
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 993 productos de "Receptor 5-HT"
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Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Forma y color:SolidPeso molecular:255.74E55888
CAS:<p>E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.</p>Fórmula:C16H23N3Forma y color:SolidPeso molecular:257.37FR260010
CAS:FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.Fórmula:C22H19N5Forma y color:SolidPeso molecular:353.42CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Fórmula:C19H28ClN5OPureza:99.72%Forma y color:SolidPeso molecular:377.91Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Fórmula:C22H27ClN2Forma y color:SolidPeso molecular:354.92SUN-C5174
CAS:<p>"SUN-C5174 is a selective 5-HT2 antagonist with pA2=8.98; inhibits platelet aggregation and reduces thromboembolic death in mice at ≥0.3 mg/kg."</p>Fórmula:C22H29FN4O2Pureza:98%Forma y color:SolidPeso molecular:400.49WAY 161503 hydrochloride
CAS:WAY 161503 hydrochloride is a 5-HT2C receptor agonist.Fórmula:C11H12Cl3N3OPureza:98%Forma y color:SolidPeso molecular:308.59SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Fórmula:C19H27IN2O4Forma y color:SolidPeso molecular:474.33(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFórmula:C9H13NOSPureza:98%Forma y color:SolidPeso molecular:183.27SGS518 oxalate
CAS:SGS518 oxalate is a 5-HT6 antagonist.Fórmula:C23H24F2N2O7SPureza:98%Forma y color:SolidPeso molecular:510.51LY314228
CAS:<p>LY314228 is an antagonist of 5-HT2A receptor.</p>Fórmula:C20H24N4O3Forma y color:SolidPeso molecular:368.43ATC0065 HCl
CAS:ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.Fórmula:C25H31BrCl2F3N5OForma y color:SolidPeso molecular:625.35(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Fórmula:C11H17ClINO2Pureza:99.88% - >99.99%Forma y color:SolidPeso molecular:357.62GR-55562 dihydrobromide
CAS:GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.Fórmula:C23H26ClN3O2Pureza:98%Forma y color:SolidPeso molecular:411.93S 14506 hydrochloride
CAS:<p>S 14506 hydrochloride is a 5-HT1A receptor full agonist.</p>Fórmula:C24H27ClFN3O2Pureza:99.92%Forma y color:SolidPeso molecular:443.94Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Fórmula:C26H31FN2O4Pureza:98%Forma y color:SolidPeso molecular:454.53Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Fórmula:C19H25N3O2S2Forma y color:SolidPeso molecular:391.55S-15535
CAS:S-15535 is a potent, orally active, partial 5-HT1A receptor agonist.Fórmula:C21H24N2O2Pureza:98%Forma y color:SolidPeso molecular:336.43PF-184298
CAS:PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Fórmula:C15H20Cl2N2OPureza:98.67%Forma y color:SolidPeso molecular:315.24PNU-96391
CAS:<p>PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.</p>Fórmula:C15H23NO2SPureza:99.53%Forma y color:SolidPeso molecular:281.41
