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Receptor GABA

Receptor GABA

Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.

Se han encontrado 351 productos de "Receptor GABA"

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  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Fórmula:C17H20N2O3
    Pureza:99.62%
    Forma y color:Solid Crystalline
    Peso molecular:300.35
  • E2730

    CAS:
    E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.
    Fórmula:C9H8F4N2O2S
    Pureza:98.22% - 98.54%
    Forma y color:Solid
    Peso molecular:284.23
  • U-89843A

    CAS:
    U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].
    Fórmula:C16H24ClN5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:321.85
  • (R)-Baclofen hydrochloride

    CAS:
    Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.
    Fórmula:C10H13Cl2NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:250.12
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Fórmula:C16H25ClN4O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:340.85
  • RO 4938581

    CAS:
    RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).
    Fórmula:C13H8BrF2N5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.14
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Fórmula:C19H29NO5
    Pureza:98.19% - 99.55%
    Forma y color:Solid
    Peso molecular:351.44
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Fórmula:C9H13ClNO3P
    Pureza:99.32%
    Forma y color:White Solid
    Peso molecular:249.63
  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Fórmula:C21H19F2N3O3
    Pureza:99.57% - 99.95%
    Forma y color:Solid
    Peso molecular:399.39
  • DSP-0565

    CAS:
    DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.
    Fórmula:C14H12FNO
    Pureza:99.51% - 99.56%
    Forma y color:Solid
    Peso molecular:229.25
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Fórmula:C19H20ClN3O
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:341.83
  • Progabide

    CAS:
    <p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>
    Fórmula:C17H16ClFN2O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:334.77
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Fórmula:C21H23Cl2N3O
    Pureza:99.56% - 99.97%
    Forma y color:White To Off-White Solid
    Peso molecular:404.33
  • Muscimol HBr

    CAS:
    Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Forma y color:Off-White Powder
    Peso molecular:195.01
  • L-838417

    CAS:
    L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders
    Fórmula:C19H19F2N7O
    Pureza:98.12% - 99.70%
    Forma y color:Solid
    Peso molecular:399.4
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Fórmula:C17H19ClN2O4
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:350.8
  • Sarmazenil

    CAS:
    <p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>
    Fórmula:C15H14ClN3O3
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:319.74
  • NS-2710

    CAS:
    NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.
    Fórmula:C22H20N4O
    Pureza:99.7% - 99.82%
    Forma y color:Solid
    Peso molecular:356.42
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Fórmula:C18H17N5O2
    Pureza:98.30% - 98.94%
    Forma y color:Solid
    Peso molecular:335.36
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Fórmula:C17H14O6
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:314.29