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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5400 productos de "Neurociencia"

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  • GSK2578215A

    CAS:
    <p>GSK2578215A is a potent and selective LRRK2 kinase inhibitor.</p>
    Fórmula:C24H18FN3O2
    Pureza:99.57% - 99.94%
    Forma y color:Solid
    Peso molecular:399.42
  • LPYFD-NH2 acetate


    <p>LPYFD-NH2 acetate shows some inhibitory effect on the aggregation of Abeta(1-42).</p>
    Fórmula:C35H48N6O10
    Pureza:96.51%
    Forma y color:Solid
    Peso molecular:712.79
  • Radiprodil

    CAS:
    <p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>
    Fórmula:C21H20FN3O4
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:397.4
  • Piboserod hydrochloride

    CAS:
    <p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>
    Fórmula:C22H32ClN3O2
    Forma y color:Solid
    Peso molecular:405.96
  • Isonipecotic acid

    CAS:
    <p>Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.</p>
    Fórmula:C6H11NO2
    Pureza:99.82%
    Forma y color:White To Faint Pink-Beige Powder
    Peso molecular:129.16
  • VU0119498

    CAS:
    <p>VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.</p>
    Fórmula:C15H10BrNO2
    Pureza:97.56%
    Forma y color:Solid
    Peso molecular:316.15
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Forma y color:Solid
    Peso molecular:463.87
  • Glypromate acetate(32302-76-4 free base)


    <p>Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.</p>
    Fórmula:C14H23N3O8
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:361.35
  • A 438079 hydrochloride

    CAS:
    <p>A 438079 hydrochloride (A-438079 HCl) is a potent and selective P2X7 receptor antagonist with pIC50 of 6.9.</p>
    Fórmula:C13H10Cl3N5
    Pureza:99.74% - >99.99%
    Forma y color:Solid
    Peso molecular:342.61
  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Forma y color:Pale Yellow Solid
    Peso molecular:469.55
  • 3-MATIDA

    CAS:
    <p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Forma y color:Solid
    Peso molecular:215.23
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    <p>7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.</p>
    Fórmula:C10H6F3NO2
    Pureza:97.31% - 97.84%
    Forma y color:Yellow Powder
    Peso molecular:229.16
  • FR 122047

    CAS:
    <p>FR 122047 (1-[(4,5-Bis(4-methoxyphenyl-2-thiazoyl)carbonyl]-4-methylpiperazine, Hydrochloride) is a potent and selective inhibitor of COX-1 with IC50 of 28 nM</p>
    Fórmula:C23H26ClN3O3S
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:459.99
  • Mivacurium dichloride

    CAS:
    <p>Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.</p>
    Fórmula:C58H80Cl2N2O14
    Pureza:99.2% - 99.48%
    Forma y color:Off-White Solid
    Peso molecular:1100.17
  • Demecarium bromide

    CAS:
    <p>Demecarium bromide (BC-48) is a potent cholinesterase inhibitor,and is treatment glaucoma agent.</p>
    Fórmula:C32H52Br2N4O4
    Pureza:98%
    Forma y color:White Powder Solid
    Peso molecular:716.59
  • Polmacoxib

    CAS:
    <p>Polmacoxib, a first-class NSAID, dual inhibitor of CA and COX-2, may hinder colorectal cancer growth in mice.</p>
    Fórmula:C18H16FNO4S
    Pureza:97.88%
    Forma y color:Solid
    Peso molecular:361.39
  • Tiprenolol

    CAS:
    <p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>
    Fórmula:C13H21NO2S
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:255.38
  • Methylbenactyzium Bromide

    CAS:
    <p>Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.</p>
    Fórmula:C21H28BrNO3
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:422.36
  • SC-58125

    CAS:
    <p>SC-58125 is a selective cyclooxygenase 2 (COX-2) inhibitor. SC-58125 exhibits antitumor activity, and also inhibits oedema at sites of inflammation.</p>
    Fórmula:C17H12F4N2O2S
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:384.35
  • Mosapride Citrate

    CAS:
    <p>Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.</p>
    Fórmula:C21H25ClFN3O3·C6H8O7
    Pureza:99.70%
    Forma y color:White Powder
    Peso molecular:614.02
  • FPS-ZM1

    CAS:
    <p>FPS-ZM1 is a high-affinity RAGE specific inhibitor that blocks Aβ binding to the V domain of RAGE.</p>
    Fórmula:C20H22ClNO
    Pureza:99.32% - 99.52%
    Forma y color:Solid
    Peso molecular:327.85
  • Sepimostat

