
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 1003 productos de "Receptor 5-HT"
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Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Fórmula:C23H29ClN2OForma y color:SolidPeso molecular:384.95VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Fórmula:C11H15BrN2Pureza:98%Forma y color:SolidPeso molecular:255.15BGC 20-761
CAS:BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.Fórmula:C19H22N2OForma y color:SolidPeso molecular:294.39Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C19H26ClN3O2S2Forma y color:SolidPeso molecular:428.01Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Fórmula:C16H17BrN2Pureza:98%Forma y color:SolidPeso molecular:317.22GSK-215083
CAS:GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.Fórmula:C20H20FN3O2SForma y color:SolidPeso molecular:385.46F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Fórmula:C26H29ClF2N4O4SForma y color:SolidPeso molecular:567.05VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Fórmula:C19H27KN3O3SPureza:98%Forma y color:SolidPeso molecular:416.6mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Fórmula:C8H10ClN5Forma y color:SolidPeso molecular:211.65p-MPPF dihydrochloride
CAS:p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.Fórmula:C25H29Cl2FN4O2Pureza:99.55%Forma y color:SolidPeso molecular:507.43Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Fórmula:C20H24N2S2Forma y color:SolidPeso molecular:356.55Fonazine mesylate
CAS:Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Fórmula:C20H29N3O5S3Forma y color:SolidPeso molecular:487.65AVN-101 free base
CAS:AVN-101: potent 5-HT7 antagonist, also targets 5-HT6, 5-HT2A, 5-HT2C. Aims to treat CNS disorders.Fórmula:C21H24N2Forma y color:SolidPeso molecular:304.43AS19
CAS:<p>AS19 is a potent, selective 5-HT7 receptor agonist (IC50: 0.83 nM; Ki: 0.6 nM).</p>Fórmula:C18H25N3Pureza:98%Forma y color:SolidPeso molecular:283.41Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Fórmula:C22H23Cl2N3OSForma y color:SolidPeso molecular:448.41L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Fórmula:C20H21N5O3SPureza:98.36%Forma y color:White SolidPeso molecular:411.48Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFórmula:C25H36N4O10Pureza:98%Forma y color:SolidPeso molecular:552.581WAY 629
CAS:WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.Fórmula:C15H18N2Forma y color:SolidPeso molecular:226.32Way 100289
CAS:Way 100289 is a selective 5-HT3 receptor antagonist.Fórmula:C20H27N3O3Forma y color:SolidPeso molecular:357.45Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Fórmula:C21H29N5O2Pureza:99.91% - 99.91%Forma y color:SolidPeso molecular:383.49
