
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(940 productos)
- ACK(1 productos)
- AChR(574 productos)
- ATP Citrato Liasa(16 productos)
- Receptor adrenérgico(2.942 productos)
- BACE(36 productos)
- Beta amiloide(204 productos)
- CAMK(68 productos)
- Inhibidores de ciclooxigenasa (COX)(562 productos)
- Receptor de dopamina(407 productos)
- Receptor GABA(336 productos)
- Gamma-secretasa(59 productos)
- GluR(255 productos)
- GlyT(24 productos)
- Receptor de histamina(358 productos)
- LRRK2(33 productos)
- Receptor de melatonina(24 productos)
- NMDAR(28 productos)
- Receptor de OX(40 productos)
- Receptor de opioides(296 productos)
Mostrar 12 subcategorías más
Se han encontrado 5400 productos de "Neurociencia"
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GSK2578215A
CAS:<p>GSK2578215A is a potent and selective LRRK2 kinase inhibitor.</p>Fórmula:C24H18FN3O2Pureza:99.57% - 99.94%Forma y color:SolidPeso molecular:399.42LPYFD-NH2 acetate
<p>LPYFD-NH2 acetate shows some inhibitory effect on the aggregation of Abeta(1-42).</p>Fórmula:C35H48N6O10Pureza:96.51%Forma y color:SolidPeso molecular:712.79Radiprodil
CAS:<p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>Fórmula:C21H20FN3O4Pureza:99.74%Forma y color:SolidPeso molecular:397.4Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Fórmula:C22H32ClN3O2Forma y color:SolidPeso molecular:405.96Isonipecotic acid
CAS:<p>Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.</p>Fórmula:C6H11NO2Pureza:99.82%Forma y color:White To Faint Pink-Beige PowderPeso molecular:129.16VU0119498
CAS:<p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>Fórmula:C15H10BrNO2Pureza:97.56%Forma y color:SolidPeso molecular:316.15Cariprazine hydrochloride
CAS:<p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>Fórmula:C21H33Cl3N4OPureza:99.78% - >99.99%Forma y color:SolidPeso molecular:463.87Glypromate acetate(32302-76-4 free base)
<p>Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.</p>Fórmula:C14H23N3O8Pureza:99.94%Forma y color:SolidPeso molecular:361.35A 438079 hydrochloride
CAS:<p>A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.</p>Fórmula:C13H10Cl3N5Pureza:99.74% - >99.99%Forma y color:SolidPeso molecular:342.61Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Forma y color:Pale Yellow SolidPeso molecular:469.553-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Forma y color:SolidPeso molecular:215.237-Amino-4-(trifluoromethyl)coumarin
CAS:<p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>Fórmula:C10H6F3NO2Pureza:97.31% - 97.84%Forma y color:Yellow PowderPeso molecular:229.16FR 122047
CAS:<p>FR 122047 (1-[(4,5-Bis(4-methoxyphenyl-2-thiazoyl)carbonyl]-4-methylpiperazine, Hydrochloride) is a potent and selective inhibitor of COX-1 with IC50 of 28 nM</p>Fórmula:C23H26ClN3O3SPureza:99.93%Forma y color:SolidPeso molecular:459.99Mivacurium dichloride
CAS:<p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>Fórmula:C58H80Cl2N2O14Pureza:99.2% - 99.48%Forma y color:Off-White SolidPeso molecular:1100.17Demecarium bromide
CAS:<p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>Fórmula:C32H52Br2N4O4Pureza:98%Forma y color:White Powder SolidPeso molecular:716.59Polmacoxib
CAS:<p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>Fórmula:C18H16FNO4SPureza:97.88%Forma y color:SolidPeso molecular:361.39Tiprenolol
CAS:<p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>Fórmula:C13H21NO2SPureza:99.43%Forma y color:SolidPeso molecular:255.38Methylbenactyzium Bromide
CAS:<p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>Fórmula:C21H28BrNO3Pureza:99.29%Forma y color:SolidPeso molecular:422.36SC-58125
CAS:<p>SC-58125 is a selective cyclooxygenase 2 (COX-2) inhibitor. SC-58125 exhibits antitumor activity, and also inhibits oedema at sites of inflammation.</p>Fórmula:C17H12F4N2O2SPureza:99.57%Forma y color:SolidPeso molecular:384.35Mosapride Citrate