    CAS:
    <p>Sepimostat is a neuroprotective NR2B NMDA receptor antagonist with a Ki of 27.7 μM at Ifenprodil-binding site.</p>
    Fórmula:C21H19N5O2
    Pureza:97.75%
    Forma y color:Solid
    Peso molecular:373.41
  • LY-404187

    CAS:
    <p>LY404187 is a positive allosteric modulator of AMPA receptors</p>
    Fórmula:C19H22N2O2S
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:342.46
  • Tandospirone citrate

    CAS:
    <p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>
    Fórmula:C27H37N5O9
    Pureza:97.84% - 99.90%
    Forma y color:Solid
    Peso molecular:575.61
  • RU 24969 free base

    CAS:
    <p>RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.</p>
    Fórmula:C14H16N2O
    Pureza:97.38%
    Forma y color:Solid
    Peso molecular:228.29
  • Clozapine HCl

    CAS:
    <p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>
    Fórmula:C18H20Cl2N4
    Forma y color:Solid
    Peso molecular:363.29
  • CRANAD 2

    CAS:
    <p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>
    Fórmula:C23H25BF2N2O2
    Pureza:99.44%
    Forma y color:Dark Blue To Black Powder
    Peso molecular:410.27
  • Ansofaxine

    CAS:
    <p>Ansofaxine, an SNRI compound, is commonly utilized in depression research as a serotonin-norepinephrine reuptake inhibitor.</p>
    Fórmula:C24H31NO3
    Forma y color:Solid
    Peso molecular:381.516
  • Oxotremorine sesquifumarate

    CAS:
    <p>Oxotremorine sesquifumarate is a muscarinic agonist.</p>
    Fórmula:C12H18N2OC4H4O4
    Pureza:97.94%
    Forma y color:Solid
    Peso molecular:380.39
  • Hemicholinium 3

    CAS:
    <p>Hemicholinium 3 is a potent and selective choline uptake blocker.</p>
    Fórmula:C24H34Br2N2O4
    Pureza:98% - 99.95%
    Forma y color:Solid
    Peso molecular:574.35
  • CZC-54252

    CAS:
    <p>CZC-54252 is a potent inhibitor of LRRK2.</p>
    Fórmula:C22H25ClN6O4S
    Pureza:99.39%
    Forma y color:Solid
    Peso molecular:504.99
  • NMDAR antagonist 1

    CAS:
    <p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>
    Fórmula:C20H20BrN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:414.3
  • PF-06447475

    CAS:
    <p>PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.</p>
    Fórmula:C17H15N5O
    Pureza:98.61% - 99.62%
    Forma y color:Solid
    Peso molecular:305.33
  • VU0238441

    CAS:
    <p>VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.</p>
    Fórmula:C16H9ClF3NO2
    Pureza:100%
    Forma y color:Solid
    Peso molecular:339.7
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Fórmula:C22H23FN2O5
    Pureza:97.39% - 99.73%
    Forma y color:White Solid
    Peso molecular:414.43
  • JI130

    CAS:
    <p>JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.</p>
    Fórmula:C23H24N2O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:376.45
  • Acotiamide monohydrochloride trihydrate

    CAS:
    <p>Acotiamide monohydrochloride trihydrate (Z-338 HCl) is the hydrochloride salt form of acotiamide, a prokinetic agent with GI motility-enhancing activity.</p>
    Fórmula:C21H37ClN4O8S
    Pureza:98% - 99.54%
    Forma y color:Solid
    Peso molecular:541.06
  • Nefazodone hydrochloride

    CAS:
    <p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>
    Fórmula:C25H33Cl2N5O2
    Pureza:99% - 99.86%
    Forma y color:White Solid
    Peso molecular:506.47
  • Piperazine citrate

    CAS:
    <p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>
    Fórmula:C24H46N6O14
    Pureza:99.8%
    Forma y color:Crystals Indication
    Peso molecular:642.65
  • VU0364770

    CAS:
    <p>VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu</p>
    Fórmula:C12H9ClN2O
    Pureza:99.65% - >99.99%
    Forma y color:Solid
    Peso molecular:232.67
  • (S)-3-Hydroxyphenylglycine

    CAS:
    <p>(S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).</p>
    Fórmula:C8H9NO3
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:167.16
  • Revefenacin

    CAS:
    <p>Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.</p>
    Fórmula:C35H43N5O4
    Pureza:98.12%
    Forma y color:Solid
    Peso molecular:597.75
  • ADX-47273

    CAS:
    <p>ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).</p>
    Fórmula:C20H17F2N3O2
    Pureza:97% - 99.18%
    Forma y color:Solid
    Peso molecular:369.36
  • JNJ-40411813

    CAS:
    <p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:344.88
  • SKF89976A hydrochloride

