Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 371 productos de "Receptor GABA"
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GABAA receptor agent 1
CAS:GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.Fórmula:C13H8ClN3O2Pureza:99.31%Forma y color:SolidPeso molecular:273.67Ref: TM-T11349
1mg35,00€5mg79,00€10mg111,00€25mg215,00€50mg323,00€100mg469,00€200mg647,00€1mL*10mM (DMSO)86,00€Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Fórmula:C25H14BrF11N2O2Pureza:99.82%Forma y color:SolidPeso molecular:663.29Ref: TM-T10618
1mg52,00€2mg74,00€5mg111,00€10mg180,00€25mg358,00€50mg588,00€100mg835,00€1mL*10mM (DMSO)131,00€Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFórmula:C15H14FN3O3Pureza:99.72% - 99.98%Forma y color:Less Crystals Colourless CrystalsPeso molecular:303.29Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Fórmula:C10H12ClNO2Pureza:98% - >99.99%Forma y color:1992)Peso molecular:213.66Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Fórmula:C9H17NO3Pureza:99.87%Forma y color:SolidPeso molecular:187.24γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Fórmula:C4H9NO2Pureza:99.95%Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecular:103.12LAU159
CAS:LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Fórmula:C17H12ClN3O2Pureza:98.7% - 99.38%Forma y color:SolidPeso molecular:325.75Ref: TM-T11822
1mg110,00€2mg160,00€5mg219,00€10mg395,00€25mg653,00€50mg888,00€100mg1.243,00€500mg2.493,00€3,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFórmula:C12H14O5Pureza:98.91%Forma y color:SolidPeso molecular:238.24Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Fórmula:C8H14N2O4SPureza:98.38% - 99.83%Forma y color:SolidPeso molecular:234.27Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFórmula:C56H81NO15Pureza:98.68%Forma y color:SolidPeso molecular:1008.2566,7-dimethylisatin
CAS:6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Fórmula:C10H9NO2Pureza:98.98%Forma y color:SolidPeso molecular:175.18α-Casozepine
CAS:α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.Fórmula:C60H94N14O16Forma y color:SolidPeso molecular:1267.47epi-Aszonalenin A
CAS:epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Fórmula:C25H25N3O3Forma y color:SolidPeso molecular:415.48Nipecotic acid
CAS:Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.
Fórmula:C6H11NO2Forma y color:Off-White To Pale Yellow-Beige PowderPeso molecular:129.16Lesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Fórmula:C13H17FNO5PSForma y color:SolidPeso molecular:349.31Flufiprole
CAS:Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.Fórmula:C16H10Cl2F6N4OSForma y color:SolidPeso molecular:491.24Atagabalin
CAS:Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Fórmula:C10H19NO2Forma y color:SolidPeso molecular:185.26Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Fórmula:C19H38ClN5O2SForma y color:SolidPeso molecular:436.06Anisatin
Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.Fórmula:C15H20O8Forma y color:SolidPeso molecular:328.317Nitrazolam
CAS:Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.Fórmula:C17H13N5O2Forma y color:SolidPeso molecular:319.32