CAS:<p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>Fórmula:C21H25ClFN3O3·C6H8O7Pureza:99.70%Forma y color:White PowderPeso molecular:614.02FPS-ZM1
CAS:<p>FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.</p>Fórmula:C20H22ClNOPureza:99.32% - 99.52%Forma y color:SolidPeso molecular:327.85Sepimostat
CAS:<p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>Fórmula:C21H19N5O2Pureza:97.75%Forma y color:SolidPeso molecular:373.41LY-404187
CAS:<p>LY404187 is a positive allosteric modulator of AMPA receptors</p>Fórmula:C19H22N2O2SPureza:99.34%Forma y color:SolidPeso molecular:342.46Tandospirone citrate
CAS:<p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>Fórmula:C27H37N5O9Pureza:97.84% - 99.90%Forma y color:SolidPeso molecular:575.61RU 24969 free base
CAS:<p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>Fórmula:C14H16N2OPureza:97.38%Forma y color:SolidPeso molecular:228.29Clozapine HCl
CAS:<p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>Fórmula:C18H20Cl2N4Forma y color:SolidPeso molecular:363.29CRANAD 2
CAS:<p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>Fórmula:C23H25BF2N2O2Pureza:99.44%Forma y color:Dark Blue To Black PowderPeso molecular:410.27Ansofaxine
CAS:<p>Ansofaxine, an SNRI compound, is commonly utilized in depression research as a serotonin-norepinephrine reuptake inhibitor.</p>Fórmula:C24H31NO3Forma y color:SolidPeso molecular:381.516Oxotremorine sesquifumarate
CAS:<p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>Fórmula:C12H18N2OC4H4O4Pureza:97.94%Forma y color:SolidPeso molecular:380.39Hemicholinium 3
CAS:<p>Hemicholinium 3 is a potent and selective choline uptake blocker.</p>Fórmula:C24H34Br2N2O4Pureza:98% - 99.95%Forma y color:SolidPeso molecular:574.35CZC-54252
CAS:<p>CZC-54252 is a potent inhibitor of LRRK2.</p>Fórmula:C22H25ClN6O4SPureza:99.39%Forma y color:SolidPeso molecular:504.99NMDAR antagonist 1
CAS:<p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>Fórmula:C20H20BrN3O2Pureza:98%Forma y color:SolidPeso molecular:414.3PF-06447475
CAS:<p>PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.</p>Fórmula:C17H15N5OPureza:98.61% - 99.62%Forma y color:SolidPeso molecular:305.33VU0238441
CAS:<p>VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.</p>Fórmula:C16H9ClF3NO2Pureza:100%Forma y color:SolidPeso molecular:339.7Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Fórmula:C22H23FN2O5Pureza:97.39% - 99.73%Forma y color:White SolidPeso molecular:414.43JI130
CAS:<p>JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.</p>Fórmula:C23H24N2O3Pureza:99.61%Forma y color:SolidPeso molecular:376.45Acotiamide monohydrochloride trihydrate
CAS:<p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>Fórmula:C21H37ClN4O8SPureza:98% - 99.54%Forma y color:SolidPeso molecular:541.06Nefazodone hydrochloride
CAS:<p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>Fórmula:C25H33Cl2N5O2Pureza:99% - 99.86%Forma y color:White SolidPeso molecular:506.47Piperazine citrate
CAS:<p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>Fórmula:C24H46N6O14Pureza:99.8%Forma y color:Crystals IndicationPeso molecular:642.65VU0364770
CAS:<p>VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu</p>Fórmula:C12H9ClN2OPureza:99.65% - >99.99%Forma y color:SolidPeso molecular:232.67(S)-3-Hydroxyphenylglycine
CAS:<p>(S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).</p>Fórmula:C8H9NO3Pureza:99.65%Forma y color:SolidPeso molecular:167.16Revefenacin
CAS:<p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>Fórmula:C35H43N5O4Pureza:98.12%Forma y color:SolidPeso molecular:597.75ADX-47273
CAS:<p>ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).</p>Fórmula:C20H17F2N3O2Pureza:97% - 99.18%Forma y color:SolidPeso molecular:369.36JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Forma y color:SolidPeso molecular:344.88SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Forma y color:SolidPeso molecular:371.9β-Amyloid (31-35)
