Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 942 productos de "Receptor 5-HT"
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FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Fórmula:C27H29F2N3O2Pureza:98%Forma y color:SolidPeso molecular:465.53S 14063
CAS:<p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>Fórmula:C22H29Cl2N3O2SForma y color:SolidPeso molecular:470.45Tertatolol
CAS:<p>Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.</p>Fórmula:C16H25NO2SPureza:98%Forma y color:SolidPeso molecular:295.44Piclozotan
CAS:<p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>Fórmula:C23H24ClN3O2Pureza:98.59%Forma y color:SolidPeso molecular:409.91Alniditan
CAS:<p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>Fórmula:C17H26N4OPureza:98%Forma y color:SolidPeso molecular:302.415-HT2A receptor agonist-2
CAS:<p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>Fórmula:C20H21ClN2O3Forma y color:SolidPeso molecular:372.85AP-521 (Free base)
CAS:<p>AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.</p>Fórmula:C20H18N2O3SForma y color:SolidPeso molecular:366.43Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Fórmula:C26H32N2O7Forma y color:SolidPeso molecular:484.549RS 39604
CAS:<p>potent and selective 5-HT4 antagonist</p>Fórmula:C26H37Cl2N3O6SPureza:98%Forma y color:SolidPeso molecular:590.56Naronapride
CAS:<p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>Fórmula:C27H41ClN4O5Forma y color:SolidPeso molecular:537.09Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Fórmula:C24H23N3O2Pureza:98%Forma y color:SolidPeso molecular:385.46TMPPAA
CAS:<p>TMPPAA is an allosteric agonist of 5-HT3 receptor.</p>Fórmula:C15H21NO2Pureza:98%Forma y color:SolidPeso molecular:247.33Ziprasidone mesylate trihydrate
CAS:<p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>Fórmula:C22H31ClN4O7S2Forma y color:SolidPeso molecular:563.085-HT7 agonist 1
CAS:<p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>Fórmula:C19H20ClN3Pureza:98.61%Forma y color:SolidPeso molecular:325.84Pruvanserin hydrochloride
CAS:<p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>Fórmula:C22H22ClFN4OPureza:99.6%Forma y color:SolidPeso molecular:412.89Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Fórmula:C19H21FN2O2Pureza:97.04%Forma y color:SolidPeso molecular:328.38SB-737050A
CAS:<p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>Fórmula:C22H23ClN2O3S2Forma y color:SolidPeso molecular:463.01EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Fórmula:C15H22N2OPureza:97.66% - 99.78%Forma y color:SolidPeso molecular:246.35GR 113808
CAS:<p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>Fórmula:C19H27N3O4SPureza:98.16%Forma y color:SolidPeso molecular:393.5PNU-142633
CAS:<p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.</p>Fórmula:C24H30N4O3Pureza:98%Forma y color:SolidPeso molecular:422.52
