Receptor 5-HT
Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.
Se han encontrado 940 productos de "Receptor 5-HT"
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R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Fórmula:C27H27ClFN3OSPureza:97.7%Forma y color:SolidPeso molecular:496.04RS 42358-197
CAS:<p>RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.</p>Fórmula:C19H23ClN2OPureza:99.70%Forma y color:SolidPeso molecular:330.85DA-6886
CAS:<p>DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.</p>Fórmula:C19H28Cl2N6O2Pureza:99.28% - 99.91%Forma y color:SolidPeso molecular:443.37Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Fórmula:C24H24FN3O2Pureza:99.83%Forma y color:SolidPeso molecular:405.46Femoxetine hydrochloride
CAS:<p>Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.</p>Fórmula:C20H26ClNO2Pureza:99.63%Forma y color:SolidPeso molecular:347.88Cyamemazine
CAS:<p>Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.</p>Fórmula:C19H21N3SPureza:97.01%Forma y color:SolidPeso molecular:323.46Masupirdine free base
CAS:<p>Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.</p>Fórmula:C21H24BrN3O3SPureza:98.36% - 99.65%Forma y color:SolidPeso molecular:478.4Landipirdine
CAS:<p>Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.</p>Fórmula:C18H19FN2O3SPureza:97.61% - 99.37%Forma y color:SolidPeso molecular:362.42Faxeladol
CAS:<p>Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.</p>Fórmula:C15H23NOPureza:98.09% - 98.77%Forma y color:SolidPeso molecular:233.35Tedatioxetine
CAS:<p>Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.</p>Fórmula:C18H21NSPureza:99.76% - >99.99%Forma y color:SolidPeso molecular:283.43Cianopramine
CAS:<p>Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.</p>Fórmula:C20H23N3Pureza:99.92% - 99.92%Forma y color:SolidPeso molecular:305.42BL-1020 Mesylate
CAS:<p>BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.</p>Fórmula:C28H45ClN4O11S4Pureza:>99.99%Forma y color:SolidPeso molecular:777.39Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Fórmula:C13H19NO3Pureza:99.67%Forma y color:SolidPeso molecular:237.29CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Fórmula:C29H21FN4OSPureza:97.81% - 99.62%Forma y color:SoildPeso molecular:492.57Cilansetron
CAS:<p>Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.</p>Fórmula:C20H21N3OPureza:99.82% - 99.98%Forma y color:SolidPeso molecular:319.4E6801
CAS:<p>E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.</p>Fórmula:C17H18ClN5O2S2Pureza:96.32% - 99.53%Forma y color:SolidPeso molecular:423.94Ticalopride
CAS:<p>Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.</p>Fórmula:C14H20ClN3O3Pureza:99.51%Forma y color:SolidPeso molecular:313.78SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Fórmula:C23H31Cl2NO8SPureza:99.37%Forma y color:SolidPeso molecular:552.47Roxindole
CAS:<p>Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.</p>Fórmula:C23H26N2OPureza:98.03% - 98.93%Forma y color:SolidPeso molecular:346.47Aplindore Fumarate
CAS:<p>Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.</p>Fórmula:C22H22N2O7Pureza:>99.99%Forma y color:SolidPeso molecular:426.42Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Fórmula:C24H40N2O3Pureza:97.87% - >99.99%Forma y color:SolidPeso molecular:404.59ATC 0175 hydrochloride
CAS:<p>ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.</p>Fórmula:C23H26ClF2N5OPureza:99.98%Forma y color:SolidPeso molecular:461.93Perphenazine dihydrochloride
CAS:<p>Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.</p>Fórmula:C21H28Cl3N3OSPureza:99.67%Forma y color:SolidPeso molecular:476.89Liafensine
CAS:<p>Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.</p>Fórmula:C24H22N4Pureza:99.91%Forma y color:SolidPeso molecular:366.46Piromelatine