CAS:<p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>Fórmula:C25H47N5O6SPureza:>99.99%Forma y color:SolidPeso molecular:545.74Donepezil
CAS:<p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>Fórmula:C24H29NO3Pureza:99.69%Forma y color:White Or Almost White Crystal PowderPeso molecular:379.49Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Fórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Intepirdine
CAS:<p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>Fórmula:C19H19N3O2SPureza:98% - 98.63%Forma y color:SolidPeso molecular:353.44Ocaperidone
CAS:<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Fórmula:C24H25FN4O2Pureza:99.33%Forma y color:SolidPeso molecular:420.48RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Fórmula:C17H16FN3Pureza:99.32%Forma y color:SolidPeso molecular:281.33Anle138b
CAS:<p>Anle138b: a novel oligomer modulator for disease-modifying therapy of neurodegenerative diseases such as prion and Parkinson's disease</p>Fórmula:C16H11BrN2O2Pureza:98.88% - 99.82%Forma y color:SolidPeso molecular:343.17α-Conotoxin MII acetate
<p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>Fórmula:C69H107N23O24S4Pureza:94.82% - 97.79%Forma y color:SolidPeso molecular:1770.99Pimavanserin tartrate
CAS:<p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>Fórmula:C50H68F2N6O4·C4H6O6Pureza:99.24% - 99.98%Forma y color:SolidPeso molecular:1005.2L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Fórmula:C18H22Cl4N4Pureza:97.52%Forma y color:SolidPeso molecular:436.21Prucalopride Succinate
CAS:<p>Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).</p>Fórmula:C18H26ClN3O3·C4H6O4Pureza:99.24%Forma y color:SolidPeso molecular:485.96GR 125743
CAS:<p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>Fórmula:C25H28N4O2Pureza:99.76%Forma y color:SolidPeso molecular:416.52SB 204741
CAS:<p>SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.</p>Fórmula:C14H14N4OSPureza:99.83%Forma y color:SolidPeso molecular:286.35N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Fórmula:C12H14N2OPureza:98.79%Forma y color:PowderPeso molecular:202.25PNU 22394 hydrochloride
CAS:<p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>Fórmula:C13H17ClN2Pureza:97.83%Forma y color:SolidPeso molecular:236.74NS-398
CAS:<p>NS-398 (N-(2-cyclohexyloxy-4-nitrophenyl)methane sulfonamide) is a COX-2 inhibitor wih anti-inflammatory activity.</p>Fórmula:C13H18N2O5SPureza:99% - >99.99%Forma y color:SolidPeso molecular:314.36Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Fórmula:C13H16N2O2Pureza:98% - 99.89%Forma y color:Pale Yellow Leaflets From Benzene SolidPeso molecular:232.28Gadoteridol
CAS:<p>Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.</p>Fórmula:C17H29GdN4O7Pureza:99.77% - 99.91%Forma y color:SolidPeso molecular:558.69DORA-22
CAS:<p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>Fórmula:C23H22F2N4O2Pureza:97.67%Forma y color:SolidPeso molecular:424.44Mavacoxib
CAS:<p>Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.</p>Fórmula:C16H11F4N3O2SPureza:99.90%Forma y color:SolidPeso molecular:385.34CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Fórmula:C19H15Cl2N3O2Pureza:>99.99%Forma y color:SolidPeso molecular:388.25Zacopride hydrochloride
CAS:<p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>Fórmula:C15H20ClN3O2·HClPureza:98.32%Forma y color:SolidPeso molecular:346.26MPEP hydrochloride
CAS:<p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>Fórmula:C14H12ClNPureza:99.87% - >99.99%Forma y color:SolidPeso molecular:229.7SB-200646
CAS:<p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>Fórmula:C15H14N4OPureza:99.61%Forma y color:SolidPeso molecular:266.3GW791343 dihydrochloride
CAS:<p>GW791343 dihydrochloride (GW791343 (HCl)) is a P2X7 allosteric modulator.</p>Fórmula:C20H26Cl2F2N4OPureza:>99.99%Forma y color:SolidPeso molecular:447.35Naluzotan
