
Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 942 productos de "Receptor 5-HT"
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Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Fórmula:C22H27ClN2Forma y color:SolidPeso molecular:354.92EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Fórmula:C24H31N3O2Pureza:95.64% - 99.39%Forma y color:SolidPeso molecular:393.522PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Fórmula:C17H21N3Pureza:98%Forma y color:SolidPeso molecular:267.37FR260010
CAS:<p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>Fórmula:C22H19N5Forma y color:SolidPeso molecular:353.42TC-2153
CAS:<p>TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.</p>Fórmula:C7H5ClF3NS5Forma y color:SolidPeso molecular:355.89Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Fórmula:C13H18ClNO2Pureza:98.29% - 98.64%Forma y color:SolidPeso molecular:255.74LP44 hydrochloride
CAS:<p>LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.</p>Fórmula:C27H38ClN3OSPureza:98.06%Forma y color:SolidPeso molecular:488.13Belaperidone
CAS:<p>Belaperidone, an antipsychotic, resembles clozapine, binds D(4) and 5-HT(2A) receptors, minimally extends Q-T without causing arrhythmias.</p>Fórmula:C22H22FN3O2Forma y color:SolidPeso molecular:379.43CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Fórmula:C12H14ClN3OPureza:98%Forma y color:SolidPeso molecular:251.71CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Fórmula:C25H25F3N4O8Pureza:98%Forma y color:SolidPeso molecular:566.485-HT6/5-HT2A receptor ligand-2
CAS:<p>Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.</p>Fórmula:C20H18FN3O2Forma y color:SolidPeso molecular:351.37CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Fórmula:C19H21N5O2Pureza:98%Forma y color:SolidPeso molecular:351.45-HT7 agonist 2
CAS:<p>Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.</p>Fórmula:C23H29N3OForma y color:SolidPeso molecular:363.5Prucalopride hydrochloride
CAS:<p>Prucalopride hydrochloride is a selective agonist of the 5-HT4.</p>Fórmula:C18H27Cl2N3O3Pureza:98%Forma y color:SolidPeso molecular:404.33WAY208466 dihydrochloride
CAS:<p>WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.</p>Fórmula:C17H20Cl2FN3O2SPureza:98.43%Forma y color:SolidPeso molecular:420.33LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Fórmula:C19H23FN4Pureza:98%Forma y color:SolidPeso molecular:326.41UCSF686
CAS:<p>UCSF686, a UCSF678 analog, lacks 5-HT5A potency but keeps affinity for 5-HT1A, 5-HT2B, 5-HT7, and serves as a control.</p>Fórmula:C14H19N3O2SForma y color:SolidPeso molecular:293.38ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Fórmula:C25H29BrF3N5OForma y color:SolidPeso molecular:552.43ZM 169369
CAS:<p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>Fórmula:C19H20N2SForma y color:SolidPeso molecular:308.44(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Fórmula:C16H26BrNOPureza:98%Forma y color:SolidPeso molecular:328.29