    CAS:
    <p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>
    Fórmula:C22H26ClNO2
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:371.9
  • β-Amyloid (31-35)

    CAS:
    <p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>
    Fórmula:C25H47N5O6S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:545.74
  • Donepezil

    CAS:
    <p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>
    Fórmula:C24H29NO3
    Pureza:99.69%
    Forma y color:White Or Almost White Crystal Powder
    Peso molecular:379.49
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Forma y color:Solid
    Peso molecular:427.41
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Fórmula:C19H19N3O2S
    Pureza:98% - 98.63%
    Forma y color:Solid
    Peso molecular:353.44
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:420.48
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Fórmula:C17H16FN3
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:281.33
  • Anle138b

    CAS:
    <p>Anle138b: a novel oligomer modulator for disease-modifying therapy of neurodegenerative diseases such as prion and Parkinson's disease</p>
    Fórmula:C16H11BrN2O2
    Pureza:98.88% - 99.82%
    Forma y color:Solid
    Peso molecular:343.17
  • α-Conotoxin MII acetate


    <p>α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.</p>
    Fórmula:C69H107N23O24S4
    Pureza:94.82% - 97.79%
    Forma y color:Solid
    Peso molecular:1770.99
  • Pimavanserin tartrate

    CAS:
    <p>Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.</p>
    Fórmula:C50H68F2N6O4·C4H6O6
    Pureza:99.24% - 99.98%
    Forma y color:Solid
    Peso molecular:1005.2
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:436.21
  • Prucalopride Succinate

    CAS:
    <p>Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).</p>
    Fórmula:C18H26ClN3O3·C4H6O4
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:485.96
  • GR 125743

    CAS:
    <p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>
    Fórmula:C25H28N4O2
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:416.52
  • SB 204741

    CAS:
    <p>SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.</p>
    Fórmula:C14H14N4OS
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:286.35
  • N-ACETYLTRYPTAMINE

    CAS:
    <p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>
    Fórmula:C12H14N2O
    Pureza:98.79%
    Forma y color:Powder
    Peso molecular:202.25
  • PNU 22394 hydrochloride

    CAS:
    <p>PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist</p>
    Fórmula:C13H17ClN2
    Pureza:97.83%
    Forma y color:Solid
    Peso molecular:236.74
  • NS-398

    CAS:
    <p>NS-398 (N-(2-cyclohexyloxy-4-nitrophenyl)methane sulfonamide) is a COX-2 inhibitor wih anti-inflammatory activity.</p>
    Fórmula:C13H18N2O5S
    Pureza:99% - >99.99%
    Forma y color:Solid
    Peso molecular:314.36
  • Melatonin

    CAS:
    <p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>
    Fórmula:C13H16N2O2
    Pureza:98% - 99.89%
    Forma y color:Pale Yellow Leaflets From Benzene Solid
    Peso molecular:232.28
  • Gadoteridol

    CAS:
    <p>Gadoteridol (Gd-HP-DO3A) is a gadolinium-based MRI contrast agent that can be used for central nervous system imaging.</p>
    Fórmula:C17H29GdN4O7
    Pureza:99.77% - 99.91%
    Forma y color:Solid
    Peso molecular:558.69
  • DORA-22

    CAS:
    <p>DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on memory</p>
    Fórmula:C23H22F2N4O2
    Pureza:97.67%
    Forma y color:Solid
    Peso molecular:424.44
  • Mavacoxib

    CAS:
    <p>Mavacoxib is a selective inhibitor of cyclooxygenase-2 (COX-2) ,with Anti-Tumour activity.</p>
    Fórmula:C16H11F4N3O2S
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:385.34
  • CCMI

    CAS:
    <p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>
    Fórmula:C19H15Cl2N3O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:388.25
  • Zacopride hydrochloride

    CAS:
    <p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>
    Fórmula:C15H20ClN3O2·HCl
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:346.26
  • MPEP hydrochloride

    CAS:
    <p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>
    Fórmula:C14H12ClN
    Pureza:99.87% - >99.99%
    Forma y color:Solid
    Peso molecular:229.7
  • SB-200646

    CAS:
    <p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>
    Fórmula:C15H14N4O
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:266.3
  • GW791343 dihydrochloride

    CAS:
    <p>GW791343 dihydrochloride (GW791343 (HCl)) is a P2X7 allosteric modulator.</p>
    Fórmula:C20H26Cl2F2N4O
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:447.35
  • Naluzotan

    CAS:
    <p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:450.64
  • A-867744

    CAS:
    <p>A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR (EC50: 1.0 μM).</p>
    Fórmula:C20H19ClN2O3S
    Pureza:95.66%
    Forma y color:Solid
    Peso molecular:402.89
  • AZD-8529