CAS:<p>Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity with</p>Fórmula:C17H16N2O4Pureza:99.89%Forma y color:SolidPeso molecular:312.32Litoxetine
CAS:<p>Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.</p>Fórmula:C16H19NOPureza:99.47%Forma y color:SolidPeso molecular:241.33Lensiprazine
CAS:<p>Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and</p>Fórmula:C24H27FN4O2Pureza:98.04%Forma y color:SolidPeso molecular:422.5H-9 dihydrochloride
CAS:<p>H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.</p>Fórmula:C11H15Cl2N3O2SPureza:97.3%Forma y color:SolidPeso molecular:324.235-HT6/7 antagonist 1
CAS:<p>5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.</p>Fórmula:C22H20FN3O3Pureza:98.78% - 99.26%Forma y color:SolidPeso molecular:393.41BMY-14802 hydrochloride
CAS:<p>BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.</p>Fórmula:C18H23ClF2N4OPureza:99.97%Forma y color:SolidPeso molecular:384.85Tiospirone
CAS:<p>Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.</p>Fórmula:C24H32N4O2SPureza:99.74%Forma y color:SolidPeso molecular:440.65-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Fórmula:C21H25N3O2SPureza:99.68%Forma y color:SolidPeso molecular:383.51Pimethixene maleate
CAS:<p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>Fórmula:C23H23NO4SPureza:99.55%Forma y color:SolidPeso molecular:409.5Ecopipam
CAS:<p>Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.</p>Fórmula:C19H20ClNOPureza:99.68%Forma y color:SolidPeso molecular:313.82Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Fórmula:C10H14Cl2N2SPureza:>99.99% - >99.99%Forma y color:SolidPeso molecular:265.20Ricasetron
CAS:<p>Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.</p>Fórmula:C19H27N3OPureza:99.52%Forma y color:SolidPeso molecular:313.44Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Fórmula:C22H20ClN3Pureza:97.76% - 99.20%Forma y color:SolidPeso molecular:361.87Sarizotan HCl
CAS:<p>Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.</p>Fórmula:C22H22ClFN2OPureza:96%Forma y color:SolidPeso molecular:384.87Agomelatine hydrochloride
CAS:<p>Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).</p>Fórmula:C15H18ClNO2Pureza:99.57%Forma y color:SolidPeso molecular:279.76Fananserin
CAS:<p>Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).</p>Fórmula:C23H24FN3O2SPureza:99.88%Forma y color:SolidPeso molecular:425.52Repinotan
CAS:<p>Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.</p>Fórmula:C21H24N2O4SPureza:99%Forma y color:SolidPeso molecular:400.49cis-Urocanic acid
CAS:<p>cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).</p>Fórmula:C6H6N2O2Pureza:99.81%Forma y color:SolidPeso molecular:138.12LY 272015 hydrochloride
CAS:<p>LY 272015 hydrochloride is a 5-HT2B receptor antagonist.</p>Fórmula:C21H25ClN2O2Pureza:99.47%Forma y color:SolidPeso molecular:372.89Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Fórmula:C26H32N2O5Pureza:99.17% - 99.67%Forma y color:SolidPeso molecular:452.54Quinupramine
CAS:<p>Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.</p>Fórmula:C21H24N2Pureza:99.77%Forma y color:SolidPeso molecular:304.43ADR-851 free base
CAS:<p>ADR-851 free base is an antagonist of the HT3 receptor.</p>Fórmula:C14H18ClN3O2Pureza:97.88% - 98.39%Forma y color:SolidPeso molecular:295.77ML 10302 hydrochloride
CAS:<p>ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.</p>Fórmula:C15H22Cl2N2O3Pureza:99.99%Forma y color:SolidPeso molecular:349.25LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Fórmula:C21H24Cl2N2O2Pureza:98.58%Forma y color:SolidPeso molecular:407.338-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Fórmula:C16H25NOPureza:98%Forma y color:SolidPeso molecular:247.38SB 699551 dihydrochloride
CAS:<p>SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.</p>Fórmula:C34H47Cl2N3OPureza:99.83%Forma y color:SolidPeso molecular:584.66
