Transporter

DMT1 blocker 2, compound 12f, is a direct inhibitor of divalent metal transporter 1 (DMT1) …

Isoferulic acid is an effective natural antioxidant in both lipid and aqueous media, it may …

WAY-213613 hydrochloride is a potent, selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 with IC 50 of …

LDN-212320 is a glutamate transporter EAAT2 activator. It also enhances EAAT2 levels by >6 fold …

Cinromide is used as a novel anticonvulsant agent.

Benztropine mesylate is a centrally active muscarinic antagonist that has been used in the symptomatic …

Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. …

GPNA hydrochloride is specific glutamine (Gln) transporter ASCT2(SLC1A5) inhibitor. GPNA reversibly induces apoptosis in A549 …

The l-carnitine hydrochloride is a constituent of striated muscle and liver. It is used therapeutically …

Sennidin A, has two hydroxyanthraquinone-like moieties, exerts inhibition on NS3 helicase with IC50 values of …

1β-Hydroxy-2-oxopomolic acid inhibits adipocyte differentiation through downregulation of various adipocytokines by blocking PPARγ and C/EBPα …

DRB18 is a potent pan-class GLUT inhibitor. DRB18 alters energy-related metabolism in A549 cells by …

Gentianine is an effective Swertiamarin derivative, which has anti-diabetic, antipsychotic, anti-inflammatory, hypotensive, diuretic and other …

Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor

Dodoviscin I can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.

GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: …

Dodoviscin H can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.

Dodoviscin J can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.

Sennidin B stimulates glucose incorporation in rat adipocytes.

Dodoviscin A may be a new promising pigmentation-altering agent for cosmetic and therapeutic applications, it …

Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food …

GLUT inhibitor-1 is an orally active GLUT inhibitor with IC50 s of 242 nM and …

Ficusin has antioxidant, antilipidemic and antidiabetic effects, it can lower the levels of fasting blood …

Valbenazine, a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of …

Nepodin has antimalarial, and anti-inflammatory activities, it shows significant cyclooxygenase (COX) inhibitory activity. Nepodin has …

V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets …

Indican is a natural protective compound that is used to protect the liver.

1.(-)-Licarin B has anti-mycobacterial activity.

Tetramethylkaempferol is a PPARγ agonist, it can improve insulin sensitivity by increasing the levels of …

WZB117 is a Glucose Transporter 1 (GLUT1) inhibitor. when IC50 of WZB117 approximate 10 μM, …

1. L-Arginine exhibits anti-atherosclerotic effect. 2. L-Arginine and soy enriched diet are effective in prevention …

BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.

Hemicholinium-3 is a potent and selective choline uptake blocker.

Disodium clodronate tetrahydrate inhibits bone resorption and soft tissue calcification.

Procyanidin A2 is a potential precursor of 5-(3',4'-dihydroxyphenyl)-γ-valerolactone, exhibits antioxidant, anti-inflammary, anti-hyperglycemia, and anti-type 2 …

Rhoifolin is extracted from Turpinia arguya Seem dried leaves.

CB-839(IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for …

Vorolanib is an orally active VEGFR/PDGFR dual inhibitor.

Jujuboside A is a glycoside extracted from Semen Ziziphi Spinosae, having neurophysiological inhibitory effects, used …

Fasentin is an inhibitor of GluT1.

KL-11743 specifically blocks glucose metabolism, triggering an acute collapse in NADH pools and a striking …

α-Cyano-4-hydroxycinnamic acid (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvate transport …

UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 …

AHN 1-055 hydrochloride is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 …

STF-31 is an inhibitor of glucose transporter 1 (GLUT1) with IC50 of 1 μM.

Nefazodone is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior …

Nitrobenzylthioinosine is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.

Marein shows neuroprotective effect on PC12 cell damage induced by methylglyoxal, which is due to …

Phloretin is a well-known inhibitor of eukaryotic urea transporters, blocks VacA-mediated urea and ion transport. …

Tormentic acid is a natural product. It has anticancer, anti-inflammatory, anti-atherogenic , anti-allodynic, and hepatoprotective …

BAY-876 is an orally active and selective inhibitor of glucose transporter 1 (GLUT1, IC50= 2 …

Dotinurad is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).

Nandrolone Decanoate is the decanoate salt form of nandrolone, an anabolic steroid analog of testosterone …

Fraxin is a glucoside of fraxetin.

TCID(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold …

CTPI-2 is an inhibitor of mitochondrial citrate carrier SLC25A1 with(KD : 3.5 μM). CTPI-2 inhibits …

T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) …

F2005-0304 is a thiopyridazine derivative that has been found to increase EAAT2 protein levels in …

Lavendustin B is a Tyrosine Kinase Inhibitor and an inhibitor of HIV-1 integrase (IN) interaction …

WAY-213613 is a potent and selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 (IC50: 85 nM EAAT2). …

DL-TBOA inhibited [14C] glutamate uptake in COS-1 cells expressing human EAAT1 and EAAT2, with Ki …