    CAS:
    <p>AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.</p>
    Fórmula:C24H24F3N5O3
    Forma y color:Solid
    Peso molecular:487.47
  • SB 242084

    CAS:
    <p>SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.</p>
    Fórmula:C21H19ClN4O2
    Pureza:99.75% - ≥98%
    Forma y color:Solid
    Peso molecular:394.85
  • GALANTHAMINONE

    CAS:
    <p>Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairments</p>
    Fórmula:C17H19NO3
    Pureza:99.93%
    Forma y color:White To Off-White Chemical
    Peso molecular:285.34
  • TCS-OX2-29

    CAS:
    <p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays &gt;250-fold selectivity for OX2 over OX1.</p>
    Fórmula:C23H31N3O3
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:397.51
  • A-804598

    CAS:
    <p>A-804598 is a competitive and selective P2X7 receptor antagonist (IC50: 10 nM, rat; 9 nM, mouse; 11 nM, human).</p>
    Fórmula:C19H17N5
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:315.37
  • PHA 568487 free base

    CAS:
    <p>PHA 568487 free base, an α7 nicotinic receptor agonist, designed to reduce bioactivation and improve in vivo tolerability.</p>
    Fórmula:C16H20N2O3
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:288.34
  • Opiranserin hydrochloride

    CAS:
    <p>Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM</p>
    Fórmula:C21H35ClN2O5
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:430.97
  • AVN-492

    CAS:
    <p>AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).</p>
    Fórmula:C17H21N5O2S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:359.45
  • CFMTI

    CAS:
    <p>CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.</p>
    Fórmula:C19H16FN5O
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:349.36
  • Tariquidar

    CAS:
    <p>Tariquidar (XR9576)(Kd=5.1 nM) is a specific and effective non-competitive inhibitor of P-glycoprotein. It can reverse drug resistance in MDR cell Lines.</p>
    Fórmula:C38H38N4O6
    Pureza:98.07% - 99.45%
    Forma y color:Solid
    Peso molecular:646.73
  • CaMKP Inhibitor

    CAS:
    <p>CaMKP Inhibitor can inhibit CaMKP.</p>
    Fórmula:C10H8NNaO7S2
    Pureza:96.55% - 99.98%
    Forma y color:Solid
    Peso molecular:341.28
  • γ-Mangostin

    CAS:
    <p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>
    Fórmula:C23H24O6
    Pureza:98.55% - 99.08%
    Forma y color:Solid
    Peso molecular:396.43
  • 4-Acetamidobutanoic acid

    CAS:
    <p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>
    Fórmula:C6H11NO3
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:145.16
  • VUF 10166

    CAS:
    <p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>
    Fórmula:C13H15ClN4
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:262.74
  • NS9283

    CAS:
    <p>NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.</p>
    Fórmula:C14H8N4O
    Pureza:99.12%
    Forma y color:Solid
    Peso molecular:248.24
  • SR 57227 hydrochloride

    CAS:
    <p>SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.</p>
    Fórmula:C10H14ClN3·HCl
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:248.15
  • Amyloid β-Protein 10-20 acetate


    <p>Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research of</p>
    Fórmula:C73H103N17O18
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:1506.65
  • Lu AF21934

    CAS:
    <p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>
    Fórmula:C14H16Cl2N2O2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:315.2
  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Fórmula:C15H13F2NO4S
    Pureza:97.98%
    Forma y color:Solid
    Peso molecular:341.33
  • Nemifitide acetate(173240-15-8 free base)


    <p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>
    Fórmula:C35H47FN10O8
    Pureza:97.97%
    Forma y color:Solid
    Peso molecular:754.85
  • pyridostigmine

    CAS:
    <p>Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.</p>
    Fórmula:C9H13N2O2
    Pureza:98.10%
    Forma y color:Solid
    Peso molecular:181.21
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Fórmula:C12H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:207.23
  • lumateperone Tosylate

    CAS:
    <p>lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.</p>
    Fórmula:C31H36FN3O4S
    Pureza:95.83% - 99.95%
    Forma y color:Solid
    Peso molecular:565.7
  • Dasotraline hydrochloride

    CAS:
    <p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>
    Fórmula:C16H16Cl3N
    Pureza:98.92% - 99.6%
    Forma y color:Solid
    Peso molecular:328.66
  • Sarpogrelate

    CAS:
    <p>Sarpogrelate (MCI-9042), an oral 5-HT2 antagonist, boosts platelet aggregation and aids in studying Buerger's disease.</p>
    Fórmula:C24H31NO6
    Forma y color:Solid
    Peso molecular:429.51
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Fórmula:C20H30N2O3S2
    Pureza:99.70%
    Forma y color:White To Off-White Solid
    Peso molecular:410.59
  • GNE-7915 tosylate

