Receptor GABA
Los receptores GABA son los principales receptores de neurotransmisores inhibitorios en el sistema nervioso central, desempeñando un papel crítico en la regulación de la excitabilidad neuronal y el mantenimiento del equilibrio entre excitación e inhibición. La disfunción de los receptores GABA está implicada en varios trastornos neurológicos y psiquiátricos, como la epilepsia, la ansiedad y la depresión. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores GABA para apoyar su investigación en neurobiología, salud mental y desarrollo terapéutico.
Se han encontrado 367 productos para "Receptor GABA".
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Furosemide sodium
CAS:Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Fórmula:C12H10ClN2NaO5SPureza:99.52% - >99.99%Forma y color:SolidPeso molecular:352.73Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Fórmula:C8H13NO2Pureza:99.89%Forma y color:SolidPeso molecular:155.19Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Fórmula:C10H12ClNO2Pureza:98% - 99.94%Forma y color:White SolidPeso molecular:213.66Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFórmula:C15H14FN3O3Pureza:99.72% - 99.98%Forma y color:White SolidPeso molecular:303.29Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Fórmula:C6H10N4Pureza:99.67% - 99.90%Forma y color:SolidPeso molecular:138.17Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Fórmula:C11H12ClNO3SPureza:99.86% - >99.99%Forma y color:White SolidPeso molecular:273.74LAU159
CAS:LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Fórmula:C17H12ClN3O2Pureza:98.7% - 99.38%Forma y color:Yellow SolidPeso molecular:325.75Ref: TM-T11822
1mg110,00€2mg160,00€5mg219,00€10mg395,00€25mg653,00€50mg888,00€100mg1.243,00€500mg2.493,00€Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Fórmula:C9H17NO3Pureza:99.87%Forma y color:White SolidPeso molecular:187.24Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Fórmula:C8H14N2O4SPureza:98.24% - 99.83%Forma y color:SolidPeso molecular:234.27Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFórmula:C56H81NO15Pureza:98.68%Forma y color:SolidPeso molecular:1008.2566,7-dimethylisatin
CAS:6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.Fórmula:C10H9NO2Pureza:98.98%Forma y color:SolidPeso molecular:175.18α-Casozepine
CAS:α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.Fórmula:C60H94N14O16Pureza:99.81%Forma y color:SolidPeso molecular:1267.47epi-Aszonalenin A
CAS:epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Fórmula:C25H25N3O3Forma y color:SolidPeso molecular:415.48Nipecotic acid
CAS:Nipecotic acid ,with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Nipecotic acid provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Fórmula:C6H11NO2Forma y color:Off-White To Pale Yellow-Beige PowderPeso molecular:129.16Lesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Fórmula:C13H17FNO5PSForma y color:SolidPeso molecular:349.31Afizagabar
CAS:Afizagabar, a first-in-class α5-GABAAR antagonist, IC50: 585 nM, Ki: 66 nM, may boost memory.Fórmula:C19H12FN3O2SForma y color:SolidPeso molecular:365.38Flufiprole
CAS:Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.Fórmula:C16H10Cl2F6N4OSForma y color:SolidPeso molecular:491.24Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Fórmula:C19H38ClN5O2SForma y color:SolidPeso molecular:436.06Atagabalin
CAS:Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.Fórmula:C10H19NO2Forma y color:SolidPeso molecular:185.26DAA-1106
CAS:DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Fórmula:C23H22FNO4Pureza:99.54%Forma y color:SolidPeso molecular:395.42