CAS:<p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>Fórmula:C23H38N4O3SPureza:>99.99%Forma y color:SolidPeso molecular:450.64A-867744
CAS:<p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>Fórmula:C20H19ClN2O3SPureza:95.66%Forma y color:SolidPeso molecular:402.89AZD-8529
CAS:<p>AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.</p>Fórmula:C24H24F3N5O3Forma y color:SolidPeso molecular:487.47SB 242084
CAS:<p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>Fórmula:C21H19ClN4O2Pureza:99.75% - ≥98%Forma y color:SolidPeso molecular:394.85GALANTHAMINONE
CAS:<p>Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairments</p>Fórmula:C17H19NO3Pureza:99.93%Forma y color:White To Off-White ChemicalPeso molecular:285.34TCS-OX2-29
CAS:<p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.</p>Fórmula:C23H31N3O3Pureza:99.81%Forma y color:SolidPeso molecular:397.51A-804598
CAS:<p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>Fórmula:C19H17N5Pureza:99.57%Forma y color:SolidPeso molecular:315.37PHA 568487 free base
CAS:<p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>Fórmula:C16H20N2O3Pureza:99.74%Forma y color:SolidPeso molecular:288.34Opiranserin hydrochloride
CAS:<p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>Fórmula:C21H35ClN2O5Pureza:99.33%Forma y color:SolidPeso molecular:430.97AVN-492
CAS:<p>AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).</p>Fórmula:C17H21N5O2SPureza:99.81%Forma y color:SolidPeso molecular:359.45CFMTI
CAS:<p>CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.</p>Fórmula:C19H16FN5OPureza:97.23%Forma y color:SolidPeso molecular:349.36Tariquidar
CAS:<p>Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.</p>Fórmula:C38H38N4O6Pureza:98.07% - 99.45%Forma y color:SolidPeso molecular:646.73CaMKP Inhibitor
CAS:<p>CaMKP Inhibitor can inhibit CaMKP.</p>Fórmula:C10H8NNaO7S2Pureza:96.55% - 99.98%Forma y color:SolidPeso molecular:341.28γ-Mangostin
CAS:<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Fórmula:C23H24O6Pureza:98.55% - 99.08%Forma y color:SolidPeso molecular:396.434-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Fórmula:C6H11NO3Pureza:98.51%Forma y color:SolidPeso molecular:145.16VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Fórmula:C13H15ClN4Pureza:99.66%Forma y color:SolidPeso molecular:262.74NS9283
CAS:<p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>Fórmula:C14H8N4OPureza:99.12%Forma y color:SolidPeso molecular:248.24SR 57227 hydrochloride
CAS:<p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>Fórmula:C10H14ClN3·HClPureza:99.89%Forma y color:SolidPeso molecular:248.15Amyloid β-Protein 10-20 acetate
<p>Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research of</p>Fórmula:C73H103N17O18Pureza:97.23%Forma y color:SolidPeso molecular:1506.65Lu AF21934
CAS:<p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>Fórmula:C14H16Cl2N2O2Pureza:99.79%Forma y color:SolidPeso molecular:315.2FK 3311
CAS:<p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>Fórmula:C15H13F2NO4SPureza:97.98%Forma y color:SolidPeso molecular:341.33Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Fórmula:C35H47FN10O8Pureza:97.97%Forma y color:SolidPeso molecular:754.85pyridostigmine
CAS:<p>Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.</p>Fórmula:C9H13N2O2Pureza:98.10%Forma y color:SolidPeso molecular:181.21Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:207.23lumateperone Tosylate
CAS:<p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>Fórmula:C31H36FN3O4SPureza:95.83% - 99.95%Forma y color:SolidPeso molecular:565.7Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Fórmula:C16H16Cl3NPureza:98.92% - 99.6%Forma y color:SolidPeso molecular:328.66Sarpogrelate
CAS:<p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>Fórmula:C24H31NO6Forma y color:SolidPeso molecular:429.51Pergolide mesylate
CAS:<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Fórmula:C20H30N2O3S2Pureza:99.70%Forma y color:White To Off-White SolidPeso molecular:410.59GNE-7915 tosylate
