Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 942 productos de "Receptor 5-HT"
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SB228357
CAS:<p>SB228357 is a potent and selective antagonist of the 5-HT receptor with pKis of 6.9, 8.0, and 9.0 for 5-HT2A, 5-HT2B, and 5-HT2C, respectively.</p>Fórmula:C22H17F4N3O2Pureza:99.82%Forma y color:SolidPeso molecular:431.38Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Fórmula:C14H20ClN3O3Pureza:99.51%Forma y color:SolidPeso molecular:313.785HT6-ligand-1
CAS:<p>5HT6-ligand-1 is an orally active ligand of 5-HT6 receptor (Ki = 1.43 nM).</p>Fórmula:C20H22BrN3O2SPureza:99.24% - 99.93%Forma y color:SolidPeso molecular:448.38SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Fórmula:C23H31Cl2NO8SPureza:99.37%Forma y color:SolidPeso molecular:552.47LY-2624803
CAS:<p>LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.</p>Fórmula:C22H25N3O3Pureza:99.78% - 99.97%Forma y color:SolidPeso molecular:379.45Roxindole
CAS:<p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>Fórmula:C23H26N2OPureza:98.03% - 98.93%Forma y color:SolidPeso molecular:346.47Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Forma y color:SolidPeso molecular:426.42Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Fórmula:C24H40N2O3Pureza:97.87% - >99.99%Forma y color:SolidPeso molecular:404.59ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Fórmula:C23H26ClF2N5OPureza:99.98%Forma y color:SolidPeso molecular:461.93Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Fórmula:C21H28Cl3N3OSPureza:99.67%Forma y color:SolidPeso molecular:476.89Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Fórmula:C24H22N4Pureza:99.91%Forma y color:SolidPeso molecular:366.46Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Fórmula:C21H24BrN3O3SPureza:98.36% - 99.65%Forma y color:SolidPeso molecular:478.4Teniloxazine
CAS:<p>Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.</p>Fórmula:C16H19NO2SPureza:99.23%Forma y color:SolidPeso molecular:289.39Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Fórmula:C17H16N2O4Pureza:99.89%Forma y color:SolidPeso molecular:312.32H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Fórmula:C11H15Cl2N3O2SPureza:97.3%Forma y color:SolidPeso molecular:324.235-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Fórmula:C22H20FN3O3Pureza:98.78% - 99.26%Forma y color:SolidPeso molecular:393.41Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Fórmula:C16H19NOPureza:99.47%Forma y color:SolidPeso molecular:241.33BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Fórmula:C18H23ClF2N4OPureza:99.97%Forma y color:SolidPeso molecular:384.85Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Fórmula:C24H32N4O2SPureza:99.74%Forma y color:SolidPeso molecular:440.65-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Fórmula:C21H25N3O2SPureza:99.68%Forma y color:SolidPeso molecular:383.51