    CAS:
    <p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>
    Fórmula:C26H29F4N5O6S
    Forma y color:Solid
    Peso molecular:615.6
  • CX516

    CAS:
    <p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>
    Fórmula:C14H15N3O
    Pureza:99.04% - ≥95%
    Forma y color:Tan Solid
    Peso molecular:241.29
  • Xanthotoxol

    CAS:
    <p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>
    Fórmula:C11H6O4
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:202.16
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Fórmula:C15H17N3O3
    Forma y color:Solid
    Peso molecular:287.31
  • 4F 4PP oxalate

    CAS:
    <p>4F 4PP oxalate is a 5-HT2A antagonist.</p>
    Fórmula:C22H26FNO·C2H2O4
    Pureza:97.34%
    Forma y color:Solid
    Peso molecular:429.49
  • (S)-Amisulpride

    CAS:
    <p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>
    Fórmula:C17H27N3O4S
    Pureza:98.38%
    Forma y color:Solid
    Peso molecular:369.48
  • PHA 543613 hydrochloride

    CAS:
    <p>PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.</p>
    Fórmula:C15H18ClN3O2
    Forma y color:Solid
    Peso molecular:307.78
  • TCN238

    CAS:
    <p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>
    Fórmula:C12H11N3
    Pureza:99.9% - 99.92%
    Forma y color:Solid
    Peso molecular:197.24
  • KN-92 hydrochloride

    CAS:
    <p>KN-92 hydrochloride is an inactive derivative of KN-93.</p>
    Fórmula:C24H26Cl2N2O3S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:493.45
  • Chelidamic acid

    CAS:
    <p>Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.</p>
    Fórmula:C7H5NO5
    Pureza:98.11%
    Forma y color:Pale Yellow Powder
    Peso molecular:183.12
  • GNE0877

    CAS:
    <p>GNE0877 (GNE 0877) is a highly effective and specific leucine-rich repeat kinase 2 (LRRK2) inhibitor (Ki: 0.7 nM).</p>
    Fórmula:C14H16F3N7
    Pureza:98.01% - 99.97%
    Forma y color:Solid
    Peso molecular:339.32
  • Alprenolol hydrochloride

    CAS:
    <p>Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.</p>
    Fórmula:C15H24ClNO2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:285.81
  • Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Fórmula:C13H15N3
    Forma y color:Solid
    Peso molecular:213.28
  • pep2-SVKI acetate


    <p>Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.</p>
    Fórmula:C62H97N13O20
    Pureza:97.14%
    Forma y color:Solid
    Peso molecular:1344.51
  • Tinoridine hydrochloride

    CAS:
    <p>Tinoridine HCl is an NSAID that inhibits lipid peroxides and renin release, unlike indomethacin and corticosteroids.</p>
    Fórmula:C17H21ClN2O2S
    Pureza:97.49%
    Forma y color:Solid
    Peso molecular:352.88
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Fórmula:C4H10N2
    Forma y color:Solid
    Peso molecular:86.14
  • m-Chlorophenylbiguanide hydrochloride

    CAS:
    <p>m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.</p>
    Fórmula:C8H11Cl2N5
    Pureza:99.43% - 99.87%
    Forma y color:Solid
    Peso molecular:248.11
  • lavendustin C

    CAS:
    <p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>
    Fórmula:C14H13NO5
    Pureza:98.06%
    Forma y color:Yellow To Tan Powder
    Peso molecular:275.26
  • CALP2 acetate(261969-04-4 free base)


    <p>CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM.</p>
    Fórmula:C68H104N14O13S
    Pureza:97.43%
    Forma y color:Solid
    Peso molecular:1357.7
  • TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Fórmula:C23H23F3N2O4
    Pureza:99.66% - ≥95%
    Forma y color:Solid
    Peso molecular:448.43
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Fórmula:C19H19FN4O2
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:354.38
  • Baclofen hydrochloride

    CAS:
    <p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:250.122
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Forma y color:Solid
    Peso molecular:248.75
  • PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Fórmula:C16H12N4S
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:292.36
  • MK 212 hydrochloride

    CAS:
    <p>MK 212 hydrochloride is a 5-HT2C receptor agonist</p>
    Fórmula:C8H11ClN4·HCl
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:235.12
  • SB 242084 dihydrochloride

    CAS:
    <p>SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.</p>
    Fórmula:C21H21Cl3N4O2
    Forma y color:Solid
    Peso molecular:467.78
  • Acamprosate