CAS:<p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>Fórmula:C26H29F4N5O6SForma y color:SolidPeso molecular:615.6CX516
CAS:<p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>Fórmula:C14H15N3OPureza:99.04% - ≥95%Forma y color:Tan SolidPeso molecular:241.29Xanthotoxol
CAS:<p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>Fórmula:C11H6O4Pureza:99.97%Forma y color:SolidPeso molecular:202.16Gabazine free base
CAS:<p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>Fórmula:C15H17N3O3Forma y color:SolidPeso molecular:287.314F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Fórmula:C22H26FNO·C2H2O4Pureza:97.34%Forma y color:SolidPeso molecular:429.49(S)-Amisulpride
CAS:<p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>Fórmula:C17H27N3O4SPureza:98.38%Forma y color:SolidPeso molecular:369.48PHA 543613 hydrochloride
CAS:<p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>Fórmula:C15H18ClN3O2Forma y color:SolidPeso molecular:307.78TCN238
CAS:<p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>Fórmula:C12H11N3Pureza:99.9% - 99.92%Forma y color:SolidPeso molecular:197.24KN-92 hydrochloride
CAS:<p>KN-92 hydrochloride is an inactive derivative of KN-93.</p>Fórmula:C24H26Cl2N2O3SPureza:99.68%Forma y color:SolidPeso molecular:493.45Chelidamic acid
CAS:<p>Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.</p>Fórmula:C7H5NO5Pureza:98.11%Forma y color:Pale Yellow PowderPeso molecular:183.12GNE0877
CAS:<p>GNE0877 (GNE 0877) is a highly effective and specific leucine-rich repeat kinase 2 (LRRK2) inhibitor (Ki: 0.7 nM).</p>Fórmula:C14H16F3N7Pureza:98.01% - 99.97%Forma y color:SolidPeso molecular:339.32Alprenolol hydrochloride
CAS:<p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>Fórmula:C15H24ClNO2Pureza:99.79%Forma y color:SolidPeso molecular:285.81Quipazine
CAS:<p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>Fórmula:C13H15N3Forma y color:SolidPeso molecular:213.28pep2-SVKI acetate
<p>Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.</p>Fórmula:C62H97N13O20Pureza:97.14%Forma y color:SolidPeso molecular:1344.51Tinoridine hydrochloride
CAS:<p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>Fórmula:C17H21ClN2O2SPureza:97.49%Forma y color:SolidPeso molecular:352.88Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Forma y color:SolidPeso molecular:86.14m-Chlorophenylbiguanide hydrochloride
CAS:<p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>Fórmula:C8H11Cl2N5Pureza:99.43% - 99.87%Forma y color:SolidPeso molecular:248.11lavendustin C
CAS:<p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>Fórmula:C14H13NO5Pureza:98.06%Forma y color:Yellow To Tan PowderPeso molecular:275.26CALP2 acetate(261969-04-4 free base)
<p>CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.</p>Fórmula:C68H104N14O13SPureza:97.43%Forma y color:SolidPeso molecular:1357.7TG6-10-1
CAS:<p>TG6-10-1 is an EP2 antagonist.</p>Fórmula:C23H23F3N2O4Pureza:99.66% - ≥95%Forma y color:SolidPeso molecular:448.43AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Forma y color:SolidPeso molecular:354.38Baclofen hydrochloride
CAS:<p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>Fórmula:C10H13Cl2NO2Pureza:99.55%Forma y color:SolidPeso molecular:250.1221-(1-Naphthyl) piperazine hydrochloride
CAS:<p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>Fórmula:C14H17ClN2Pureza:98.27%Forma y color:SolidPeso molecular:248.75PU02
CAS:<p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>Fórmula:C16H12N4SPureza:99.35%Forma y color:SolidPeso molecular:292.36MK 212 hydrochloride
CAS:<p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>Fórmula:C8H11ClN4·HClPureza:99.88%Forma y color:SolidPeso molecular:235.12SB 242084 dihydrochloride
CAS:<p>SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.</p>Fórmula:C21H21Cl3N4O2Forma y color:SolidPeso molecular:467.78Acamprosate
