Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 363 productos para "Receptor GABA".
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(+)-Bicuculline methiodide
CAS:(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.Fórmula:C21H20INO6Pureza:99.24%Forma y color:SolidPeso molecular:509.29CP-409092
CAS:CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.Fórmula:C17H19N3O2Pureza:98%Forma y color:SolidPeso molecular:297.35mGAT3/4-IN-2
CAS:mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.Fórmula:C26H32ClN3OS2Forma y color:SolidPeso molecular:502.13COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Fórmula:C16H16ClNO3SPureza:99.75%Forma y color:SolidPeso molecular:337.82Ref: TM-T36520
1mg38,00€5mg86,00€1mL*10mM (DMSO)94,00€10mg123,00€25mg215,00€50mg299,00€100mg411,00€200mg560,00€Diproqualone
CAS:Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].Fórmula:C12H14N2O3Forma y color:SolidPeso molecular:234.255ADX71441
CAS:ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.Fórmula:C19H15ClF2N4O4Forma y color:SolidPeso molecular:436.8Adipiplon
CAS:Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.Fórmula:C18H18FN7Forma y color:SolidPeso molecular:351.38PZ-II-029
CAS:PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.Fórmula:C18H15N3O3Pureza:99.79%Forma y color:Yellow SolidPeso molecular:321.33Ref: TM-T28479
1mg50,00€5mg105,00€10mg167,00€1mL*10mM (DMSO)192,00€25mg289,00€50mg447,00€100mg685,00€500mg1.378,00€CGP 64213
CAS:CGP 64213 is a GABAb receptor agonist.Fórmula:C26H36IN2O7PPureza:98%Forma y color:SolidPeso molecular:646.45CGP 55845 hydrochloride
CAS:CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].Fórmula:C18H23Cl3NO3PForma y color:SolidPeso molecular:438.71(-)-Bicuculline methochloride
CAS:(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.Fórmula:C21H20ClNO6Pureza:98%Forma y color:SolidPeso molecular:417.84GABAA receptor agent 2 TFA
CAS:Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.Fórmula:C22H22F3N3O3Forma y color:SolidPeso molecular:433.42JM-1232
CAS:JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.Fórmula:C24H27N3O2Forma y color:SolidPeso molecular:389.49CGP-54626 free base
CAS:CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).Fórmula:C18H28Cl2NO3PPureza:98%Forma y color:SolidPeso molecular:408.3Afizagabar
CAS:Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.38mGAT-IN-1
CAS:mGAT-IN-1 is a potent, non-selective GAT inhibitor that inhibits mGAT3 activity well (IC50: 2.5 μM, pIC50: 5.61).Fórmula:C28H34ClN3O2S2Forma y color:SolidPeso molecular:544.17L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Fórmula:C17H16ClN5O2Pureza:98%Forma y color:SolidPeso molecular:357.796,2'-Dihydroxyflavone
CAS:6,2'-Dihydroxyflavone is a novel antagonist of GABAA receptor.Fórmula:C15H10O4Pureza:99.44% - 99.67%Forma y color:Yellow SolidPeso molecular:254.24NCS-382 sodium
CAS:NCS-382 (sodium) is a potent antagonist of the GABA receptor, exhibiting anti-sedative and anti-hypnotic properties, with applications in neurological diseaseFórmula:C13H13NaO3Pureza:98%Forma y color:SolidPeso molecular:240.23SCS
CAS:SCS is a GABAA receptor antagonist.Fórmula:C14H12N2O3Pureza:99.73%Forma y color:SolidPeso molecular:256.26
