS:<p>CGP 64213 is a GABAb receptor agonist.</p>Fórmula:C26H36IN2O7PPureza:98%Forma y color:SolidPeso molecular:646.45(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84GABAA receptor agent 2 TFA
CAS:<p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>Fórmula:C22H22F3N3O3Forma y color:SolidPeso molecular:433.42JM-1232
CAS:<p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>Fórmula:C24H27N3O2Forma y color:SolidPeso molecular:389.49CGP-54626 free base
CAS:<p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>Fórmula:C18H28Cl2NO3PPureza:98%Forma y color:SolidPeso molecular:408.3Afizagabar
CAS:<p>Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.</p>Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.38mGAT-IN-1
CAS:<p>mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).</p>Fórmula:C28H34ClN3O2S2Forma y color:SolidPeso molecular:544.17CGP 54626 hydrochloride
CAS:<p>CGP 54626 hydrochloride is a GABAB receptor antagonist.</p>Fórmula:C18H29Cl3NO3PPureza:98%Forma y color:SolidPeso molecular:444.76Piperidine-4-sulfonic acid
CAS:<p>Piperidine-4-sulfonic acid is a potent GABA agonist, demonstrating an IC50 value of 0.034 μM for the inhibition of H-GABA binding [1].</p>Fórmula:C5H11NO3SPureza:98%Forma y color:SolidPeso molecular:165.21CGP36216 hydrochloride
CAS:<p>CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].</p>Fórmula:C5H15ClNO2PForma y color:SolidPeso molecular:187.6L 663581
CAS:<p>L 663581 is the benzodiazepine receptor partial agonist.</p>Fórmula:C17H16ClN5O2Pureza:98%Forma y color:SolidPeso molecular:357.796,2'-Dihydroxyflavone
CAS:<p>6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.</p>Fórmula:C15H10O4Pureza:99.44% - 99.67%Forma y color:SolidPeso molecular:254.24NCS-382 sodium
CAS:<p>NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological disease</p>Fórmula:C13H13NaO3Pureza:98%Forma y color:SolidPeso molecular:240.23TPA 023
CAS:<p>TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).</p>Fórmula:C20H22FN7OPureza:99.75%Forma y color:SolidPeso molecular:395.43SCS
CAS:<p>SCS is a GABAA receptor antagonist.</p>Fórmula:C14H12N2O3Pureza:99.73%Forma y color:SolidPeso molecular:256.26L-822179
CAS:<p>L-822179 (α5IA) is a selective inverse agonist for the Α5 subtype of GABAA receptor with higher intrinsic activity at the A5 subtype than other drugs.</p>Fórmula:C17H14N8O2Pureza:98.5% - 99.61%Forma y color:SolidPeso molecular:362.35PHP 501 trifluoroacetate
CAS:<p>GABAA antagonist</p>Fórmula:C20H21N3OPureza:98%Forma y color:SolidPeso molecular:319.4GABA-IN-4
CAS:<p>GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.</p>Fórmula:C17H13ClN2O2Forma y color:SolidPeso molecular:312.75Moxetomidate
CAS:<p>Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.</p>Fórmula:C15H18N2O3Forma y color:SolidPeso molecular:274.315Desmethylflunitrazepam
CAS:<p>Desmethylflunitrazepam (Norflunitrazepam) is a benzodiazepine derivative and an active metabolite of Flunitrazepam.</p>Fórmula:C15H10FN3O3Forma y color:SolidPeso molecular:299.26SGE-516
CAS:<p>SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.</p>Fórmula:C23H35N3O2Pureza:98%Forma y color:SolidPeso molecular:385.54Cyproflanilide
CAS:<p>Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.</p>Fórmula:C28H17BrF12N2O2Forma y color:SolidPeso molecular:721.33Tuclazepam
CAS:<p>Tuclazepam (KC 1956) is a derivative of the benzodiazepine class of drugs, exhibiting anti-anxiety and sedative properties.</p>Fórmula:C17H16Cl2N2OForma y color:SolidPeso molecular:335.23GABAA receptor agonist 1
<p>Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.</p>Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45ZK 93426 hydrochloride
CAS:<p>benzodiazepine receptor antagonist,competitive</p>Fórmula:C18H21ClN2O3Pureza:98%Forma y color:SolidPeso molecular:348.82S-8510 phosphate
CAS:<p>S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).</p>Fórmula:C12H13N4O6PPureza:98%Forma y color:SolidPeso molecular:340.23Gabaculine HCl
CAS:<p>Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.</p>Fórmula:C7H10ClNO2Forma y color:SolidPeso molecular:175.61EF1502 free base
CAS:<p>EF1502 is a potent and selective GABA transporter inhibitor.</p>Fórmula:C22H26N2O2S2Pureza:98%Forma y color:SolidPeso molecular:414.58Fletazepam
CAS:<p>Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.</p>Fórmula:C17H13ClF4N2Forma y color:SolidPeso molecular:356.74BGT1-IN-1
CAS:<p>BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.</p>Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.14GABAA receptor agonist 2
<p>Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.</p>Fórmula:C22H36O5Forma y color:SolidPeso molecular:380.52TP003
CAS:<p>TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.</p>Fórmula:C23H16F3N3OPureza:99.17%Forma y color:SolidPeso molecular:407.39(-)-Bicuculline methobromide
CAS:<p>(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .</p>Fórmula:C21H20BrNO6Forma y color:WhitePeso molecular:462.292-AEMP TFA
CAS:<p>2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.</p>Fórmula:C3H10NO3PPureza:98%Forma y color:SolidPeso molecular:139.0913-Methylglutaconic acid
CAS:<p>3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].</p>Fórmula:C6H8O4Pureza:98%Forma y color:SolidPeso molecular:144.13Alfadolone acetate
CAS:<p>Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C23H34O5Forma y color:SolidPeso molecular:390.51Pazinaclone
CAS:<p>Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.</p>Fórmula:C25H23ClN4O4Pureza:97.79% - 99.07%Forma y color:SolidPeso molecular:478.93CGP 44532
CAS:<p>CGP 44532 a GABAB receptor agonist.</p>Fórmula:C4H12NO3PPureza:98%Forma y color:SolidPeso molecular:153.12Pipequaline
CAS:<p>Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.</p>Fórmula:C22H24N2Pureza:98%Forma y color:SolidPeso molecular:316.44Ref: TM-T4655
Producto descatalogadoXilmenolone
CAS:<p>Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].</p>Fórmula:C26H37N3O2Pureza:98%Forma y color:SolidPeso molecular:423.59Ref: TM-T78670
Producto descatalogadoCGP 56999A
CAS:<p>CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.</p>Fórmula:C19H30NO5PPureza:98%Forma y color:SolidPeso molecular:383.42
