Caseína quinasa
Las caseína quinasas son una familia de quinasas de proteínas serina/treonina que regulan varios procesos celulares, incluyendo la reparación del ADN, los ritmos circadianos y la transducción de señales. Estas quinasas están involucradas en la fosforilación de numerosas proteínas y están implicadas en enfermedades como el cáncer, los trastornos neurodegenerativos y los síndromes metabólicos. En CymitQuimica, ofrecemos una selección de inhibidores de caseína quinasa para apoyar su investigación en transducción de señales, regulación del ciclo celular y desarrollo terapéutico.
Se han encontrado 151 productos para "Caseína quinasa".
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IWP-2
CAS:IWP-2 is a Wnt pathway inhibitor and an ATP-competitive CK1δ inhibitor. IWP-2 inhibits self-renewal of embryonic stem cells. Cost effective and quality assured.Fórmula:C22H18N4O2S3Pureza:96.1% - 99.86%Forma y color:White SolidPeso molecular:466.599IC261
CAS:IC261 (SU-5607) is a novel inhibitor of CK1, triggers the mitotic checkpoint control. The IC50 of IC261 for CK1 was 16 μM and for Cdk5 is 4.5 mM.Fórmula:C18H17NO4Pureza:98.77% - 99.91%Forma y color:SolidPeso molecular:311.3319LY-294002 hydrochloride
CAS:LY-294002 HCl (NSC 697286) is a stable PI3K inhibitor (IC50: 0.5-0.97 µM) and prevents autophagosome formation.Fórmula:C19H17NO3·HClPureza:99.95% - 99.98%Forma y color:Purple LiquidPeso molecular:343.81LH846
CAS:LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and 2.5 uM for CK1δ, ε and α); exhibits no inhibitory activity at CK2.Fórmula:C16H13ClN2OSPureza:90% - 98.26%Forma y color:SolidPeso molecular:316.805PF-4800567
CAS:PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.Fórmula:C17H18ClN5O2Pureza:99.74% - 99.76%Forma y color:White SolidPeso molecular:359.81XL413
CAS:XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell growth.Fórmula:C14H12ClN3O2Pureza:98.40% - 99.94%Forma y color:SolidPeso molecular:289.717HDAC/CK2-IN-1
CAS:HDAC/CK2-IN-1 (compound 38) acts as an inhibitor of HDAC1 (IC 50 = 1.46 μM), HDAC6 (IC 50 = 0.66 μM), and CK2 (IC 50 = 3.67 μM). It demonstrates promising antiproliferative effects on various cell lines, including Jurkat, MCF-7, HCT-116, and HL-60.Fórmula:C15H18Br4N4O2Forma y color:SolidPeso molecular:605.95CK2/PIM1-IN-1
CAS:CK2/PIM1-IN-1 inhibits CK2 & PIM1 (IC50s: 3.787 & 4.327 μM), aimed for cancer research.Fórmula:C15H9NO4S2Pureza:98%Forma y color:SolidPeso molecular:331.3664,5,6,7-Tetrabromobenzimidazole
CAS:4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].Fórmula:C7H2Br4N2Forma y color:SolidPeso molecular:433.72CK2-IN-9
CAS:CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporterFórmula:C23H29N9OForma y color:SolidPeso molecular:447.54SRPIN-803
CAS:SRPIN-803 is a selective dual SRPK1 and CK2 inhibitor.Fórmula:C14H9F3N4O3SPureza:98%Forma y color:SolidPeso molecular:370.31AMG-548
CAS:AMG-548, oral p38α inhibitor (Ki=0.5 nM), >1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.Fórmula:C29H27N5OPureza:99.91%Forma y color:SolidPeso molecular:461.56BTX161
CAS:BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.Fórmula:C15H16N2O3Forma y color:SolidPeso molecular:272.2991SR-1277
CAS:SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.Fórmula:C21H19N9O3SForma y color:SolidPeso molecular:477.5CK2α-IN-1
CAS:CK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 µM and a Ki of 1.6 µM.CK2α-IN-1 exhibits potential anticancer activity and canFórmula:C16H11N3O4SPureza:98%Forma y color:SolidPeso molecular:341.341TMCB
CAS:CK2 and ERK8 inhibitorFórmula:C11H9Br4N3O2Pureza:98%Forma y color:SolidPeso molecular:534.82Umbralisib sulfate
CAS:Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.Fórmula:C31H26F3N5O7SForma y color:SolidPeso molecular:669.63Quinalizarin
CAS:Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.Fórmula:C14H8O6Pureza:98%Forma y color:SolidPeso molecular:272.2097CK1-IN-2
CAS:CK1-IN-2 (compound Nr.4) is a potent CK1 inhibitor p38a, and is used in DUX4 overexpression-associated diseases, such as muscular dystrophy.Fórmula:C17H12FN3O2Pureza:99.31%Forma y color:SolidPeso molecular:309.29CK2-IN-4
CAS:CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.Fórmula:C18H11N3O4SPureza:99.65%Forma y color:SolidPeso molecular:365.363