    CAS:
    <p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C5H11NO4S
    Pureza:98.30%
    Forma y color:Solid
    Peso molecular:181.21
  • Naratriptan hydrochloride

    CAS:
    <p>Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.</p>
    Fórmula:C17H25N3O2S·HCl
    Pureza:99.17% - 99.93%
    Forma y color:Beige Solid
    Peso molecular:371.93
  • PBD-150

    CAS:
    <p>PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)</p>
    Fórmula:C15H20N4O2S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:320.41
  • Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Fórmula:C22H25ClN4O4S2
    Forma y color:Solid
    Peso molecular:509.04
  • γ-secretase modulator 1 hydrochloride

    CAS:
    <p>gamma-secretase inhibitior-1 is a gamma-secretase modulator that is useful to Alzheimer's disease [1].</p>
    Fórmula:C24H25ClN4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:453
  • Lerisetron

    CAS:
    <p>Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.</p>
    Fórmula:C18H20N4
    Pureza:99.15% - 99.82%
    Forma y color:Solid
    Peso molecular:292.38
  • pep2-EVKI acetate(1315378-67-6 free base)


    <p>Pep2-EVKI acetate, a cell-permeable peptide, disrupts PICK1-GluR2 AMPA receptor binding.</p>
    Fórmula:C64H99N13O21
    Pureza:97.63%
    Forma y color:Solid
    Peso molecular:1386.55
  • Basmisanil

    CAS:
    <p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>
    Fórmula:C21H20FN3O5S
    Pureza:99.21% - 99.42%
    Forma y color:Solid
    Peso molecular:445.46
  • PF-06454589

    CAS:
    <p>PF-06454589 is a potent inhibitor of LRRK2.</p>
    Fórmula:C14H16N6O
    Pureza:99.06%
    Forma y color:Solid
    Peso molecular:284.32
  • AZ 11645373

    CAS:
    <p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>
    Fórmula:C24H21N3O5S
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:463.51
  • Imidafenacin

    CAS:
    <p>Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.</p>
    Fórmula:C20H21N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:319.4
  • Dihydroergotoxine mesylate

    CAS:
    <p>Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.</p>
    Fórmula:C20H29N3O5S
    Pureza:99.39% - ≥95%
    Forma y color:Solid
    Peso molecular:423.53
  • Aminooxyacetic acid hemihydrochloride

    CAS:
    <p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>
    Fórmula:C2H5NO3·5HCl
    Pureza:98.03%
    Forma y color:Light Beige Crystalline Powder
    Peso molecular:109.3
  • Indophagolin

    CAS:
    <p>Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.</p>
    Fórmula:C19H15BrClF3N2O3S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:523.75
  • A-740003

    CAS:
    <p>A-740003 is a potent P2X7 receptor blocker, inhibiting rat/human receptors (IC50: 18/40 nM), lessens pain in animals, and shrinks mouse neuroblastoma.</p>
    Fórmula:C26H30N6O3
    Pureza:96.53% - 99.68%
    Forma y color:Solid
    Peso molecular:474.55
  • Prifinium bromide

    CAS:
    <p>Prifinium bromide is a quaternary ammon antimuscarinic. It inhibits hyperkinesia of the digestive organs and urinary tract and has a spasmolytic action.</p>
    Fórmula:C22H28BrN
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:386.37
  • Vortioxetine

    CAS:
    <p>Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.</p>
    Fórmula:C18H22N2S
    Pureza:99.34% - 99.34%
    Forma y color:Solid
    Peso molecular:298.45
  • S26131

    CAS:
    <p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>
    Fórmula:C31H34N2O4
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:498.61
  • Metadoxine

    CAS:
    <p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>
    Fórmula:C8H11NO3·C5H7NO3
    Pureza:99.19%
    Forma y color:Off-White Powder
    Peso molecular:298.29
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:256.73
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C8H4N4O6
    Pureza:97.27% - 99.1%
    Forma y color:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14
  • VU-1545

    CAS:
    <p>VU-1545 is mGlu5 positive allosteric modulator.</p>
    Fórmula:C22H15FN4O3
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:402.38
  • Pitofenone hydrochloride

    CAS:
    <p>Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and</p>
    Fórmula:C22H26ClNO4
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:403.9
  • Syk Inhibitor II dihydrochloride dihydrate

    CAS:
    <p>Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.</p>
    Fórmula:C14H21Cl2F3N6O3
    Forma y color:Solid
    Peso molecular:449.26
  • TAE-1

    CAS:
    <p>TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.</p>
    Fórmula:C39H51I3N6O9
    Pureza:94.58%
    Forma y color:Solid
    Peso molecular:1128.57
  • 1,1'-Methylenedi-2-naphthol

