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Receptor 5-HT

Receptor 5-HT

Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.

Se han encontrado 993 productos de "Receptor 5-HT"

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  • Alaproclate

    CAS:
    <p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>
    Fórmula:C13H18ClNO2
    Pureza:98.29% - 98.64%
    Forma y color:Solid
    Peso molecular:255.74
  • E55888

    CAS:
    <p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>
    Fórmula:C16H23N3
    Forma y color:Solid
    Peso molecular:257.37
  • FR260010

    CAS:
    FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.
    Fórmula:C22H19N5
    Forma y color:Solid
    Peso molecular:353.42
  • CJ 033466

    CAS:
    <p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>
    Fórmula:C19H28ClN5O
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:377.91
  • Zicronapine

    CAS:
    Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.
    Fórmula:C22H27ClN2
    Forma y color:Solid
    Peso molecular:354.92
  • SUN-C5174

    CAS:
    <p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>
    Fórmula:C22H29FN4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:400.49
  • WAY 161503 hydrochloride

    CAS:
    WAY 161503 hydrochloride is a 5-HT2C receptor agonist.
    Fórmula:C11H12Cl3N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:308.59
  • SB 207710

    CAS:
    SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.
    Fórmula:C19H27IN2O4
    Forma y color:Solid
    Peso molecular:474.33
  • (Rac)-SEP-363856

    CAS:
    (Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique
    Fórmula:C9H13NOS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:183.27
  • SGS518 oxalate

    CAS:
    SGS518 oxalate is a 5-HT6 antagonist.
    Fórmula:C23H24F2N2O7S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:510.51
  • LY314228

    CAS:
    <p>LY314228 is an antagonist of 5-HT2A receptor.</p>
    Fórmula:C20H24N4O3
    Forma y color:Solid
    Peso molecular:368.43
  • ATC0065 HCl

    CAS:
    ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.
    Fórmula:C25H31BrCl2F3N5O
    Forma y color:Solid
    Peso molecular:625.35
  • (R)-DOI hydrochloride

    CAS:
    (R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.
    Fórmula:C11H17ClINO2
    Pureza:99.88% - >99.99%
    Forma y color:Solid
    Peso molecular:357.62
  • GR-55562 dihydrobromide

    CAS:
    GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.
    Fórmula:C23H26ClN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:411.93
  • S 14506 hydrochloride

    CAS:
    <p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>
    Fórmula:C24H27ClFN3O2
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:443.94
  • Lidanserin

    CAS:
    Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.
    Fórmula:C26H31FN2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.53
  • Fonazine

    CAS:
    Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.
    Fórmula:C19H25N3O2S2
    Forma y color:Solid
    Peso molecular:391.55
  • S-15535

    CAS:
    S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.
    Fórmula:C21H24N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:336.43
  • PF-184298

    CAS:
    PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.
    Fórmula:C15H20Cl2N2O
    Pureza:98.67%
    Forma y color:Solid
    Peso molecular:315.24
  • PNU-96391

    CAS:
    <p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>
    Fórmula:C15H23NO2S
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:281.41