
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 993 productos de "Receptor 5-HT"
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SC 53116 Hydrochloride
CAS:SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.Fórmula:C16H23Cl2N3O2Forma y color:SolidPeso molecular:360.28Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Fórmula:C22H31N5Forma y color:SolidPeso molecular:365.52SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Fórmula:C18H28N2O3SPureza:98%Forma y color:SolidPeso molecular:352.49Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Fórmula:C19H28N2Pureza:99.54%Forma y color:SolidPeso molecular:284.44EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Fórmula:C15H22N2OPureza:97.66% - 99.78%Forma y color:SolidPeso molecular:246.35Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Forma y color:SolidPeso molecular:328.385-HT7 agonist 1
CAS:<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Fórmula:C19H20ClN3Pureza:98.61%Forma y color:SolidPeso molecular:325.84Eptapirone fumarate
CAS:Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.Fórmula:C20H27N7O6Forma y color:SolidPeso molecular:461.479Ziprasidone mesylate trihydrate
CAS:<p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>Fórmula:C22H31ClN4O7S2Forma y color:SolidPeso molecular:563.08Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Fórmula:C23H28N2O5SForma y color:SolidPeso molecular:444.546CP94253 hydrochloride
CAS:<p>CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).</p>Fórmula:C15H20ClN3OPureza:99.78%Forma y color:SolidPeso molecular:293.79Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Fórmula:C23H30ClN3O2S2Forma y color:SolidPeso molecular:480.084-Chloro Trazodone hydrochloride
CAS:4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Fórmula:C19H23Cl2N5OForma y color:SolidPeso molecular:408.32Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Fórmula:C23H29ClN2OForma y color:SolidPeso molecular:384.95VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Fórmula:C11H15BrN2Pureza:98%Forma y color:SolidPeso molecular:255.15Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Fórmula:C27H41ClN4O5Forma y color:SolidPeso molecular:537.09Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C19H26ClN3O2S2Forma y color:SolidPeso molecular:428.01Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Fórmula:C26H32N2O7Forma y color:SolidPeso molecular:484.549Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Fórmula:C16H17BrN2Pureza:98%Forma y color:SolidPeso molecular:317.22AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Fórmula:C20H18N2O3SForma y color:SolidPeso molecular:366.43