    CAS:
    <p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>
    Fórmula:C21H16O2
    Pureza:98.91%
    Forma y color:Light Pink To Light Brown Crystalline Powder
    Peso molecular:300.35
  • Saclofen

    CAS:
    <p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>
    Fórmula:C9H12ClNO3S
    Pureza:99.17%
    Forma y color:White Crystalline Solid
    Peso molecular:249.71
  • Acotiamide

    CAS:
    <p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>
    Fórmula:C21H30N4O5S
    Forma y color:Solid
    Peso molecular:450.55
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Fórmula:C14H25Cl2N3O3
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:354.27
  • PE859

    CAS:
    <p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>
    Fórmula:C28H24N4O2
    Pureza:98.8% - 99.09%
    Forma y color:Solid
    Peso molecular:448.52
  • Loreclezole

    CAS:
    <p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>
    Fórmula:C10H6Cl3N3
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:274.53
  • NH125

    CAS:
    <p>NH125 is a selective eEF-2 kinase inhibitor with IC50 of 60 nM, &gt;125-fold selectivity over PKC, PKA, and CaMKII, and also a potent histidine kinase inhibitor.</p>
    Fórmula:C27H45IN2
    Pureza:98.60%
    Forma y color:Solid
    Peso molecular:524.56
  • Risperidone hydrochloride

    CAS:
    <p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>
    Fórmula:C23H28ClFN4O2
    Forma y color:Solid
    Peso molecular:446.95
  • Aftin-4

    CAS:
    <p>Aftin-4, an amyloid forty-two inducer, activates γ-secretase, promoting the generation of amyloid-β-1-42 (Aβ1-42) from amyloid-β protein precursor.</p>
    Fórmula:C20H28N6O
    Pureza:98.51%
    Forma y color:Solid
    Peso molecular:368.48
  • 6-Aminonicotinic acid

    CAS:
    <p>6-Aminonicotinic acid is a natural product.</p>
    Fórmula:C6H6N2O2
    Pureza:99.94%
    Forma y color:Soild
    Peso molecular:138.1238
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Forma y color:Solid
    Peso molecular:415.53
  • Cinanserin

    CAS:
    <p>Cinanserin is a serotonin 5-HT2 antagonist.</p>
    Fórmula:C20H24N2OS
    Forma y color:Solid
    Peso molecular:340.48
  • RU 24969 succinate

    CAS:
    <p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>
    Fórmula:C18H22N2O5
    Forma y color:Solid
    Peso molecular:346.38
  • Azeliragon HCl

    CAS:
    <p>Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.</p>
    Fórmula:C32H40Cl3N3O2
    Forma y color:Solid
    Peso molecular:605.04
  • Ondansetron hydrochloride

    CAS:
    <p>Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiation</p>
    Fórmula:C18H19N3O·HCl
    Pureza:99.78%
    Forma y color:White Powder
    Peso molecular:329.82
  • Succinylcholine Chloride Dihydrate

    CAS:
    <p>Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.</p>
    Fórmula:C14H30N2O4·2Cl·2H2O
    Pureza:99.87%
    Forma y color:White Solid
    Peso molecular:397.34
  • Piperidolate hydrochloride

    CAS:
    <p>Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.</p>
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:359.89
  • ZL006

    CAS:
    <p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>
    Fórmula:C14H11Cl2NO4
    Pureza:98.29%
    Forma y color:Solid
    Peso molecular:328.15
  • PNU-282987

    CAS:
    <p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>
    Fórmula:C14H18Cl2N2O
    Pureza:99% - >99.99%
    Forma y color:Solid
    Peso molecular:301.21
  • Alosetron (Hydrochloride(1:X))

    CAS:
    <p>Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.</p>
    Fórmula:C17H18ClN4O
    Forma y color:Solid
    Peso molecular:329.11691
  • trans-ACPD

    CAS:
    <p>trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.</p>
    Fórmula:C7H11NO4
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:173.17
  • Melitracen hydrochloride

    CAS:
    <p>Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.</p>
    Fórmula:C21H26ClN
    Pureza:99.99%
    Forma y color:Crystalline Solid
    Peso molecular:327.90
  • MTEP hydrochloride

    CAS:
    <p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>
    Fórmula:C11H9ClN2S
    Pureza:99.58%
    Forma y color:Solid
    Peso molecular:236.72
  • Acotiamide hydrochloride

    CAS:
    <p>Acotiamide hydrochloride, an oral AChE inhibitor (IC50: 1.79 μM), boosts gastric movement and treats functional dyspepsia.</p>
    Fórmula:C21H31ClN4O5S
    Forma y color:Solid
    Peso molecular:487.01
  • Quipazine maleate

