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Receptor 5-HT

Receptor 5-HT

Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.

Se han encontrado 939 productos de "Receptor 5-HT"

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  • Nemonapride

    CAS:
    <p>Nemonapride is a dopamine D2-like receptor antagonist.</p>
    Fórmula:C21H26ClN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:387.9
  • Gepirone

    CAS:
    <p>Gepirone is a 5-HT1A receptor agonist belonging to the buspirone family. Gepirone HCl possesses greater selectivity for the 5-HT1A receptor than SSRIs.</p>
    Fórmula:C19H29N5O2
    Pureza:99.35% - 99.89%
    Forma y color:Solid
    Peso molecular:359.47
  • SB 258719

    CAS:
    <p>SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.</p>
    Fórmula:C18H30N2O2S
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:338.51
  • LY-426965

    CAS:
    <p>LY-426965 is a selective, potent, orally bioavailable 5-HT1A antagonist.</p>
    Fórmula:C28H38N2O2
    Forma y color:Solid
    Peso molecular:434.61
  • LY 53857

    CAS:
    <p>LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.</p>
    Fórmula:C27H36N2O7
    Forma y color:Solid
    Peso molecular:500.592
  • FPPQ

    CAS:
    <p>FPPQ blocks 5-HT3 and 5-HT6 receptors (Ki: 0.9 &amp; 3 nM) and may improve psychosis and cognition.</p>
    Fórmula:C21H19FN4O2S
    Forma y color:Solid
    Peso molecular:410.46
  • NAS181

    CAS:
    <p>rat 5-HT1B receptor antagonist</p>
    Fórmula:C21H34N2O10S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:538.63
  • R-96544

    CAS:
    <p>R-96544 is an orally active antagonist of the 5-HT2A receptor that has demonstrated the ability to inhibit platelet aggregation in vitro [1].</p>
    Fórmula:C22H30ClNO3
    Forma y color:Solid
    Peso molecular:391.93
  • 5-HT3 antagonist 1

    CAS:
    <p>5-HT3 antagonist 1 is a potent and selective antagonist of 5-HT3 receptor.</p>
    Fórmula:C22H27N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:377.48
  • PNU109291

    CAS:
    <p>PNU109291, a potent and selective agonist of the 5-HT1D receptor, effectively mitigates dural plasma extravasation induced by trigeminal ganglion stimulation.</p>
    Fórmula:C24H31N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:409.52
  • 5-HT2A receptor agonist-3

    CAS:
    <p>5-HT2A receptor agonist-3 represents the highest selectivity for the human 5-HT2A receptor currently identified, exhibiting a K i of 2.5 nM.</p>
    Fórmula:C21H26BrNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.34
  • (±)-Fabesetron hydrochloride

    CAS:
    <p>FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.</p>
    Fórmula:C18H20ClN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:329.82
  • Facinicline hydrochloride

    CAS:
    <p>Facinicline hydrochloride (RG3487) is both a novel nicotinic alpha-7 receptor (alpha7nAChR) partial agonist (Ki = 6 nM) and an antagonist of 5-HT3(Ki = 1.2 nM).</p>
    Fórmula:C15H19ClN4O
    Pureza:98.70%
    Forma y color:Solid
    Peso molecular:306.79
  • Flesinoxan

    CAS:
    <p>Flesinoxan is a hypotensive agent and is an effective, high affinity, and selective 5-hydroxytryptamine1A receptor agonist (EC50: 24 nM).</p>
    Fórmula:C22H26FN3O4
    Forma y color:Solid
    Peso molecular:415.46
  • GR 125487 sulfamate

    CAS:
    <p>GR 125487 sulfamate is a 5-HT4 receptor antagonist.</p>
    Fórmula:C19H29FN4O8S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:524.58
  • 4-Chloro-L-phenylalanine

    CAS:
    <p>4-Chloro-L-phenalanine (L-PCPA) is an inhibitor of 5-HT biosynthesis and a non-specific antagonist of tryptophan hydroxylases (TPH1 and TPH2).</p>
    Fórmula:C9H10ClNO2
    Pureza:99.76% - 99.96%
    Forma y color:Solid
    Peso molecular:199.63
  • Capeserod HCl

    CAS:
    <p>Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.</p>
    Fórmula:C23H26Cl2N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:493.38
  • YM348

    CAS:
    <p>YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).</p>
    Fórmula:C14H17N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:243.3
  • L-772,405

    CAS:
    <p>L-772,405 is a highly selective agonists of h5-HT(1D) receptor.</p>
    Fórmula:C26H31FN6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:462.56
  • DU-125530

    CAS:
    <p>DU-125530 is a 5-HT1A receptor antagonist.</p>
    Fórmula:C23H26ClN3O5S
    Forma y color:Solid
    Peso molecular:491.99