Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 336 productos de "Receptor GABA"
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CP-409092 hydrochloride
CAS:<p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>Fórmula:C17H20ClN3O2Forma y color:SolidPeso molecular:333.81CGP 46381
CAS:<p>CGP 46381 is a GABAB receptor antagonist.</p>Fórmula:C10H22NO2PPureza:98%Forma y color:White SolidPeso molecular:219.26GABAA receptor agent 5
CAS:<p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>Fórmula:C21H25N3O2SForma y color:SolidPeso molecular:383.51BGT1-IN-9
CAS:<p>BGT1-IN-9 is an M1 muscarinic agonist.</p>Fórmula:C5H10ClN3O2Forma y color:SolidPeso molecular:179.605CCD-3693
CAS:<p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>Fórmula:C21H31F3O2Pureza:98%Forma y color:SolidPeso molecular:372.46GABA-AT-IN-1
CAS:<p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4GABAA receptor agent 8
CAS:<p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>Fórmula:C19H16N4OForma y color:SolidPeso molecular:316.36ZAPA sulfate
CAS:<p>GABAA receptors agonist</p>Fórmula:C4H8N2O6S2Pureza:98%Forma y color:SolidPeso molecular:244.25TPMPA
CAS:<p>GABAA-ρ antagonist</p>Fórmula:C6H12NO2PPureza:98%Forma y color:SolidPeso molecular:161.14TG41
CAS:<p>TG41 is a GABAA receptors positive modulator.</p>Fórmula:C18H13BrCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:440.12FG8119
CAS:<p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>Fórmula:C17H15N5O2Pureza:>99.99%Forma y color:SolidPeso molecular:321.33GABAA receptor agent 6
CAS:<p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41TB 21007
CAS:<p>GABAA receptor inverse agonist</p>Fórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5SL-651498
CAS:<p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42Bamaluzole
CAS:<p>Bamaluzole is an agonist of GABA receptor.</p>Fórmula:C14H12ClN3OPureza:98%Forma y color:SolidPeso molecular:273.72NAP-1
CAS:<p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>Fórmula:C20H18ClNO2Forma y color:SolidPeso molecular:339.82GABAA receptor agent 7
CAS:<p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>Fórmula:C18H13ClN4OForma y color:SolidPeso molecular:336.77MRK-623
CAS:<p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>Fórmula:C20H17FN4OForma y color:SolidPeso molecular:348.37Etbicyphat
CAS:<p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>Fórmula:C6H11O4PForma y color:SolidPeso molecular:178.12TCS 1105
CAS:<p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>Fórmula:C17H13FN2O2Pureza:99.75%Forma y color:SolidPeso molecular:296.3Pipazethate
CAS:<p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>Fórmula:C21H25N3O3SForma y color:SolidPeso molecular:399.51NNC052090
CAS:<p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54RU 33965
CAS:<p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>Fórmula:C16H15N3O2Pureza:98%Forma y color:SolidPeso molecular:281.31ZK93423
CAS:<p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43GABAA receptor modulator-2
CAS:<p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>Fórmula:C22H22FN3O5SForma y color:SolidPeso molecular:459.49Carburazepam
CAS:<p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>Fórmula:C17H16ClN3O2Pureza:98%Forma y color:SolidPeso molecular:329.78UMB68 sodium
CAS:<p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.</p>Fórmula:C6H12NaO3Forma y color:SolidPeso molecular:155.149(+)-Nipecotic acid
CAS:<p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>Fórmula:C6H11NO2Pureza:99.38%Forma y color:SolidPeso molecular:129.16(S)-SNAP5114
CAS:<p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>Fórmula:C30H35NO6Pureza:97%Forma y color:SolidPeso molecular:505.6Radequinil
CAS:<p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>Fórmula:C18H14N4O3Pureza:98%Forma y color:SolidPeso molecular:334.333α,21-Dihydroxy-5α-pregnan-20-one
CAS:<p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>Fórmula:C21H34O3Pureza:98.00%Forma y color:SolidPeso molecular:334.49Chlormethiazole edisylate
CAS:<p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>Fórmula:C8H14ClNO6S3Pureza:98%Forma y color:SolidPeso molecular:351.85COR628
CAS:<p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>Fórmula:C16H23NO3SForma y color:SolidPeso molecular:309.42trans-4-Hydroxycrotonic acid
CAS:<p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>Fórmula:C4H6O3Pureza:98%Forma y color:SolidPeso molecular:102.09LY 81067
CAS:<p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>Fórmula:C22H24N4OForma y color:SolidPeso molecular:360.45U 90042
CAS:<p>GABAA receptor ligand</p>Fórmula:C17H13ClN6OPureza:98%Forma y color:SolidPeso molecular:352.78COR627
CAS:<p>COR627 is the GABA receptor positive allosteric modulator.</p>Fórmula:C20H27NO3SPureza:98%Forma y color:SolidPeso molecular:361.5CPP-115
CAS:<p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>Fórmula:C7H9F2NO2Forma y color:SolidPeso molecular:177.15JY-XHe-053
CAS:<p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>Fórmula:C22H16FN3O2Pureza:98%Forma y color:SolidPeso molecular:373.38HIE-124
CAS:<p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>Fórmula:C10H12N2O3SPureza:98%Forma y color:SolidPeso molecular:240.28Suclofenide
CAS:<p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>Fórmula:C16H13ClN2O4SPureza:98%Forma y color:SolidPeso molecular:364.8(S)-Baclofen
CAS:<p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>Fórmula:C10H12ClNO2Pureza:98%Forma y color:SolidPeso molecular:213.66ABP-700
CAS:<p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>Fórmula:C17H18N2O4Pureza:98%Forma y color:SolidPeso molecular:314.34DAA-1097
CAS:<p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>Fórmula:C24H24ClNO3Pureza:98%Forma y color:SolidPeso molecular:409.91(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:<p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>Fórmula:C9H9NO5Pureza:98%Forma y color:SolidPeso molecular:211.17PNU-107484A
CAS:<p>PNU-107484A is a unique GABA(A) receptor ligand.</p>Fórmula:C18H23ClN6Pureza:98%Forma y color:SolidPeso molecular:358.87GS 39783
CAS:<p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>Fórmula:C15H23N5O2SPureza:99.92%Forma y color:SolidPeso molecular:337.44SCH 50911
CAS:<p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>Fórmula:C8H15NO3Pureza:98%Forma y color:SolidPeso molecular:173.21Anxiolytic/nonsedative agent-1
CAS:<p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>Fórmula:C18H15N3O4Pureza:98.61%Forma y color:SolidPeso molecular:337.33SCH 50911 hydrochloride
CAS:<p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>Fórmula:C8H16ClNO3Pureza:98%Forma y color:SolidPeso molecular:209.67