    CAS:
    <p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>
    Fórmula:C17H19N3O4
    Forma y color:Solid
    Peso molecular:329.36
  • Caroverine hydrochloride

    CAS:
    <p>Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.</p>
    Fórmula:C22H28ClN3O2
    Pureza:98.37% - 98.75%
    Forma y color:Solid
    Peso molecular:401.9
  • Eslicarbazepine Acetate

    CAS:
    <p>Eslicarbazepine Acetate (Zebinix) is an anticonvulsant medication approved for use as an adjunctive therapy for partial-onset seizures.</p>
    Fórmula:C17H16N2O3
    Pureza:99.58% - >99.99%
    Forma y color:White To Off-White Solid
    Peso molecular:296.32
  • CaM kinase II inhibitor TFA salt


    <p>CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>
    Fórmula:C66H117F3N22O21
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1611.77
  • S 14506 HCl

    CAS:
    <p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), &lt;6.0 (5-HT3).</p>
    Fórmula:C24H26FN3O2
    Forma y color:Solid
    Peso molecular:407.48
  • Nor-benzetimide

    CAS:
    <p>Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.</p>
    Fórmula:C16H20N2O2
    Pureza:98.63%
    Forma y color:Solid
    Peso molecular:272.34
  • Eltoprazine dihydrochloride

    CAS:
    <p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>
    Fórmula:C12H18Cl2N2O2
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:293.19
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:477.57
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Fórmula:C19H25NOS
    Pureza:98.08% - 99.59%
    Forma y color:Solid
    Peso molecular:315.47
  • CaMKII-IN-1

    CAS:
    <p>CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM).</p>
    Fórmula:C29H30ClN5O2S
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:548.1
  • BRL-15572 dihydrochloride

    CAS:
    <p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:479.87
  • Arecaidine hydrochloride

    CAS:
    <p>Arecaidine hydrochloride may have carcinogenesis.</p>
    Fórmula:C7H12ClNO2
    Pureza:99.69% - ≥95%
    Forma y color:Solid
    Peso molecular:177.63
  • Mofezolac

    CAS:
    <p>Mofezolac (formerly known as Disopain or N-22) is a highly selective COX-1 (cyclooxygenase-1) inhibitor with COXs selectivity index &gt; 6000</p>
    Fórmula:C19H17NO5
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:339.34
  • Duloxetine

    CAS:
    <p>Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.</p>
    Fórmula:C18H19NOS
    Pureza:99.71% - 99.89%
    Forma y color:Solid
    Peso molecular:297.41
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Fórmula:C20H25N3O2
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:339.43
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Fórmula:C21H30N4O4
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:402.49
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Fórmula:C21H29Cl2N3O4S
    Pureza:98.5%
    Forma y color:Solid
    Peso molecular:490.44
  • Syn-Ake acetate

    CAS:
    <p>Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.</p>
    Fórmula:C19H29N5O3·2(C2H4O2)
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:495.58
  • Trihexyphenidyl hydrochloride

    CAS:
    <p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>
    Fórmula:C20H32ClNO
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:337.927
  • CNQX

    CAS:
    <p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C9H4N4O4
    Pureza:99.70%
    Forma y color:Pale Yellow Solid
    Peso molecular:232.15
  • (-)-Securinine

    CAS:
    <p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>
    Fórmula:C13H15NO2
    Pureza:99.58% - 99.87%
    Forma y color:Solid
    Peso molecular:217.26
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Fórmula:C19H26ClNOS
    Pureza:99.53% - 99.56%
    Forma y color:Almost White To White Crystalline Powder
    Peso molecular:351.93
  • Harmine hydrochloride

    CAS:
    <p>Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.</p>
    Fórmula:C13H13ClN2O
    Pureza:99.61% - >99.99%
    Forma y color:Yellow To Slightly Green Crystalline Powder
    Peso molecular:248.71
  • Afloqualone

    CAS:
    <p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>
    Fórmula:C16H14FN3O
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:283.3
  • Darifenacin

    CAS:
    <p>Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.</p>
    Fórmula:C28H30N2O2
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:426.55
  • Ethyl (triphenylphosphoranylidene) acetate

    CAS:
    <p>Ethyl (triphenylphosphoranylidene) acetate ((Carbethoxymethylene)triphenylphosphorane) may act as an cholinesterase inhibitor that inhibits AChE and BChE.</p>
    Fórmula:C22H21O2P
    Pureza:97.985%
    Forma y color:White Or Slight Yellow Powder
    Peso molecular:348.37
  • Sarpogrelate hydrochloride

    CAS:
    <p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>
    Fórmula:C24H32ClNO6
    Pureza:99.73%
    Forma y color:Colorless Liquid
    Peso molecular:465.97