Transportador
Las proteínas transportadoras están involucradas en el movimiento de moléculas a través de las membranas celulares, desempeñando roles vitales en la absorción de nutrientes, la eliminación de desechos y la resistencia a los medicamentos. Los inhibidores de proteínas transportadoras se utilizan para estudiar la función de estas proteínas en varios procesos fisiológicos y patológicos, incluidos los trastornos metabólicos, el cáncer y la administración de fármacos. Al modular la actividad de los transportadores, los investigadores pueden obtener información sobre los mecanismos de transporte celular y desarrollar nuevas estrategias terapéuticas. En CymitQuimica, ofrecemos una gama de inhibidores de transportadores para apoyar su investigación en farmacología, biología celular y regulación metabólica.
Se han encontrado 44 productos para "Transportador".
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Indican
CAS:Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver.Fórmula:C14H17NO6Pureza:99.78% - 99.92%Forma y color:Yellow SolidPeso molecular:295.29Nefazodone hydrochloride
CAS:Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Forma y color:SolidPeso molecular:506.47Ref: TM-T3275
5mg44,00€1mL*10mM (DMSO)50,00€10mg66,00€25mg114,00€50mg205,00€100mg309,00€200mg447,00€500mg735,00€Vorolanib
CAS:Vorolanib (X-82) is an orally active VEGFR/PDGFR dual inhibitor.Fórmula:C23H26FN5O3Pureza:97.35%Forma y color:SolidPeso molecular:439.48Ref: TM-T8491
1mg101,00€2mg142,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg583,00€50mg842,00€100mg1.144,00€200mg1.521,00€KL-11743
CAS:KL-11743 blocks glucose metabolism, collapses NADH, and increases aspartate, shifting cells to oxidative phosphorylation.Fórmula:C30H30N6O3Pureza:98.46% - 99.57%Forma y color:SolidPeso molecular:522.6Ref: TM-T9558
1mg107,00€5mg222,00€1mL*10mM (DMSO)255,00€10mg358,00€25mg597,00€50mg850,00€100mg1.153,00€UCPH-101
CAS:UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Fórmula:C27H22N2O3Pureza:98.58%Forma y color:White SolidPeso molecular:422.48Ref: TM-T4138
1mg50,00€2mg75,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg203,00€25mg409,00€50mg655,00€100mg954,00€200mg1.288,00€AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Fórmula:C21H24ClF2NOPureza:99.89%Forma y color:SolidPeso molecular:379.87Ref: TM-T39429
2mg34,00€5mg49,00€1mL*10mM (DMSO)50,00€10mg75,00€25mg130,00€50mg192,00€100mg295,00€200mg442,00€Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.Fórmula:C17H17N5O6SPureza:99.69% - 99.74%Forma y color:White SolidPeso molecular:419.41WAY-213613
CAS:WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.Fórmula:C16H13BrF2N2O4Pureza:98%Forma y color:SolidPeso molecular:415.19Tormentic acid
CAS:Tormentic acid is a natural product. It has anticancer, anti-inflammatory, anti-atherogenic , anti-allodynic, and hepatoprotective properties,Fórmula:C30H48O5Pureza:97.02% - 99.86%Forma y color:SolidPeso molecular:488.7BAY-876
CAS:BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.Fórmula:C24H16F4N6O2Pureza:98.61% - 99.78%Forma y color:White SolidPeso molecular:496.42Ref: TM-T3713
1mg55,00€2mg78,00€5mg95,00€1mL*10mM (DMSO)96,00€10mg131,00€25mg221,00€50mg334,00€100mg533,00€200mg755,00€Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Fórmula:C14H9Cl2NO4SPureza:97.43% - 98.04%Forma y color:SolidPeso molecular:358.2Ref: TM-T15160
1mg123,00€1mL*10mM (DMSO)226,00€5mg289,00€10mg447,00€25mg737,00€50mg982,00€100mg1.341,00€CTPI-2
CAS:CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.Fórmula:C13H9ClN2O6SPureza:97.23%Forma y color:SolidPeso molecular:356.74Valbenazine
CAS:Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.Fórmula:C24H38N2O4Pureza:97.58%Forma y color:SolidPeso molecular:418.57Ref: TM-T7147
1mg46,00€2mg58,00€5mg101,00€1mL*10mM (DMSO)113,00€10mg167,00€25mg313,00€50mg485,00€100mg708,00€200mg964,00€Clodronate disodium tetrahydrate
CAS:Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.Fórmula:CH10Cl2Na2O10P2Pureza:98%Forma y color:SolidPeso molecular:360.92TCID
CAS:TCID (UCH-L3 Inhibitor)(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold selectivity to L1.Fórmula:C9H2Cl4O2Pureza:98.87% - 99.34%Forma y color:SolidPeso molecular:283.92WZB117
CAS:WZB117 inhibits GLUT1; IC50 ~10μM slows A549 lung & MCF7 breast cancer cell growth.Fórmula:C20H13FO6Pureza:99.03% - 99.18%Forma y color:White SolidPeso molecular:368.31Ref: TM-T7018
5mg48,00€1mL*10mM (DMSO)50,00€10mg73,00€25mg133,00€50mg212,00€100mg314,00€200mg467,00€500mg748,00€DA-023
CAS:DA-023 (Compound 4) acts as a selective positive allosteric modulator (PAM) of EAAT2, exhibiting an EC 50 value of 1 nM [1].Fórmula:C20H25N7Forma y color:SolidPeso molecular:363.46GT 949
CAS:GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).Fórmula:C30H37N7O2Pureza:99.95%Forma y color:SolidPeso molecular:527.66V-9302
CAS:V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uMFórmula:C34H38N2O4Pureza:98% - 99.54%Forma y color:SolidPeso molecular:538.68Nisoxetine hydrochloride
CAS:Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitorFórmula:C17H21NO2·HClPureza:99.21%Forma y color:White SolidPeso molecular:307.82