CAS:<p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>Fórmula:C5H11NO4SPureza:98.30%Forma y color:SolidPeso molecular:181.21Naratriptan hydrochloride
CAS:<p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>Fórmula:C17H25N3O2S·HClPureza:99.17% - 99.93%Forma y color:Beige SolidPeso molecular:371.93PBD-150
CAS:<p>PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)</p>Fórmula:C15H20N4O2SPureza:99.68%Forma y color:SolidPeso molecular:320.41Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Fórmula:C22H25ClN4O4S2Forma y color:SolidPeso molecular:509.04γ-secretase modulator 1 hydrochloride
CAS:<p>gamma-secretase inhibitior-1 is a gamma-secretase modulator that is useful to Alzheimer's disease [1].</p>Fórmula:C24H25ClN4OSPureza:98%Forma y color:SolidPeso molecular:453Lerisetron
CAS:<p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>Fórmula:C18H20N4Pureza:99.15% - 99.82%Forma y color:SolidPeso molecular:292.38pep2-EVKI acetate(1315378-67-6 free base)
<p>Pep2-EVKI acetate, a cell-permeable peptide, disrupts PICK1-GluR2 AMPA receptor binding.</p>Fórmula:C64H99N13O21Pureza:97.63%Forma y color:SolidPeso molecular:1386.55Basmisanil
CAS:<p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>Fórmula:C21H20FN3O5SPureza:99.21% - 99.42%Forma y color:SolidPeso molecular:445.46PF-06454589
CAS:<p>PF-06454589 is a potent inhibitor of LRRK2.</p>Fórmula:C14H16N6OPureza:99.06%Forma y color:SolidPeso molecular:284.32AZ 11645373
CAS:<p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>Fórmula:C24H21N3O5SPureza:99.47%Forma y color:SolidPeso molecular:463.51Imidafenacin
CAS:<p>Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.</p>Fórmula:C20H21N3OPureza:99.17%Forma y color:SolidPeso molecular:319.4Dihydroergotoxine mesylate
CAS:<p>Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.</p>Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Forma y color:SolidPeso molecular:423.53Aminooxyacetic acid hemihydrochloride
CAS:<p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>Fórmula:C2H5NO3·5HClPureza:98.03%Forma y color:Light Beige Crystalline PowderPeso molecular:109.3Indophagolin
CAS:<p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>Fórmula:C19H15BrClF3N2O3SPureza:99.76%Forma y color:SolidPeso molecular:523.75A-740003
CAS:<p>A-740003 is a potent P2X7 receptor blocker, inhibiting rat/human receptors (IC50: 18/40 nM), lessens pain in animals, and shrinks mouse neuroblastoma.</p>Fórmula:C26H30N6O3Pureza:96.53% - 99.68%Forma y color:SolidPeso molecular:474.55Prifinium bromide
CAS:<p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>Fórmula:C22H28BrNPureza:97.99%Forma y color:SolidPeso molecular:386.37Vortioxetine
CAS:<p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>Fórmula:C18H22N2SPureza:99.34% - 99.34%Forma y color:SolidPeso molecular:298.45S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Fórmula:C31H34N2O4Pureza:99.77%Forma y color:SolidPeso molecular:498.61Metadoxine
CAS:<p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>Fórmula:C8H11NO3·C5H7NO3Pureza:99.19%Forma y color:Off-White PowderPeso molecular:298.29Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Fórmula:C12H17ClN2O2Pureza:99.35%Forma y color:SolidPeso molecular:256.73DNQX
CAS:<p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C8H4N4O6Pureza:97.27% - 99.1%Forma y color:Off-White Powder With A Yellow TingePeso molecular:252.14VU-1545
CAS:<p>VU-1545 is mGlu5 positive allosteric modulator.</p>Fórmula:C22H15FN4O3Pureza:98.8%Forma y color:SolidPeso molecular:402.38Pitofenone hydrochloride
CAS:<p>Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and</p>Fórmula:C22H26ClNO4Pureza:99.97%Forma y color:SolidPeso molecular:403.9Syk Inhibitor II dihydrochloride dihydrate
CAS:<p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>Fórmula:C14H21Cl2F3N6O3Forma y color:SolidPeso molecular:449.26TAE-1
