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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5400 productos de "Neurociencia"

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  • DL-Thyroxine

    CAS:
    <p>DL-Thyroxine is a thyroid hormone that acts as a monoamine oxidase (monoamine oxidase) inhibitor.</p>
    Fórmula:C15H11I4NO4
    Forma y color:Solid
    Peso molecular:776.87
  • Monoamine Oxidase B inhibitor 2


    <p>MAO-B inhibitor 2: potent, reversible, oral, selective (IC50=1.33 nM), BBB-penetrant, with anti-oxidant and anti-inflammatory effects for Parkinson's study.</p>
    Fórmula:C19H19FO3
    Forma y color:Solid
    Peso molecular:314.35
  • Befiradol hydrochloride

    CAS:
    <p>Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 aggregation.</p>
    Fórmula:C20H23Cl2F2N3O
    Pureza:99.1%
    Forma y color:Solid
    Peso molecular:430.32
  • eeAChE-IN-1


    <p>eeAChE-IN-1 is a strong inhibitor of eeAChE (IC50: 23 nM).</p>
    Fórmula:C27H30N6O5S
    Forma y color:Solid
    Peso molecular:550.63
  • AChE-IN-24


    <p>AChE-IN-24: Strong AChE blocker, crosses blood-brain barrier, IC50=0.053 μM, useful for AD research.</p>
    Fórmula:C22H30N2O4S2
    Forma y color:Solid
    Peso molecular:450.61
  • CVN636

    CAS:
    <p>CVN636, a potent and selective allosteric agonist for the mGluR7 receptor, exhibits oral activity and CNS permeability [1], with an EC50 of 7 nM for human</p>
    Fórmula:C19H20FNO4S
    Forma y color:Solid
    Peso molecular:377.43
  • Dihydro-β-erythroidine

    CAS:
    <p>Dihydro-β-erythroidine, a competitive nicotinic receptor antagonist, effectively blocks the discriminative stimulus properties and inhibits the anxiolytic</p>
    Fórmula:C16H21NO3
    Forma y color:Solid
    Peso molecular:275.34
  • LY2794193

    CAS:
    <p>LY2794193, a potent and selective mGlu3 receptor agonist, reduces akathisia seizures and increases GAT1, GLAST and GLT-1 protein levels in rats.</p>
    Fórmula:C16H18N2O6
    Pureza:98.15%
    Forma y color:Solid
    Peso molecular:334.32
  • Remlifanserin

    CAS:
    <p>Remlifanserin is a potent inverse agonist of the serotonin receptor (5-HT2A).</p>
    Fórmula:C24H29F2N3O2
    Forma y color:Solid
    Peso molecular:429.50
  • Sulamserod hydrochloride

    CAS:
    <p>Sulamserod hydrochloride is a 5-HT4 receptor antagonist. It is utilized in research related to gastrointestinal disorders.</p>
    Fórmula:C19H29Cl2N3O5S
    Forma y color:Solid
    Peso molecular:482.42
  • Cyproflanilide

    CAS:
    <p>Cyproflanilide is a GABAR antagonist that exhibits high activity against a variety of pests, including those from the Lepidoptera, Coleoptera, and Thysanoptera orders.</p>
    Fórmula:C28H17BrF12N2O2
    Forma y color:Solid
    Peso molecular:721.33
  • P2X7 receptor antagonist-5

    CAS:
    <p>P2X7 receptor antagonist-5 (compound 13a) is a potent, orally active, and long-lasting antagonist of the P2X7 receptor.</p>
    Fórmula:C21H17F3N6O3S2
    Forma y color:Solid
    Peso molecular:522.52
  • AAK1-IN-3 TFA


    <p>AAK1-IN-3 TFA, an AAK1 inhibitor with IC50 of 11 nM, crosses the blood-brain barrier, is a quinoline analogue, and may aid neuropathic pain research.</p>
    Fórmula:C24H22F6N4O4
    Forma y color:Solid
    Peso molecular:544.45
  • SB 243213 dihydrochloride

    CAS:
    <p>SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8 for</p>
    Fórmula:C22H21Cl2F3N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:501.33
  • DA-8031

    CAS:
    <p>DA-8031 is a selective and orally active serotonin reuptake inhibitor. It is utilized in research related to premature ejaculation (PE).</p>
    Fórmula:C21H24N2O2
    Forma y color:Solid
    Peso molecular:336.43
  • TDI-11861

    CAS:
    <p>TDI-11861 is a second-gen sAC (ADCY10) inhibitor with an IC50 of 5.5 nM and slow dissociation.</p>
    Fórmula:C22H25ClF2N6O3
    Forma y color:Solid
    Peso molecular:494.92
  • γ-secretase modulator 5


    <p>Compound 22d is a GSM that crosses the blood-brain barrier, inhibits Aβ42 production (IC50: 60 nM), and may help study Alzheimer's.</p>
    Forma y color:Solid
  • AChE-IN-5


    <p>AChE-IN-5: oral, crosses blood-brain barrier, targets AChE/5-HT1A/SERT, potent with 2.29 nM IC50.</p>
    Fórmula:C38H45N5O
    Forma y color:Solid
    Peso molecular:587.8
  • Nafimidone hydrochloride

    CAS:
    <p>Nafimidone hydrochloride, an antiepileptic agent, inhibits acetylcholinesterase, protects neurons, and ameliorates cognitive decline. It is utilized in epilepsy research.</p>
    Fórmula:C15H13ClN2O
    Forma y color:Solid
    Peso molecular:272.73
  • Rodatristat

    CAS:
    <p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>
    Fórmula:C27H27ClF3N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:561.98