Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 373 productos de "Receptor GABA"
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Alfadolone
CAS:Alfadolone is an anesthetic derivative of pregnanedione.Fórmula:C21H32O4Forma y color:SolidPeso molecular:348.48Y 23684
CAS:Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.Fórmula:C18H13ClN2O2SPureza:98%Forma y color:SolidPeso molecular:356.83Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Fórmula:C18H12Cl2N2OForma y color:SolidPeso molecular:343.21Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Fórmula:C13H25NO2Forma y color:SolidPeso molecular:227.34Ref: TM-T72977
1mg37,00€5mg72,00€1mL*10mM (DMSO)79,00€10mg99,00€25mg169,00€50mg229,00€100mg320,00€200mg479,00€Ro 19-4603
CAS:Benzodiazepine inverse agonistFórmula:C15H17N3O3SPureza:98%Forma y color:SolidPeso molecular:319.38Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Fórmula:C14H12ClN3OPureza:98%Forma y color:SolidPeso molecular:273.72SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Fórmula:C23H20FN3O2Pureza:98%Forma y color:SolidPeso molecular:389.42TB 21007
CAS:GABAA receptor inverse agonistFórmula:C15H17NO2S3Pureza:98%Forma y color:SolidPeso molecular:339.5Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Fórmula:C16H25ClN4O2Pureza:99.52%Forma y color:SolidPeso molecular:340.85ZK-91296
CAS:ZK-91296: GABA agonist, lowers anxiety without sedation, may target specific BZ receptor subtype.Fórmula:C23H22N2O4Pureza:98%Forma y color:SolidPeso molecular:390.43DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Fórmula:C18H10Br2ClN3OSForma y color:SolidPeso molecular:511.623α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Fórmula:C21H34O3Pureza:98.00%Forma y color:SolidPeso molecular:334.49GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Fórmula:C18H25N3O2Forma y color:SolidPeso molecular:315.41SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Fórmula:C8H15NO3Forma y color:SolidPeso molecular:173.21GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Fórmula:C17H24N2OForma y color:SolidPeso molecular:272.39Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Fórmula:C14H22ClNOPureza:98%Forma y color:SolidPeso molecular:255.783-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Fórmula:C20H30N2O10S2Pureza:98%Forma y color:SolidPeso molecular:522.59Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Fórmula:C15H14N6O3Pureza:98%Forma y color:SolidPeso molecular:326.31Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Fórmula:C15H15N3O3Forma y color:SolidPeso molecular:285.3Phaclofen
CAS:GABAB antagonistFórmula:C9H13ClNO3PPureza:99.32%Forma y color:White SolidPeso molecular:249.63Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Fórmula:C20H22ClN5O3SPureza:98%Forma y color:SolidPeso molecular:447.94Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Fórmula:C15H14ClN3O3Forma y color:SolidPeso molecular:319.74mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Fórmula:C26H31ClN2O2S2Forma y color:SolidPeso molecular:503.12GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Fórmula:C23H18N2O6Forma y color:SolidPeso molecular:418.4AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Fórmula:C19H29NO5Pureza:98.19% - 99.55%Forma y color:SolidPeso molecular:351.44CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Fórmula:C21H31F3O2Pureza:98%Forma y color:SolidPeso molecular:372.462-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Fórmula:C9H12ClNO4SPureza:98.56%Forma y color:White SolidPeso molecular:265.71CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFórmula:C18H19N3O2Pureza:99.61%Forma y color:SolidPeso molecular:309.36SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Fórmula:C18H18N4O3Pureza:98%Forma y color:SolidPeso molecular:338.36NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Fórmula:C21H22N2O3Pureza:99.70%Forma y color:SolidPeso molecular:350.41(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:98%Forma y color:SolidPeso molecular:250.12U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Fórmula:C16H24ClN5Pureza:98%Forma y color:SolidPeso molecular:321.85E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Fórmula:C9H8F4N2O2SPureza:98.22% - 98.54%Forma y color:SolidPeso molecular:284.23CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Fórmula:C18H17N3O3Pureza:99.06% - 99.74%Forma y color:SolidPeso molecular:323.35(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Fórmula:C6H11NO2Pureza:99.38%Forma y color:SolidPeso molecular:129.16Org 20599
CAS:GABAA receptor agonistFórmula:C25H40ClNO3Pureza:98%Forma y color:SolidPeso molecular:438.04U-101017
CAS:U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.Fórmula:C23H27ClN4O3Pureza:98%Forma y color:SolidPeso molecular:442.94BPDBA
CAS:BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 andFórmula:C19H20Cl2N2OPureza:99.43% - 99.95%Forma y color:SolidPeso molecular:363.28Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Fórmula:C17H17N3O2Pureza:97.44% - 98.25%Forma y color:SolidPeso molecular:295.34Suriclone
CAS:Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Forma y color:SolidPeso molecular:477.99Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Fórmula:C26H25ClN2O3Pureza:98.54%Forma y color:SolidPeso molecular:448.94Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Fórmula:C15H14ClN3O3Pureza:99.46%Forma y color:SolidPeso molecular:319.74Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Fórmula:C8H6ClF3N2OSPureza:99.76%Forma y color:SolidPeso molecular:270.66DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Fórmula:C14H12FNOPureza:99.51% - 99.56%Forma y color:SolidPeso molecular:229.25Ref: TM-T11106
1mg109,00€2mg163,00€1mL*10mM (DMSO)208,00€5mg241,00€10mg354,00€25mg532,00€50mg745,00€100mg1.018,00€500mg2.035,00€Nerisopam
CAS:Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.Fórmula:C18H19N3O2Pureza:98.52%Forma y color:SolidPeso molecular:309.36Ref: TM-T28159
1mg88,00€5mg190,00€1mL*10mM (DMSO)256,00€10mg286,00€25mg464,00€50mg672,00€100mg945,00€200mg1.279,00€Fengabine
CAS:Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.Fórmula:C17H17Cl2NOPureza:99.37%Forma y color:SolidPeso molecular:322.23Panadiplon
CAS:Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment ofFórmula:C18H17N5O2Pureza:98.30% - 98.94%Forma y color:SolidPeso molecular:335.36Progabide
CAS:Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.Fórmula:C17H16ClFN2O2Pureza:99.68%Forma y color:SolidPeso molecular:334.77Ref: TM-T16581
2mgA consultar5mg55,00€1mL*10mM (DMSO)62,00€10mg84,00€25mg150,00€50mg219,00€100mg340,00€Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Fórmula:C4H7BrN2O2Pureza:98.13%Forma y color:Off-White PowderPeso molecular:195.01Ref: TM-T20657
1mg113,00€2mg169,00€1mL*10mM (DMSO)205,00€5mg240,00€10mg385,00€25mg622,00€50mg898,00€100mg1.198,00€500mg2.422,00€Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Fórmula:C19H20ClN3OPureza:98.42%Forma y color:SolidPeso molecular:341.83