CAS:<p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>Fórmula:C39H51I3N6O9Pureza:94.58%Forma y color:SolidPeso molecular:1128.571,1'-Methylenedi-2-naphthol
CAS:<p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>Fórmula:C21H16O2Pureza:98.91%Forma y color:Light Pink To Light Brown Crystalline PowderPeso molecular:300.35Saclofen
CAS:<p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>Fórmula:C9H12ClNO3SPureza:99.17%Forma y color:White Crystalline SolidPeso molecular:249.71Acotiamide
CAS:<p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>Fórmula:C21H30N4O5SForma y color:SolidPeso molecular:450.55Metoclopramide hydrochloride hydrate
CAS:<p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>Fórmula:C14H25Cl2N3O3Pureza:99.33%Forma y color:SolidPeso molecular:354.27PE859
CAS:<p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>Fórmula:C28H24N4O2Pureza:98.8% - 99.09%Forma y color:SolidPeso molecular:448.52Loreclezole
CAS:<p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>Fórmula:C10H6Cl3N3Pureza:99.78%Forma y color:SolidPeso molecular:274.53NH125
CAS:<p>NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, >125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.</p>Fórmula:C27H45IN2Pureza:98.60%Forma y color:SolidPeso molecular:524.56Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Fórmula:C23H28ClFN4O2Forma y color:SolidPeso molecular:446.95Aftin-4
CAS:<p>Aftin-4, an amyloid forty-two inducer, activates γ-secretase, promoting the generation of amyloid-β-1-42 (Aβ1-42) from amyloid-β protein precursor.</p>Fórmula:C20H28N6OPureza:98.51%Forma y color:SolidPeso molecular:368.486-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Fórmula:C6H6N2O2Pureza:99.94%Forma y color:SoildPeso molecular:138.1238GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Forma y color:SolidPeso molecular:415.53Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Fórmula:C20H24N2OSForma y color:SolidPeso molecular:340.48RU 24969 succinate
CAS:<p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>Fórmula:C18H22N2O5Forma y color:SolidPeso molecular:346.38Azeliragon HCl
CAS:<p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>Fórmula:C32H40Cl3N3O2Forma y color:SolidPeso molecular:605.04Ondansetron hydrochloride
CAS:<p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>Fórmula:C18H19N3O·HClPureza:99.78%Forma y color:White PowderPeso molecular:329.82Succinylcholine Chloride Dihydrate
CAS:<p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>Fórmula:C14H30N2O4·2Cl·2H2OPureza:99.87%Forma y color:White SolidPeso molecular:397.34Piperidolate hydrochloride
CAS:<p>Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.</p>Fórmula:C21H26ClNO2Pureza:99.5%Forma y color:SolidPeso molecular:359.89ZL006
CAS:<p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>Fórmula:C14H11Cl2NO4Pureza:98.29%Forma y color:SolidPeso molecular:328.15PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Forma y color:SolidPeso molecular:301.21Alosetron (Hydrochloride(1:X))
CAS:<p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>Fórmula:C17H18ClN4OForma y color:SolidPeso molecular:329.11691trans-ACPD
CAS:<p>trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.</p>Fórmula:C7H11NO4Pureza:99.53%Forma y color:SolidPeso molecular:173.17Melitracen hydrochloride
CAS:<p>Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.</p>Fórmula:C21H26ClNPureza:99.99%Forma y color:Crystalline SolidPeso molecular:327.90MTEP hydrochloride
CAS:<p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>Fórmula:C11H9ClN2SPureza:99.58%Forma y color:SolidPeso molecular:236.72Acotiamide hydrochloride
CAS:<p>Acotiamide hydrochloride, an oral AChE inhibitor (IC50: 1.79 μM), boosts gastric movement and treats functional dyspepsia.</p>Fórmula:C21H31ClN4O5SForma y color:SolidPeso molecular:487.01Quipazine maleate
CAS:<p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>Fórmula:C17H19N3O4Forma y color:SolidPeso molecular:329.36Caroverine hydrochloride
