Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 363 productos para "Receptor GABA".
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Fletazepam
CAS:Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.Fórmula:C17H13ClF4N2Forma y color:SolidPeso molecular:356.74ZK 93426 hydrochloride
CAS:benzodiazepine receptor antagonist,competitiveFórmula:C18H21ClN2O3Pureza:98%Forma y color:SolidPeso molecular:348.82Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Fórmula:C4H6N2OSPureza:98%Forma y color:SolidPeso molecular:130.17CGS-9895
CAS:CGS-9895 is a GABA antagonist that operates by interacting with the benzodiazepine binding site on GABA receptors containing the γ subunit (ag).Fórmula:C17H13N3O2Forma y color:SolidPeso molecular:291.304BGT1-IN-1
CAS:BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.14S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Fórmula:C12H13N4O6PPureza:98%Forma y color:SolidPeso molecular:340.23GABA-IN-4
CAS:GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.Fórmula:C17H13ClN2O2Forma y color:SolidPeso molecular:312.75Moxetomidate
CAS:Moxetomidate is a GABAA receptor (GABAA receptor) agonist with hypnotic properties.Fórmula:C15H18N2O3Forma y color:SolidPeso molecular:274.315Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Fórmula:C7H10ClNO2Forma y color:SolidPeso molecular:175.61GABAA receptor agonist 2
Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.Fórmula:C22H36O5Forma y color:SolidPeso molecular:380.52TP003
CAS:TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.Fórmula:C23H16F3N3OPureza:99.17%Forma y color:White SolidPeso molecular:407.39SGE-516
CAS:SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.Fórmula:C23H35N3O2Pureza:98%Forma y color:SolidPeso molecular:385.54Cyproflanilide
CAS:Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.Fórmula:C28H17BrF12N2O2Forma y color:SolidPeso molecular:721.33