CAS:<p>Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.</p>Fórmula:C22H28ClN3O2Pureza:98.37% - 98.75%Forma y color:SolidPeso molecular:401.9Eslicarbazepine Acetate
CAS:<p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>Fórmula:C17H16N2O3Pureza:99.58% - >99.99%Forma y color:White To Off-White SolidPeso molecular:296.32CaM kinase II inhibitor TFA salt
<p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>Fórmula:C66H117F3N22O21Pureza:>99.99%Forma y color:SolidPeso molecular:1611.77S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Fórmula:C24H26FN3O2Forma y color:SolidPeso molecular:407.48Nor-benzetimide
CAS:<p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>Fórmula:C16H20N2O2Pureza:98.63%Forma y color:SolidPeso molecular:272.34Eltoprazine dihydrochloride
CAS:<p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>Fórmula:C12H18Cl2N2O2Pureza:99.64%Forma y color:SolidPeso molecular:293.19Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Forma y color:SolidPeso molecular:477.57Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Fórmula:C19H25NOSPureza:98.08% - 99.59%Forma y color:SolidPeso molecular:315.47CaMKII-IN-1
CAS:<p>CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM).</p>Fórmula:C29H30ClN5O2SPureza:99.69%Forma y color:SolidPeso molecular:548.1BRL-15572 dihydrochloride
CAS:<p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>Fórmula:C25H27ClN2O·2HClPureza:99.74%Forma y color:SolidPeso molecular:479.87Arecaidine hydrochloride
CAS:<p>Arecaidine hydrochloride may have carcinogenesis.</p>Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Forma y color:SolidPeso molecular:177.63Mofezolac
CAS:<p>Mofezolac (formerly known as Disopain or N-22) is a highly selective COX-1 (cyclooxygenase-1) inhibitor with COXs selectivity index > 6000</p>Fórmula:C19H17NO5Pureza:99.29%Forma y color:SolidPeso molecular:339.34Duloxetine
CAS:<p>Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.</p>Fórmula:C18H19NOSPureza:99.71% - 99.89%Forma y color:SolidPeso molecular:297.41SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Fórmula:C20H25N3O2Pureza:99.02%Forma y color:SolidPeso molecular:339.43Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Fórmula:C21H30N4O4Pureza:99.52%Forma y color:SolidPeso molecular:402.49PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Fórmula:C21H29Cl2N3O4SPureza:98.5%Forma y color:SolidPeso molecular:490.44Syn-Ake acetate
CAS:<p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>Fórmula:C19H29N5O3·2(C2H4O2)Pureza:99.60%Forma y color:SolidPeso molecular:495.58Trihexyphenidyl hydrochloride
CAS:<p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>Fórmula:C20H32ClNOPureza:99.65%Forma y color:SolidPeso molecular:337.927CNQX
CAS:<p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C9H4N4O4Pureza:99.70%Forma y color:Pale Yellow SolidPeso molecular:232.15(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Fórmula:C13H15NO2Pureza:99.58% - 99.87%Forma y color:SolidPeso molecular:217.26Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Forma y color:Almost White To White Crystalline PowderPeso molecular:351.93Harmine hydrochloride
CAS:<p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>Fórmula:C13H13ClN2OPureza:99.61% - >99.99%Forma y color:Yellow To Slightly Green Crystalline PowderPeso molecular:248.71Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Fórmula:C16H14FN3OPureza:99.72%Forma y color:SolidPeso molecular:283.3Darifenacin
CAS:<p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>Fórmula:C28H30N2O2Pureza:99.78%Forma y color:SolidPeso molecular:426.55Ethyl (triphenylphosphoranylidene) acetate
CAS:<p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>Fórmula:C22H21O2PPureza:97.985%Forma y color:White Or Slight Yellow PowderPeso molecular:348.37Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Fórmula:C24H32ClNO6Pureza:99.73%Forma y color:Colorless LiquidPeso molecular:465.97
